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US 4,005,208 AGranted
N-Heterocyclic-9-xanthenylamines
AssigneeSmithKline Corporation
InventorsPaul E. Bender, Bernard Loev
Life of this patent
Estimating the term…
Abstract
The compounds are N-piperidinyl and pyrrolidinyl-9-xanthenylamines which are inhibitors of gastric acid secretion.
Claims6
A compound of the formula:
- ##STR3## in which:
- R.sub.1 is hydrogen, halogen, hydroxy, lower alkyl or lower alkoxy;
- R.sub.2 is hydrogen, halogen, lower alkyl or lower alkoxy;
- R.sub.3 is hydrogen or lower alkyl;
- R.sub.4 is hydrogen, lower alkyl, allyl, propargyl, cycloalkyl having 3 to 6 carbon atoms, lower alkanoyl, lower alkoxycarbonyl, carbamoyl, N-lower alkylcarbamoyl, N,N-di- lower alkylcarbamoyl, phenyl or benzyl;
- m is 1 or 2 and n is 2 or 3, the sum of m and n being 3 or 4
- or a pharmaceutically acceptable acid addition salt thereof.
4 more elements
Dependencies are inferred from the claim text.