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US 2022/0015364 A1Published application
Microbiocidal quinoline (thio)carboxamide derivatives
AssigneeSyngenta Participations AG
InventorsMatthias WEISS, Laura QUARANTA, Farhan BOU HAMDAN
Life of this patent
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Abstract
Compounds of the formula (I) wherein the substituents are as defined in claim 1. Furthermore, the present invention relates to agrochemical compositions which comprise compounds of formula (I), to preparation of these compositions, and to the use of the compounds or compositions in agriculture or horticulture for combating, preventing or controlling infestation of plants, harvested food crops, seeds or non-living materials by phytopathogenic microorganisms, in particular fungi.
Claims18
A compound of formula (I)
- wherein
- X is O or S;
- R1 is hydrogen, halogen, methyl or cyano;
- R2 and R3 are each independently selected from hydrogen, halogen, methoxy and methyl;
- R4 is hydrogen, C1-C4 alkyl, C1-C2 haloakyl, C2-C4 alkenyl or C3-C6 cycloalkyl, wherein the alkyl, alkenyl and cycloalkyl may be optionally substituted with 1 to 3 substituents independently selected from halogen, cyano, C1-C3 alkyl, C1-C3 alkoxy and C1-C3 alkylthio;
- R5 is hydrogen, cyano or C1-C4 alkyl;
- R6 is C1-C5 alkyl, C3-C7 cycloalkyl, C3-C5 alkenyl, C3-C6 cycloalkenyl, C3-C5 alkynyl, a C5-C10 saturated or partially unsaturated bicyclic carbocycle, aryl, aryl(C1-C4)alkyl, a saturated or partially unsaturated heterocycle or heteroaryl, wherein the alkyl, cycloalkyl, alkenyl, cycloalkenyl, carbocycle, alkynyl, may be optionally substituted with one or more substituents independently selected from halogen, cyano, C1-C3 alkyl, C1-C3 alkoxy, C1-C3 alkylthio, C1-C3 haloalkoxy, C1-C3 haloalkylthio, C3-C5 cycloalkyl or phenyl, and wherein the aryl, heterocycle or heteroaryl may be optionally substituted with one or more substituents independently selected from halogen, cyano, C1-C3 alkyl, C1-C3 alkoxy, C1-C3 alkylthio, C1-C3 haloalkoxy, C1-C3 haloalkylthio or C3-C5 cycloalkyl;
- and
- R11 is hydrogen, methyl or halogen;
- or a salt, enantiomer or N-oxide thereof.
7 more elements
A compound selected from the group consisting of:
- N-[1-(2,2-dimethylpropoxymethyl)-3,3,3-trifluoro-1-methyl-propyl]-8-fluoro-quinoline-3-carboxamide;
- 8-chloro-N-[1-[(3,3-dimethylcyclobutoxy)methyl]-3,3,3-trifluoro-1-methyl-propyl]quinoline-3-carboxamide;
- N-[1-[(4,4-difluorocyclohexoxy)methyl]-3,3,3-trifluoro-1-methyl-propyl]-8-fluoro-quinoline-3-carboxamide;
- N-[1-[(3,3-dimethylcyclobutoxy)methyl]-3,3,3-trifluoro-1-methyl-propyl]-8-fluoro-quinoline-3-carboxamide;
- N-[1-[(4-chlorophenoxy)methyl]-3,3,3-trifluoro-1-methyl-propyl]-8-fluoro-quinoline-3-carboxamide;
- N-[1-(cyclopropylmethoxymethyl)-1,3,3-trimethyl-butyl]-8-fluoro-quinoline-3-carboxamide;
- N-[1-(cyclobutoxymethyl)-3,3,3-trifluoro-1-methyl-propyl]-8-fluoro-4-methyl-quinoline-3-carboxamide;
- N-[1-(cyclobutoxymethyl)-3,3,3-trifluoro-1-methyl-propyl]-7,8-difluoro-quinoline-3-carboxamide;
- N-[1-(cyclobutoxymethyl)-3,3,3-trifluoro-1-methyl-propyl]-8-fluoro-2-methyl-quinoline-3-carboxamide;
- 8-fluoro-N-[3,3,3-trifluoro-1-methyl-1-[(1-methylcyclopentoxy)methyl]propyl]quinoline-3-carboxamide;
- N-[1-(cyclobutoxymethyl)-3,3,3-trifluoro-1-methyl-propyl]-8-methyl-quinoline-3-carboxamide;
- 8-chloro-N-[1-(cyclobutoxymethyl)-3,3,3-trifluoro-1-methyl-propyl]quinoline-3-carboxamide;
- N-[(1S)-1-(cyclobutoxymethyl)-3,3,3-trifluoro-1-methyl-propyl]-8-fluoro-quinoline-3-carboxamide;
- N-[(1S)-1-(cyclobutoxymethyl)-3,3,3-trifluoro-1-methyl-propyl]-8-fluoro-quinoline-3-carboxamide;
- 8-fluoro-N-[3,3,3-trifluoro-1-methyl-1-[(1-methylcyclohexoxy)methyl]propyl]quinoline-3-carboxamide;
- N-[(1R)-1-(cyclohexoxymethyl)-3,3,3-trifluoro-1-methyl-propyl]-8-fluoro-quinoline-3-carboxamide;
- N-[(1S)-1-(cyclohexoxymethyl)-3,3,3-trifluoro-1-methyl-propyl]-8-fluoro-quinoline-3-carboxamide;
- N-[1-(benzyloxymethyl)-1-methyl-2-(1-methylcyclopropyl)ethyl]-8-fluoro-quinoline-3-carboxamide;
- 8-fluoro-N-[3,3,3-trifluoro-1-methyl-1-(phenoxymethyl)propyl]quinoline-3-carboxamide;
- N-[1,3-dimethyl-1-(2-methylallyloxymethyl)butyl]-8-fluoro-quinoline-3-carboxamide;
- N-[1-(cyclobutoxymethyl)-3,3,3-trifluoro-1-methyl-propyl]-8-fluoro-quinoline-3-carboxamide;
- N-[1-(1-ethylpropoxymethyl)-1,3-dimethyl-butyl]-8-fluoro-quinoline-3-carboxamide;
- N-[1-(cyclobutoxymethyl)-1,3-dimethyl-butyl]-8-fluoro-quinoline-3-carboxamide;
- 8-fluoro-N-[1-(isopropoxymethyl)-1,3-dimethyl-butyl]quinoline-3-carboxamide;
- 8-fluoro-N-[1-(isobutoxymethyl)-1,3-dimethyl-butyl]quinoline-3-carboxamide;
- N-[1-(cycloheptoxymethyl)-3,3,3-trifluoro-1-methyl-propyl]-8-fluoro-quinoline-3-carboxamide;
- N-[1-(cyclohexoxymethyl)-3,3,3-trifluoro-1-methyl-propyl]-8-fluoro-quinoline-3-carboxamide;
- N-[1,3-dimethyl-1-(phenoxymethyl)butyl]-8-fluoro-quinoline-3-carboxamide;
- N-[1-(cyclohexoxymethyl)-1,3-dimethyl-butyl]-8-fluoro-quinoline-3-carboxamide;
- N-[1-(benzyloxymethyl)-1,3-dimethyl-butyl]-8-fluoro-quinoline-3-carboxamide;
- N-[1-(cyclopentoxymethyl)-1,3-dimethyl-butyl]-8-fluoro-quinoline-3-carboxamide;
- 8-fluoro-N-[1-(methoxymethyl)-1,3-dimethyl-butyl]quinoline-3-carboxamide;
- and
- 8-fluoro-N-[1-(methoxymethyl)-1-methyl-nonyl]quinoline-3-carboxamide.
31 more elements
Dependencies are inferred from the claim text.