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US 2023/0339876 A1Published application
Process for preparing aminofuranes
AssigneeBayer Aktiengesellschaft
InventorsSergii PAZENOK, Winfried ETZEL
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Abstract
The present invention relates to a novel method for preparing 4-aminofurans of the general formula (I) and salts thereof.
Claims11
A method for preparing a compound of formula (I) and/or salt thereof,
- in which
- R1 is CF3, CF2H, C2F5, CF2Cl, CCl3, COO(C1-C4)alkyl, COOH,
- R2 is H, CH3CO, CCl3CO, CF3CO, phenyl-CO, CH3OCO, (CH3)3COCO, phenyl, phenyl-CH2, (diphenyl)CH,
- Comprising converting a compound of formula (II)
- in which
- R3 and R4 are each independently H and C1-C4-alkyl
- and
- R1 has the definitions specified above,
- with aid of an amine of formula R5-NH2 (V) to a compound of formula (III)
- in which
- R5 is H, phenyl, phenyl-CH2, (diphenyl)CH,
- and then reacting said compound of formula III in presence of a dehydrating reagent to give a compound of formula (I).
9 more elements
Dependencies are inferred from the claim text.