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US 2026/0297029 A1Published application
Alkoxy and carbamoyl quaternary amine salts as prodrugs of tryptamines
OwnerAlan GIBBS, Tanweer KHAN +2inventors
InventorsAlan GIBBS, Tanweer KHAN, Robert B PERNI, Glenn SHORT
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Abstract
Pharmaceutical compounds with potential for treating mental health disorders which overcome solubility and oral bioavailability issues to act as (partial) agonists of the CNS serotonin receptor, 5-HT2A.
Claims44
A compound having the structure of Formula (I):
- wherein:
- L is a counter ion;
- X, Y, and Z are independently hydrogen, deuterium, OR1, CO2R1, or NR1R2;
- W is NR1, OR1, or CR1R2;
- M is a CR5R6R7, OR5, or NR5R6;
- and
- R1, R2, R4, R5, R6 and R7 are independently hydrogen, deuterium, alkyl, cycloalkyl, heteroatom substituted and halogen substituted alkyl or cycloalkyl, aromatic, or heteroaromatic.
4 more elements
Dependencies are inferred from the claim text.