Novel triazole derivatives
AssigneesBayer CropScience AG, Bayer Aktiengesellschaft
InventorsRicarda MILLER, Pierre-Yves COQUERON, David BERNIER, Sebastien NAUD, Pierre GENIX, Philippe KENNEL, Stephane BRUNET
Life of this patent
Estimating the term…
Abstract
The present invention relates to novel triazole derivatives of formula to processes for preparing these compounds, to certain intermediates, to compositions comprising these compounds, and to the use thereof as biologically active compounds, especially for control of harmful microorganisms in crop protection and in the protection of materials and as plant growth regulators.
Claims20
A triazole derivative of formula (I)
- wherein
- R1 represents hydrogen, C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C8-cycloalkyl, C3-C8-cycloalkyl-C1-C4-alkyl, phenyl, phenyl-C1-C4-alkyl, phenyl-C2-C4-alkenyl or phenyl-C2-C4-alkynyl,
- R2 represents hydrogen, C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C8-cycloalkyl, C3-C8-cycloalkyl-C1-C4-alkyl, phenyl, phenyl-C1-C4-alkyl, phenyl-C2-C4-alkenyl or phenyl-C2-C4-alkynyl,
- wherein the aliphatic moieties, excluding cycloalkyl moieties, of R1 and/or R2 may carry 1, 2, 3 or up to the maximum possible number of identical or different groups Ra which independently of one another are selected from halogen, CN, nitro, phenyl, C1-C4-alkoxy and C1-C4-halogenalkoxy, wherein the phenyl may be substituted by 1, 2, 3, 4 or 5 substituents selected independently from each other from halogen, CN, nitro, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-halogenalkyl, C1-C4-halogenalkoxy,
- and wherein the cycloalkyl and/or phenyl moieties of R1 and/or R2 may carry 1, 2, 3, 4, 5 or up to the maximum number of identical or different groups Rb which independently of one another are selected from halogen, CN, nitro, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-halogenalkyl and C1-C4-halogenalkoxy;
- each R4 represents independently of one another C3-C6-cycloalkyl, C3-C6-halogencycloalkyl, C1-C4-alkyl-C3-C6-cycloalkyl, C2-C6-alkenyl, C2-C6-halogenalkenyl, C2-C6-alkynyl, C2-C6-halogenalkynyl, C1-C4-alkylsulfanyl, C1-C4-halogenalkylsulfanyl, C1-C6-alkylsulfonyl, C6-C10-arylsulfonyl, C1-C6-alkyl-SO2NH—, C6-C10-aryl-SO2NH—, formyl, 5-, 6- or 7-membered saturated heterocycloalkyl containing up to 4 heteroatoms selected from N, O and S, or —C(R4a)═N—OR4b, wherein R4a and R4b represent independently from each other hydrogen, C1-C6-alkyl or phenyl;
- m is an integer and is 1, 2, 3, 4 or 5;
- Y represents a 6-membered aromatic heterocycle containing 1 or 2 nitrogen atom(s) as heteroatom(s) selected from
- wherein Y is connected to the O of formula (I) via the bonds identified with “U” and Y is connected to the CR1(OR2) moiety of formula (I) via the bonds identified with “V” and
- wherein
- R represents hydrogen, C1-C2-halogenalkyl, C1-C2-halogenalkoxy, C1-C2-alkylcarbonyl or halogen;
- each R3 represents independently from each other halogen, CN, nitro, C1-C4-alkyl, C1-C4-halogenalkyl, C1-C4-alkoxy or C1-C4-halogenalkoxy;
- n is an integer and is 0 or 1;
- and/or a salt or N-oxide thereof.
A compound of formula (VII)
- wherein
- each R4 represents independently of one another C3-C6-cycloalkyl, C3-C6-halogencycloalkyl, C1-C4-alkyl-C3-C6-cycloalkyl, C2-C6-alkenyl, C2-C6-halogenalkenyl, C2-C6-alkynyl, C2-C6-halogenalkynyl, C1-C4-alkylsulfanyl, C1-C4-halogenalkylsulfanyl, C1-C6-alkylsulfonyl, C6-C10-arylsulfonyl, C1-C6-alkyl-SO2NH—, C6-C10-aryl-SO2NH—, formyl, 5-, 6- or 7-membered saturated heterocycloalkyl containing up to 4 heteroatoms selected from N, O and S, or —C(R4a)═N—OR4b, wherein R4a and R4b represent independently from each other hydrogen, C1-C6-alkyl or phenyl;
- m is an integer and is 1, 2, 3, 4 or 5;
- Y represents a 6-membered aromatic heterocycle containing 1 or 2 nitrogen atom(s) as heteroatom(s) selected from
- wherein Y is connected to the O of formula (VII) via the bonds identified with “U” and Y is connected to the C(O)CH2— moiety of formula (VII) via the bonds identified with “V” and
- wherein
- R represents hydrogen, C1-C2-halogenalkyl, C1-C2-halogenalkoxy, C1-C2-alkylcarbonyl or halogen;
- each R3 represents independently from each other halogen, CN, nitro, C1-C4-alkyl, C1-C4-halogenalkyl, C1-C4-alkoxy or C1-C4-halogenalkoxy;
- n is an integer and is 0 or 1;
- and/or a salt or N-oxide thereof.
(canceled)
(canceled)
(canceled)
(canceled)
(canceled)
(canceled)
(canceled)
(canceled)
Dependencies are inferred from the claim text.