US 2017/0304403 A1Published application

METHOD FOR INHIBITING INFLAMMATION and PRO-INFLAMMATORY CYTOKINE/CHEMOKINE EXPRESSION USING A GHRELIN ANALOGUE

AssigneeIpsen Pharma S.A.S.

InventorsZheng Xin DONG, John E. TAYLOR, Rakesh DATTA, Michael DeWitt CULLER

Life of this patent

Estimating the term…

Abstract

The present invention provides a method of ameliorating inflammation, inhibiting proinflammatory cytokine and/or chemokine expression and treating various diseases and/or conditions incidental to the onset of inflammation, in a subject in need of treatment for such conditions, by administering select analogues of native hGhrelin.

Claims4

Dependent claims

A method of limiting myocardial damage during an acute myocardial infarction in a subject in need thereof which comprises administering to said subject an effective amount of a peptidyl analogue of ghrelin, a prodrug thereof, or a pharmaceutically acceptable salt thereof wherein said analogue or said prodrug thereof is selected from the group consisting of:

(Dap3(octanesulfonyl))hGhrelin(1-28)-NH2;
(SEQ ID:
6)
(Aib2, A6c5)hGhrelin(1-28)-NH2;
(SEQ ID:
7)
(A6c5)hGhrelin(1-28)-NH2;
(SEQ ID:
8)
(Aib2,6)hGhrelin(1-28)-NH2;
(SEQ ID:
9)
(Aib2, A5c12)hGhrelin(1-28)-NH2;
(SEQ ID:
10)
(Aib2, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
11)
(Aib2, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
12)
(Aib2, Act6)hGhrelin(1-28)-NH2;
(SEQ ID:
9)
(Aib2, 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
13)
(Aib2, Dmt7)hGhrelin(1-28)-NH2;
(SEQ ID:
14)
(Aib2, Thz7)hGhrelin(1-28)-NH2;
(SEQ ID:
14)
(A5c2)hGhrelin(1-28)-NH2;
(SEQ ID:
15)
(Act2)hGhrelin(1-28)-NH2;
(SEQ ID:
15)
(Aib2, A5c5)hGhrelin(1-28)-NH2;
(SEQ ID:
7)
(Aib2, A6c5)hGhrelin(1-28)-NH2;
(SEQ ID:
7)
(Aib2,5)hGhrelin(1-28)-NH2;
(SEQ ID:
7)
(Aib2, hLeu5)hGhrelin(1-28)-NH2;
(SEQ ID:
7)
(Aib2, Cha5)hGhrelin(1-28)-NH2;
(SEQ ID:
7)
(Aib2,6)hGhrelin(1-28)-NH2;
(SEQ ID:
9)
(Aib2,Act6)hGhrelin(1-28)-NH2;
(SEQ ID:
9)
(Aib2, Thr6)hGhrelin(1-28)-NH2;
(SEQ ID:
9)
(Aib2, Abu6)hGhrelin(1-28)-NH2;
(SEQ ID:
9)
(Aib2, 4-Hyp7)hGhrelin(1-28)-NH2;
(SEQ ID:
14)
(Aib2,Thz7)hGhrelin(1-28)-NH2;
(SEQ ID:
14)
(Aib2, Pip7)hGhrelin(1-28)-NH2;
(SEQ ID:
14)
(Aib2, Dhp7)hGhrelin(1-28)-NH2;
(SEQ ID:
14)
(Aib2, Ktp7)hGhrelin(1-28)-NH2;
(SEQ ID:
14)
(Aib2,8)hGhrelin(1-28)-NH2;
(SEQ ID:
16)
(Aib2, 2-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
13)
(Aib2, 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
13)
(Aib2, 4-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
13)
(Aib2, Taz9)hGhrelin(1-28)-NH2;
(SEQ ID:
13)
(Aib2, 2-Thi9)hGhrelin(1-28)-NH2;
(SEQ ID:
13)
(Aib2, 2-Fua9)hGhrelin(1-28)-NH2;
(SEQ ID:
13)
(Aib2, Apc9)hGhrelin(1-28)-NH2;
(SEQ ID:
13)
(Aib2,9)hGhrelin(1-28)-NH2;
(SEQ ID:
13)
(Aib2,10)hGhrelin(1-28)-NH2;
(SEQ ID:
17)
(Aib2, Tic7)hGhrelin(1-28)-NH2;
(SEQ ID:
14)
(Aib6)hGhrelin(1-28)-NH2;
(SEQ ID:
18)
(A5c5)hGhrelin(1-28)-NH2;
(SEQ ID:
8)
(A6c5)hGhrelin(1-28)-NH2;
(SEQ ID:
8)
(Act6)hGhrelin(1-28)-NH2;
(SEQ ID:
18)
(3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
19)
(Dmt7)hGhrelin(1-28)-NH2;
(SEQ ID:
20)
(Thz7)hGhrelin(1-28)-NH2;
(SEQ ID:
20)
(Aib5)hGhrelin(1-28)-NH2;
(SEQ ID:
8)
(hLeu5)hGhrelin(1-28)-NH2;
(SEQ ID:
8)
(Cha5)hGhrelin(1-28)-NH2;
(SEQ ID:
8)
(Thr6)hGhrelin(1-28)-NH2;
(SEQ ID:
18)
(Abu6)hGhrelin(1-28)-NH2;
(SEQ ID:
18)
(4-Hyp7)hGhrelin(1-28)-NH2;
(SEQ ID:
20)
(Pip7)hGhrelin(1-28)-NH2;
(SEQ ID:
20)
(Dhp7)hGhrelin(1-28)-NH2;
(SEQ ID:
20)
(Ktp7)hGhrelin(1-28)-NH2;
(SEQ ID:
20)
(Aib8)hGhrelin(1-28)-NH2;
(SEQ ID:
21)
(2-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
19)
(4-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
19)
(Taz9)hGhrelin(1-28)-NH2;
(SEQ ID:
19)
(2-Thi9)hGhrelin(1-28)-NH2;
(SEQ ID:
19)
(2-Fua9)hGhrelin(1-28)-NH2;
(SEQ ID:
19)
(Apc9)hGhrelin(1-28)-NH2;
(SEQ ID:
19)
(Aib9)hGhrelin(1-28)-NH2;
(SEQ ID:
19)
(Aib10)hGhrelin(1-28)-NH2;
(SEQ ID:
22)
(Aib2, Dap3(octanesulfonyl), A6c5)hGhrelin(1-28)-NH2;
(SEQ ID:
23)
(Dap3(octanesulfonyl), A6c5)hGhrelin(1-28)-NH2;
(SEQ ID:
24)
(Aib2,6, Dap3(octanesulfonyl))hGhrelin(1-28)-NH2;
(SEQ ID:
25)
(Aib2, Dap3(octanesulfonyl), A5c12)hGhrelin(1-28)-NH2;
(SEQ ID:
26)
(Aib2, Dap3(octanesulfonyl), A5c12,Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
27)
(Aib2, Dap3(octanesulfonyl), A5c12,Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
28)
(Aib2, Dap3(octanesulfonyl), Act6)hGhrelin(1-28)-NH2;
(SEQ ID:
25)
(Aib2, Dap3(octanesulfonyl), 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
29)
(Aib2, Dap3(octanesulfonyl), Dmt7)hGhrelin(1-28)-NH2;
(SEQ ID:
30)
(Aib2, Dap3(octanesulfonyl), Thz7)hGhrelin(1-28)-NH2;
(SEQ ID:
30)
(A5c2, Dap3(octanesulfonyl))hGhrelin(1-28)-NH2;
(SEQ ID:
31)
(Acte, Dap3(octanesulfonyl))hGhrelin(1-28)-NH2;
(SEQ ID:
31)
(Aib2, Dap3(octanesulfonyl), A5c5)hGhrelin(1-28)-NH2;
(SEQ ID:
32)
(Aib2,5, Dap3(octanesulfonyl))hGhrelin(1-28)-NH2;
(SEQ ID:
32)
(Aib2, Dap3(octanesulfonyl), hLeu5)hGhrelin(1-28)-NH2;
(SEQ ID:
32)
(Aib2, Dap3(octanesulfonyl), Cha5)hGhrelin(1-28)-NH2;
(SEQ ID:
32)
(Aib2,6, Dap3(octanesulfonyl))hGhrelin(1-28)-NH2;
(SEQ ID:
25)
(Aib2, Dap3(octanesulfonyl), Thr6)hGhrelin(1-28)-NH2;
(SEQ ID:
25)
(Aib2, Dap3(octanesulfonyl), Abu6)hGhrelin(1-28)-NH2;
(SEQ ID:
25)
(Aib2, Dap3(octanesulfonyl), 4-Hyp7)hGhrelin(1-28)-NH2;
(SEQ ID:
30)
(Aib2, Dap3(octanesulfonyl), Pip7)hGhrelin(1-28)-NH2;
(SEQ ID:
30)
(Aib2, Dap3(octanesulfonyl), Dhp7)hGhrelin(1-28)-NH2;
(SEQ ID:
30)
(Aib2, Dap3(octanesulfonyl), Ktp7)hGhrelin(1-28)-NH2;
(SEQ ID:
30)
(Aib2,8, Dap3(octanesulfonyl))hGhrelin(1-28)-NH2;
(SEQ ID:
33)
(Aib2, Dap3(octanesulfonyl), 2-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
29)
(Aib2, Dap3(octanesulfonyl), 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
29)
(Aib2, Dap3(octanesulfonyl), 4-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
29)
(Aib2, Dap3(octanesulfonyl), Taz9)hGhrelin(1-28)-NH2;
(SEQ ID:
29)
(Aib2, Dap3(octanesulfonyl), 2-Thi9)hGhrelin(1-28)-NH2;
(SEQ ID:
29)
(Aib2, Dap3(octanesulfonyl), 2-Fua9)hGhrelin(1-28)-NH2;
(SEQ ID:
29)
(Aib2, Dap3(octanesulfonyl), Apc9)hGhrelin(1-28)-NH2;
(SEQ ID:
29)
(Aib2,9, Dap3(octanesulfonyl))hGhrelin(1-28)-NH2;
(SEQ ID:
29)
(Aib2,10, Dap3(octanesulfonyl))hGhrelin(1-28)-NH2;
(SEQ ID:
34)
(Dap3(octanesulfonyl), A6c5)hGhrelin(1-28)-NH2;
(SEQ ID:
24)
(Dap3(octanesulfonyl), Aib6)hGhrelin(1-28)-NH2;
(SEQ ID:
35)
(Dap3(octanesulfonyl), A5c12)hGhrelin(1-28)-NH2;
(SEQ ID:
36)
(Dap3(octanesulfonyl), A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
37)
(Dap3(octanesulfonyl), A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
38)
(Dap3(octanesulfonyl), Act6)hGhrelin(1-28)-NH2;
(SEQ ID:
35)
(Dap3(octanesulfonyl), 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
39)
(Dap3(octanesulfonyl), Dmt7)hGhrelin(1-28)-NH2;
(SEQ ID:
40)
(Dap3(octanesulfonyl), Thz7)hGhrelin(1-28)-NH2;
(SEQ ID:
40)
(Dap3(octanesulfonyl), A5c5)hGhrelin(1-28)-NH2;
(SEQ ID:
24)
(Dap3(octanesulfonyl), Aib5)hGhrelin(1-28)-NH2;
(SEQ ID:
24)
(Dap3(octanesulfonyl), hLeu5)hGhrelin(1-28)-NH2;
(SEQ ID:
24)
(Dap3(octanesulfonyl), Cha5)hGhrelin(1-28)-NH2;
(SEQ ID:
24)
(Dap3(octanesulfonyl), Thr6)hGhrelin(1-28)-NH2;
(SEQ ID:
35)
(Dap3(octanesulfonyl), Abu6)hGhrelin(1-28)-NH2;
(SEQ ID:
35)
(Dap3(octanesulfonyl), 4-Hyp7)hGhrelin(1-28)-NH2;
(SEQ ID:
40)
(Dap3(octanesulfonyl), Pip7)hGhrelin(1-28)-NH2;
(SEQ ID:
40)
(Dap3(octanesulfonyl), Dhp7)hGhrelin(1-28)-NH2;
(SEQ ID:
40)
(Dap3(octanesulfonyl), Ktp7)hGhrelin(1-28)-NH2;
(SEQ ID:
40)
(Dap3(octanesulfonyl), Aib8)hGhrelin(1-28)-NH2;
(SEQ ID:
41)
(Dap3(octanesulfonyl), 2-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
39)
(Dap3(octanesulfonyl), 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
39)
(Dap3(octanesulfonyl), 4-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
39)
(Dap3(octanesulfonyl), Taz9)hGhrelin(1-28)-NH2;
(SEQ ID:
39)
(Dap3(octanesulfonyl), 2-Thi9)hGhrelin(1-28)-NH2;
(SEQ ID:
39)
(Dap3(octanesulfonyl), 2-Fua9)hGhrelin(1-28)-NH2;
(SEQ ID:
39)
(Dap3(octanesulfonyl), Apc9)hGhrelin(1-28)-NH2;
(SEQ ID:
39)
(Dap3(octanesulfonyl), Aib9)hGhrelin(1-28)-NH2;
(SEQ ID:
39)
(Dap3(octanesulfonyl), Aib10hGhrelin(1-28)-NH2;
(SEQ ID:
42)
(Dap3(octanesulfonyl), A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
37)
(Dab3(octanesulfonyl), A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
37)
(Aib2, A6c5, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
43)
(A6c5, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
44)
(Aib2,6, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
45)
(Aib2, Actio, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
45)
(Aib2, 3-Pal9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
46)
(Aib2, Dmt7, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
47)
(Aib2, Thz7, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
47)
(Aib2, A5c5, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
43)
(Aib2,5, A5c12,Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
43)
(Aib2, hLeu5, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
43)
(Aib2, Cha5, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
43)
(Aib2,6, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
45)
(Aib2, Thr6, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
45)
(Aib2, Abu6, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
45)
(Aib2, 4-Hyp', A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
47)
(Aib2, Pip', A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
47)
(Aib2, Dhp7, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
47)
(Aib2, Ktp7, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
47)
(Aib2,8, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
48)
(Aib2, 2-Pal9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
46)
(Aib2, 3-Pal9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
46)
(Aib2, 4-Pal9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
46)
(Aib2, Taz9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
46)
(Aib2, 2-Thi9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
46)
(Aib2, 2-Fua9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
46)
(Aib2, Apc9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
46)
(Aib2,9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
46)
(Aib2,10, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
49)
(Dap3(octanesulfonyl), A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
38)
(Dab3(octanesulfonyl), A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
38)
(Aib2, A6c5, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
50)
(A6c5, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
51)
(Aib2,6, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
52)
(Aib2, Actio, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
52)
(Aib2, 3-Pal9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
53)
(Aib2, Dmt7, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
54)
(Aib2, Thz7, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
54)
(Aib2, A5c5,12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
50)
(Aib2,5, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
50)
(Aib2, hLeu5, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
50)
(Aib2, Cha5, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
50)
(Aib2,6, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
52)
(Aib2, Thr6, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
52)
(Aib2, Abu6, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
52)
(Aib2, 4-Hyp', A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
54)
(Aib2, Pip', A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
54)
(Aib2, Dhp7, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
54)
(Aib2, Ktp7, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
54)
(Aib2,8, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
55)
(Aib2, 2-Pal9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
53)
(Aib2, 3-Pal9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
53)
(Aib2, 4-Pal9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
53)
(Aib2, Taz9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
53)
(Aib2, 2-Thi9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
53)
(Aib2, 2-Fua9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
53)
(Aib2, Apc9,16, A5c12)hGhrelin(1-28)-NH2;
(SEQ ID:
53)
(Aib2,9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
53)
(Aib2,10, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
56)
(A6c5, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
44)
(Aib6, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
57)
(Act6, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
57)
(3-Pal9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
58)
(Dmt7, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
59)
(Thz7, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
59)
(A5c5,12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
44)
(Aib5, A5c12,Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
44)
(hLeu5, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
44)
(Cha5, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
44)
(Aib6, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
57)
(Thr6, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
57)
(Abu6, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
57)
(4-Hyp', A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
59)
(Pip7, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
59)
(Dhp7, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
59)
(Ktp7, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
59)
(Aib8, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
60)
(2-Pal9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
58)
(3-Pal9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
58)
(4-Pal9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
58)
(Taz9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
58)
(2-Thi9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
58)
(2-Fua9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
58)
(Apc9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
58)
(Aib9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
58)
(Aib10, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
61)
(Aib6, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
62)
(A5c5,12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
51)
(Actio, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
62)
(3-Pal9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
63)
(Dmt7, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
64)
(Thz7, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
64)
(Aib5, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
51)
(hLeu5, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
51)
(Cha5, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
51)
(Thr6, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
62)
(Abu6, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
62)
(4-Hyp A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
64)
(Pip7, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
64)
(Dhp7, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
64)
(Ktp7, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
64)
(Aib8, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
65)
(2-Pal9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
63)
(3-Pal9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
63)
(4-Pal9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
63)
(Taz9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
63)
(2-Thi9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
63)
(2-Fua9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
63)
(Apc9,16, A5c12)hGhrelin(1-28)-NH2;
(SEQ ID:
63)
(Aib9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
63)
(Aib10, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
66)
(Aib2, Glu3(NH-hexyl), A6c5)hGhrelin(1-28)-NH2;
(SEQ ID:
67)
(Glu3(NH-hexyl), A6c5)hGhrelin(1-28)-NH2;
(SEQ ID:
68)
(Aib2,6, Glu3(NH-hexyl))hGhrelin(1-28)-NH2;
(SEQ ID:
69)
(Aib2, Glu3(NH-hexyl), Act6)hGhrelin(1-28)-NH2;
(SEQ ID:
69)
(Aib2, Glu3(NH-hexyl), 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
70)
(Aib2, Glu3(NH-hexyl), Dmt7)hGhrelin(1-28)-NH2;
(SEQ ID:
71)
(Aib2, Glu3(NH-hexyl), Thz7)hGhrelin(1-28)-NH2;
(SEQ ID:
71)
(Aib2, Glu3(NH-hexyl), A5c5)hGhrelin(1-28)-NH2;
(SEQ ID:
67)
(Aib2,5, Glu3(NH-hexyl))hGhrelin(1-28)-NH2;
(SEQ ID:
67)
(Aib2, Glu3(NH-hexyl), hLeu5)hGhrelin(1-28)-NH2;
(SEQ ID:
67)
(Aib2, Cha5)hGhrelin(1-28)-NH2;
(SEQ ID:
7)
(Aib2′6, Glu3(NH-hexyl))hGhrelin(1-28)-NH2;
(SEQ ID:
69)
(Aib2, Glu3(NH-hexyl), Thr6)hGhrelin(1-28)-NH2;
(SEQ ID:
69)
(Aib2, Glu3(NH-hexyl), Abu6)hGhrelin(1-28)-NH2;
(SEQ ID:
69)
(Aib2, Glu3(NH-hexyl), 4-Hyp7)hGhrelin(1-28)-NH2;
(SEQ ID:
71)
(Aib2, Glu3(NH-hexyl), Pip7)hGhrelin(1-28)-NH2;
(SEQ ID:
71)
(Aib2, Glu3(NH-hexyl), Dhp7)hGhrelin(1-28)-NH2;
(SEQ ID:
71)
(Aib2, Glu3(NH-hexyl), Ktp7)hGhrelin(1-28)-NH2;
(SEQ ID:
71)
(Aib2,8, Glu3(NH-hexyl))hGhrelin(1-28)-NH2;
(SEQ ID:
72)
(Aib2, Glu3(NH-hexyl), 2-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
70)
(Aib2, Glu3(NH-hexyl), 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
70)
(Aib2, Glu3(NH-hexyl), 4-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
70)
(Aib2, Glu3(NH-hexyl), Taz9)hGhrelin(1-28)-NH2;
(SEQ ID:
70)
(Aib2, Glu3(NH-hexyl), 2-Thi9)hGhrelin(1-28)-NH2;
(SEQ ID:
70)
(Aib2, Glu3(NH-hexyl), 2-Fua9)hGhrelin(1-28)-NH2;
(SEQ ID:
70)
(Aib2, Glu3(NH-hexyl), Apc9)hGhrelin(1-28)-NH2;
(SEQ ID:
70)
(Aib2,9, Glu3(NH-hexyl))hGhrelin(1-28)-NH2;
(SEQ ID:
70)
(Aib2,10, Glu3(NH-hexyl))hGhrelin(1-28)-NH2;
(SEQ ID:
73)
(Glu3(NH-hexyl), Aib6)hGhrelin(1-28)-NH2;
(SEQ ID:
74)
(Glu3(NH-hexyl), A5c5)hGhrelin(1-28)-NH2;
(SEQ ID:
68)
(Glu3(NH-hexyl), Act6)hGhrelin(1-28)-NH2;
(SEQ ID:
74)
(Glu3(NH-hexyl), 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
75)
(Glu3(NH-hexyl), Dmt7)hGhrelin(1-28)-NH2;
(SEQ ID:
76)
(Glu3(NH-hexyl), Thz7)hGhrelin(1-28)-NH2;
(SEQ ID:
76)
(Glu3(NH-hexyl), Aib5)hGhrelin(1-28)-NH2;
(SEQ ID:
68)
(Glu3(NH-hexyl), hLeu5)hGhrelin(1-28)-NH2;
(SEQ ID:
68)
(Glu3(NH-hexyl), Cha5)hGhrelin(1-28)-NH2;
(SEQ ID:
68)
(Glu3(NH-hexyl), Thr6)hGhrelin(1-28)-NH2;
(SEQ ID:
74)
(Glu3(NH-hexyl), Abu6)hGhrelin(1-28)-NH2;
(SEQ ID:
74)
(Glu3(NH-hexyl), 4-Hyp7)hGhrelin(1-28)-NH2;
(SEQ ID:
76)
(Glu3(NH-hexyl), Pip7)hGhrelin(1-28)-NH2;
(SEQ ID:
76)
(Glu3(NH-hexyl), Dhp7)hGhrelin(1-28)-NH2;
(SEQ ID:
76)
(Glu3(NH-hexyl), Ktp7)hGhrelin(1-28)-NH2;
(SEQ ID:
76)
(Glu3(NH-hexyl), Aib8)hGhrelin(1-28)-NH2;
(SEQ ID:
41)
(Glu3(NH-hexyl), 2-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
75)
(Glu3(NH-hexyl), 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
75)
(Glu3(NH-hexyl), 4-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
75)
(Glu3(NH-hexyl), Taz9)hGhrelin(1-28)-NH2;
(SEQ ID:
75)
(Glu3(NH-hexyl), 2-Thi9)hGhrelin(1-28)-NH2;
(SEQ ID:
75)
(Glu3(NH-hexyl), 2-Fua9)hGhrelin(1-28)-NH2;
(SEQ ID:
75)
(Glu3(NH-hexyl), Apc9)hGhrelin(1-28)-NH2;
(SEQ ID:
75)
(Glu3(NH-hexyl), Aib9)hGhrelin(1-28)-NH2;
(SEQ ID:
75)
(Glu3(NH-hexyl), Aib9hGhrelin(1-28)-NH2;
(SEQ ID:
42)
(Aib2, Glu3(NH-hexyl), A6c5, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
77)
(A6c5, Glu3(NH-hexyl), A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
78)
(Aib2,6, Glu3(NH-hexyl), A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
79)
(Aib2, Glu3(NH-hexyl), Actio, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
79)
(Aib2, Glu3(NH-hexyl), 3-Pal9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
80)
(Aib2, Glu3(NH-hexyl), Dmt7, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
81)
(Aib2, Glu3(NH-hexyl), Thz7, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
81)
(Aib2, Glu3(NH-hexyl), A5c5,12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
77)
(Aib2,5, Glu3(NH-hexyl), A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
77)
(Aib2, hLeu5, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
43)
(Aib2, Glu3(NH-hexyl), Cha5, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
77)
(Aib2,6, Glu3(NH-hexyl), A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
79)
(Aib2, Glu3(NH-hexyl), Thr6, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
79)
(Aib2, Glu3(NH-hexyl), Abu6, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
79)
(Aib2, Glu3(NH-hexyl), 4-Hyp', A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
81)
(Aib2, Glu3(NH-hexyl), Pip', A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
81)
(Aib2, Glu3(NH-hexyl), Dhp7, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
81)
(Aib2, Glu3(NH-hexyl), Ktp7, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
81)
(Aib2,8, Glu3(NH-hexyl), A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
82)
(Aib2, Glu3(NH-hexyl), 2-Pal9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
80)
(Aib2, Glu3(NH-hexyl), 3-Pal9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
80)
(Aib2, Glu3(NH-hexyl), 4-Pal9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
80)
(Aib2, Glu3(NH-hexyl), Taz9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
80)
(Aib2, Glu3(NH-hexyl), 2-Thi9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
80)
(Aib2, Glu3(NH-hexyl), 2-Fua9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
80)
(Aib2, Glu3(NH-hexyl), Apc9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
80)
(Aib2,9, Glu3(NH-hexyl), A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
80)
(Aib2,12, Glu3(NH-hexyl), 4-Pal9, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
125)
(Aib2,10, Glu3(NH-hexyl), A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
83)
(Aib2, Glu3(NH-hexyl), A6c5, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
84)
(Glu3(NH-hexyl), A6c5, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
85)
(Aib2,6, Glu3(NH-hexyl), A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
86)
(Aib2, Glu3(NH-hexyl), Act6, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
86)
(Aib2, Glu3(NH-hexyl), 3-Pal9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
87)
(Aib2, Glu3(NH-hexyl), Dmt7, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
88)
(Aib2, Glu3(NH-hexyl), Thz7, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
88)
(Aib2, Glu3(NH-hexyl), A5c5,12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
84)
(Aib2,5, Glu3(NH-hexyl), A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
84)
(Aib2, Glu3(NH-hexyl), hLeu5, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
84)
(Aib2, Glu3(NH-hexyl), Cha5, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
84)
(Aib2,6, Glu3(NH-hexyl), A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
86)
(Aib2, Glu3(NH-hexyl), Thr6, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
86)
(Aib2, Glu3(NH-hexyl), Abu6, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
86)
(Aib2, Glu3(NH-hexyl), 4-Hyp', A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
88)
(Aib2, Glu3(NH-hexyl), Pip', A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
88)
(Aib2, Glu3(NH-hexyl), Dhp7, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
88)
(Aib2, Glu3(NH-hexyl), Ktp7, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
88)
(Aib2,8, Glu3(NH-hexyl), A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
89)
(Aib2, Glu3(NH-hexyl), 2-Pal9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
87)
(Aib2, Glu3(NH-hexyl), 3-Pal9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
87)
(Aib2, Glu3(NH-hexyl), 4-Pal9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
87)
(Aib2, Glu3(NH-hexyl), Taz9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
87)
(Aib2, Glu3(NH-hexyl), 2-Thi9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
87)
(Aib2, Glu3(NH-hexyl), 2-Fua9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
87)
(Aib2, Glu3(NH-hexyl), Apc9,16, A5c12)hGhrelin(1-28)-NH2;
(SEQ ID:
87)
(Aib2,9, Glu3(NH-hexyl), A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
87)
(Aib2,10, Glu3(NH-hexyl), A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
90)
(Glu3(O-hexyl))hGhrelin(1-28)-NH2;
(SEQ ID:
91)
(Aib2)hGhrelin(1-28)-NH2;
(SEQ ID:
15)
(Glu3(NH-hexyl))hGhrelin(1-28)-NH2;
(SEQ ID:
91)
(Aib2, Glu3(O-hexyl))hGhrelin(1-28)-NH2;
(SEQ ID:
92)
Glu3(O-hexyl))hGhrelin(1-28)-NH2;
(SEQ ID:
93)
(Aib2, Glu3(NH-hexyl))hGhrelin(1-28)-NH2;
(SEQ ID:
92)
(Dap3(octanesulfonyl))hGhrelin(1-28)-NH2;
(SEQ ID:
6)
(Aib2, Dap3(octanesulfonyl))hGhrelin(1-28)-NH2;
(SEQ ID:
94)
Dap3(octanesulfonyl))hGhrelin(1-28)-NH2;
(SEQ ID:
93)
(Ava2, Dap3(octanesulfonyl))hGhrelin(2-28)-NH2;
(SEQ ID:
126)
(Ac-Gly1)hGhrelin(1-5)-NH2;
(SEQ ID:
95)
(Ac-Gly1)hGhrelin(1-6)-NH2;
(SEQ ID:
96)
(Ac-Gly1)hGhrelin(1-7)-NH2;
(SEQ ID:
97)
(Ac-Gly1, Aib2)hGhrelin(1-28)-NH2;
(SEQ ID:
98)
(Ac-Gly1, Aib2, Glu3(NH-hexyl))hGhrelin(1-5)-NH2;
(SEQ ID:
99)
(Ac-Gly1, Aib2, Glu3(NH-hexyl))hGhrelin(1-6)-NH2;
(SEQ ID:
100)
(Ac-Gly1, Aib2, Glu3(NH-hexyl))hGhrelin(1-7)-NH2;
(SEQ ID:
101)
(Ac-Gly1, Aib2, Glu3(NH-hexyl))hGhrelin(1-28)-NH2;
(SEQ ID:
102)
(Ac-Gly1, Aib2, Glu3(NH-hexyl), Arg8)hGhrelin(1-8)-NH2;
(SEQ ID:
103)
(Ac-Gly1, Aib2, Glu3(NH-hexyl), Lys8)hGhrelin(1-8)-NH2;
(SEQ ID:
103)
(n-butyryl-Gly1)hGhrelin(1-28)-NH2;
(SEQ ID:
104)
(n-butyryl-Gly1, Aib2, Glu3(NH-hexyl))hGhrelin(1-28)-NH2;
(SEQ ID:
105)
(isobutyryl-Gly1)hGhrelin(1-28)-NH2;
(SEQ ID:
104)
(n-octanoyl-Gly1)hGhrelin(1-28)-NH2, (SEQ ID:
104)
Cys3(S(CH2)9CH3)hGhrelin(1-28)-NH2;
(SEQ ID:
106)
(Aib2, Ser3)hGhrelin(1-28)-NH2;
(SEQ ID:
15)
(Aib2,6, Ser3)hGhrelin(1-28)-NH2 (SEQ ID:
9)
(Aib2, Ser3, 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
13)
(Aib2, Ser3, Thz7)hGhrelin(1-28)-NH2;
(SEQ ID:
14)
(Aib2, Ser3, Cha5)hGhrelin(1-28)-NH2;
(SEQ ID:
7)
(Aib2, Ser3, Abu6)hGhrelin(1-28)-NH2;
(SEQ ID:
9)
(Aib2, Ser3, 4-Hyp7)hGhrelin(1-28)-NH2;
(SEQ ID:
14)
(Aib2, Ser3, Taz9)hGhrelin(1-28)-NH2;
(SEQ ID:
13)
(Aib2, Ser3, Dhp7)hGhrelin(1-28)-NH2;
(SEQ ID:
14)
(Aib2,8, Ser3)hGhrelin(1-28)-NH2;
(SEQ ID:
16)
(Aib2, Ser3, Pip7)hGhrelin(1-28)-NH2;
(SEQ ID:
14)
(Ac-Gly1, Aib2,10, Ser3)hGhrelin(1-28)-NH2;
(SEQ ID:
107)
(Aib2,10, Ser3)hGhrelin(1-28)-NH2;
(SEQ ID:
17)
(n-butyryl-Gly1, Aib2, Ser3)hGhrelin(1-28)-NH2;
(SEQ ID:
108)
(Ac-Gly1, Aib2, Ser3)hGhrelin(1-28)-NH2;
(SEQ ID:
98)
(Aib2, Ser3, Tic7)hGhrelin(1-28)-NH2;
(SEQ ID:
14)
(Ac-Gly1, Aib2, Ser3, Arg8)hGhrelin(1-28)-NH2;
(SEQ ID:
109)
(Ser3, Aib8)hGhrelin(1-28)-NH2;
(SEQ ID:
110)
(Ser3, Taz9)hGhrelin(1-28)-NH2;
(SEQ ID:
19)
(Ser3, 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
19)
(Ser3, 4-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
19)
(Aib2, Ser3, 2-Thi9)hGhrelin(1-28)-NH2;
(SEQ ID:
13)
(Ser3, 2-Thi9)hGhrelin(1-28)-NH2;
(SEQ ID:
19)
(Ser3, 4-Hyp7)hGhrelin(1-28)-NH2;
(SEQ ID:
20)
(Aib2, Ser3, Tic7)hGhrelin(1-28)-NH2;
(SEQ ID:
14)
(Aib2, Thr3)hGhrelin(1-28)-NH2;
(SEQ ID:
111)
(Aib2,6, Thr3)hGhrelin(1-28)-NH2;
(SEQ ID:
112)
(A5c5, Thr3)hGhrelin(1-28)-NH2;
(SEQ ID:
113)
(Aib2, Thr3, 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
114)
(Aib2, Thr3, Thz7)hGhrelin(1-28)-NH2;
(SEQ ID:
115)
(Aib2, Thr3, Cha5)hGhrelin(1-28)-NH2;
(SEQ ID:
116)
(Aib2, Thr3, Abu6)hGhrelin(1-28)-NH2;
(SEQ ID:
112)
(Aib2, Thr3, 4-Hyp7)hGhrelin(1-28)-NH2;
(SEQ ID:
115)
(Aib2, Thr3, Taz9)hGhrelin(1-28)-NH2;
(SEQ ID:
114)
(Aib2, Thr3, Dhp7)hGhrelin(1-28)-NH2;
(SEQ ID:
115)
(Aib2,8, Thr3)hGhrelin(1-28)-NH2;
(SEQ ID:
117)
(Aib2, Thr3, Pip7)hGhrelin(1-28)-NH2;
(SEQ ID:
115)
(Ac-Gly1, Aib2,10, Thr3)hGhrelin(1-28)-NH2;
(SEQ ID:
118)
(Aib2,10, Thr3)hGhrelin(1-28)-NH2;
(SEQ ID:
118)
(n-butyryl-Gly1, Aib2, Thr3)hGhrelin(1-28)-NH2;
(SEQ ID:
119)
(Ac-Gly1, Aib2, Thr3)hGhrelin(1-28)-NH2;
(SEQ ID:
119)
(Aib2, Thr3, Tic7)hGhrelin(1-28)-NH2;
(SEQ ID:
115)
(Ac-Gly1, Aib2, Thr3, Arg8)hGhrelin(1-28)-NH2;
(SEQ ID:
120)
(Thr3, Aib8)hGhrelin(1-28)-NH2;
(SEQ ID:
121)
(Thr3, Taz9)hGhrelin(1-28)-NH2;
(SEQ ID:
122)
(Thr3, 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
122)
(Thr3, 4-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
122)
(Aib2, Thr3, 2-Thi9)hGhrelin(1-28)-NH2;
(SEQ ID:
114)
(Thr3, 2-Thi9)hGhrelin(1-28)-NH2;
(SEQ ID:
122)
(Thr3, 4-Hyp7)hGhrelin(1-28)-NH2;
(SEQ ID:
123)
(Aib2, Thr3, Tic7)hGhrelin(1-28)-NH2;
(SEQ ID:
115)
(Ac-Gly1, Glu3(NH-hexyl))hGhrelin(1-28)-NH2;
(SEQ ID:
124)
H-Inp-D-1-Nal-D-Trp-3-Pal-Lys-NH2;
(SEQ ID:
128)
H-Inp-D-2-Nal-D-Trp-4-Pal-Lys-NH2;
(SEQ ID:
129)
H-Inp-D-2-Nal-D-Trp-Om-Lys-NH2;
(SEQ ID:
129)
H-Inp-D-Bip-D-Trp-Phe-Lys-NH2;
(SEQ ID:
130)
H-Inp-D-2-Nal-D-Trp-Thr(Bzl)-Lys-NH2;
(SEQ ID:
131)
H-Inp-D-2-Nal-D-Trp-Pff-Lys-NH2;
(SEQ ID:
131)
H-Inp-D-2-Nal-D-Trp-2-Thi-Lys-NH2;
(SEQ ID:
132)
H-Inp-D-2-Nal-D-Trp-Taz-Lys-NH2;
(SEQ ID:
132)
H-Inp-D-Dip-D-Trp-Phe-Lys-NH2;
(SEQ ID:
133)
H-Inp-D-Bpa-D-Trp-Phe-Lys-NH2;
(SEQ ID:
133)
H-Inp-D-2-Nal-D-Bpa-Phe-Lys-NH2;
(SEQ ID:
134)
H-Inp-D-2-Nal-D-Trp-3-Pal-NH2;
(SEQ ID:
135)
H-Inp-D-2-Nal-D-Trp-4-Pal-NH2;
(SEQ ID:
135)
H-Inp-D-1-Nal-D-Trp-3-Pal-NH2;
(SEQ ID:
136)
H-Inp-D-Bip-D-Trp-Phe-NH2;
(SEQ ID:
137)
H-Inp-D-2-Nal-D-Trp-Thr(Bzl)-NH2;
(SEQ ID:
138)
H-Inp-D-2-Nal-D-Trp-Pff-NH2;
(SEQ ID:
138)
H-Inp-D-2-Nal-D-Trp-2-Thi-NH2;
(SEQ ID:
138)
H-Inp-D-2-Nal-D-Trp-Taz-NH2;
(SEQ ID:
138)
H-Inp-D-Dip-D-Trp-Phe-NH2;
(SEQ ID:
139)
H-Inp-D-2-Nal-D-Dip-Phe-NH2;
(SEQ ID:
140)
H-Inp-D-Bal -D-Trp-Phe-NH2;
(SEQ ID:
141)
H-Inp-D-2-Nal-D-Bal -Phe-NH2;
(SEQ ID:
142)
H-Inp-D-2-Nal-D-Trp-3-Pal-Lys-NH2;
(SEQ ID:
143)
H-Inp-D-Trp-D-2-Nal(Ψ)-Pim;
(SEQ ID:
127)
H-Inp-D-Bal -D-Trp-2-Thi-Lys-NH2;
(SEQ ID:
144)
H-Inp-D-Bal -D-Trp-Phe-Lys-NH2;
(SEQ ID:
144)
H-Inp-D-1-Nal-D-Trp-2-Thi-Lys-NH2;
(SEQ ID:
128)
H-Inp-D-2-Nal-D-Trp-Phe-Apc-NH2;
(SEQ ID:
2)
H-Inp-D-1-Nal-D-Trp-Phe-Apc-NH2;
(SEQ ID:
2)
H-Inp-D-Bal-D-Trp-Phe-Apc-NH2;
(SEQ ID:
2)
H-Apc-D-2-Nal-D-Trp-Phe-Lys-NH2;
(SEQ ID:
145)
H-Apc-D-1-Nal-D-Trp-2-Thi-Lys-NH2;
(SEQ ID:
146)
H-Inp-D-1-Nal-D-Trp-2-Thi-NH2;
(SEQ ID:
147)
H-Apc-D-1-Nal-D-Trp-Phe-NH2;
(SEQ ID:
148)
H-Inp-D-2-Nal-D-Trp(Ψ)-Pim;
(SEQ ID:
149)
H-Inp-D-1-Nal-D-Trp(Ψ)-Pim;
(SEQ ID:
149)
H-Inp-D-Bal-D-Trp(Ψ)-Pim;
(SEQ ID:
149)
H-Aib-D-Ser(Bzl)-D-Trp(Ψ)-Pim;
(SEQ ID:
150)
H-Inp-D-1-Nal-D-Trp-Taz-Lys-NH2;
(SEQ ID:
151)
H-Inp-D-Bal -D-Trp-Taz-Lys-NH2;
(SEQ ID:
151)
H-Apc-D-1-Nal-D-Trp-Taz-Lys-NH2;
(SEQ ID:
152)
H-Apc-D-Bal -D-Trp-Taz-Lys-NH2;
(SEQ ID:
152)
H-Apc-D-Bal -D-Trp-2-Thi-Lys-NH2;
(SEQ ID:
153)
H-Apc-D-Bal -D-Trp-Phe-Lys-NH2;
(SEQ ID:
153)
H-Apc-D-1-Nal-D-Trp-Phe-Apc-NH2;
(SEQ ID:
154)
H-Apc-D-Bal -D-Trp-Phe-Apc-NH2;
(SEQ ID:
154)
H-Apc-D-1-Nal-D-1-Nal-Phe-Apc-NH2;
(SEQ ID:
155)
H-Apc-D-1-Nal-D-2-Nal-Phe-Apc-NH2;
(SEQ ID:
155)
H-Apc-D-1-Nal-D-1-Nal-Phe-Lys-NH2;
(SEQ ID:
156)
H-Apc-D-Bal-D-1-Nal-Phe-Apc-NH2;
(SEQ ID:
157)
H-Apc-D-Bal-D-2-Nal-Phe-Apc-NH2;
(SEQ ID:
157)
H-Apc-D-Bal-D-1-Nal-Phe-Lys-NH2;
(SEQ ID:
158)
H-Apc-D-Bal-D-2-Nal-Phe-Lys-NH2;
(SEQ ID:
158)
H-Apc-D-1-Nal-D-Trp-2-Thi-NH2;
(SEQ ID:
159)
H-Apc-D-Bal -D-Trp-Phe-NH2;
(SEQ ID:
160)
H-Apc-D-1-Nal-D-Trp-Taz-NH2;
(SEQ ID:
159)
H-Apc-D-Bal -D-Trp-2-Thi-NH2;
(SEQ ID:
161)
H-Apc-D-Bal -D-Trp-Taz-NH2;
(SEQ ID:
161)
H-Apc-D-2-Nal-D-Trp-2-Thi-NH2;
(SEQ ID:
162)
H-Apc-D-2-Nal-D-Trp-Taz-NH2;
(SEQ ID:
162)
H-Inp-D-1-Nal-D-Trp-Taz-Apc-NH2;
(SEQ ID:
163)
H-Inp-D-Bal-D-Trp-Taz-Apc-NH2;
(SEQ ID:
163)
H-Apc-D-1-Nal-D-Trp-Taz-Apc-NH2;
(SEQ ID:
164)
H-Apc-D-Bal -D-Trp-Taz-Apc-NH2;
(SEQ ID:
164)
H-Apc-D-1-Nal-D-Trp-2-Fua-Apc-NH2;
(SEQ ID:
165)
H-Apc-D-1-Nal-D-Trp-2-Fua-Lys-NH2;
(SEQ ID:
165)
H-Apc-D-1-Nal-D-Trp-2-Fua-NH2;
(SEQ ID:
165)
H-Apc-D-1-Nal-D-Trp-2-Pal-NH2;
(SEQ ID:
166)
H-Apc-D-1-Nal-D-Trp-3-Pal-NH2;
(SEQ ID:
166)
H-Apc-D-1-Nal-D-Trp-3-Thi-Apc-NH2;
(SEQ ID:
167)
H-Apc-D-1-Nal-D-Trp-3-Thi-Lys-NH2;
(SEQ ID:
167)
H-Apc-D-1-Nal-D-Trp-3-Thi-NH2;
(SEQ ID:
168)
H-Apc-D-1-Nal-D-Trp-4-Pal-NH2;
(SEQ ID:
168)
H-Apc-D-1-Nal-D-Trp-Pff-Apc-NH2;
(SEQ ID:
169)
H-Apc-D-1-Nal-D-Trp-Pff-Lys-NH2;
(SEQ ID:
169)
H-Apc-D-1-Nal-D-Trp-Pff-NH2;
(SEQ ID:
168)
H-Apc-D-2-Nal-D-Trp-2-Fua-Apc-NH2;
(SEQ ID:
170)
H-Apc-D-2-Nal-D-Trp-2-Fua-Lys-NH2;
(SEQ ID:
170)
H-Apc-D-2-Nal-D-Trp-2-Fua-NH2;
(SEQ ID:
171)
H-Apc-D-2-Nal-D-Trp-2-Pal-NH2;
(SEQ ID:
171)
H-Apc-D-2-Nal-D-Trp-2-Thi-Apc-NH2;
(SEQ ID:
172)
H-Apc-D-2-Nal-D-Trp-2-Thi-Lys-NH2;
(SEQ ID:
172)
H-Apc-D-2-Nal-D-Trp-3-Pal-NH2;
(SEQ ID:
171)
H-Apc-D-2-Nal-D-Trp-3-Thi-Apc-NH2;
(SEQ ID:
173)
H-Apc-D-2-Nal-D-Trp-3-Thi-Lys-NH2;
(SEQ ID:
173)
H-Apc-D-2-Nal-D-Trp-3-Thi-NH2;
(SEQ ID:
171)
H-Apc-D-2-Nal-D-Trp-4-Pal-NH2;
(SEQ ID:
171)
H-Apc-D-2-Nal-D-Trp-Pff-Apc-NH2;
(SEQ ID:
174)
H-Apc-D-2-Nal-D-Trp-Pff-Lys-NH2;
(SEQ ID:
174)
H-Apc-D-2-Nal-D-Trp-Pff-NH2;
(SEQ ID:
171)
H-Apc-D-2-Nal-D-Trp-Taz-Apc-NH2;
(SEQ ID:
175)
H-Apc-D-2-Nal-D-Trp-Taz-Lys-NH2;
(SEQ ID:
175)
H-Apc-D-Bal -D-Bal -2-Fua-Apc-NH2;
(SEQ ID:
176)
H-Apc-D-Bal -D-Bal -2-Fua-Lys-NH2;
(SEQ ID:
176)
H-Apc-D-Bal -D-Bal -2-Fua-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Bal -2-Pal-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Bal -2-Thi-Apc-NH2;
(SEQ ID:
178)
H-Apc-D-Bal -D-Bal -2-Thi-Lys-NH2;
(SEQ ID:
178)
H-Apc-D-Bal -D-Bal -2-Thi-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Bal -3-Pal-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Bal -3-Thi-Apc-NH2;
(SEQ ID:
179)
H-Apc-D-Bal -D-Bal -3-Thi-Lys-NH2;
(SEQ ID:
179)
H-Apc-D-Bal -D-Bal -3-Thi-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Bal -4-Pal-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Bal -Pff-Apc-NH2;
(SEQ ID:
180)
H-Apc-D-Bal -D-Bal -Pff-Lys-NH2;
(SEQ ID:
180)
H-Apc-D-Bal -D-Bal -Pff-NH2;
(SEQ ID:
177)
H-Apc-D-Bal-D-Bal-Phe-Apc-NH2;
(SEQ ID:
181)
H-Apc-D-Bal -D-Bal -Phe-Lys-NH2;
(SEQ ID:
181)
H-Apc-D-Bal -D-Bal -Phe-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Bal -Taz-Apc-NH2;
(SEQ ID:
182)
H-Apc-D-Bal -D-Bal -Taz-Lys-NH2;
(SEQ ID:
182)
H-Apc-D-Bal -D-Bal -Taz-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Trp-2-Fua-Apc-NH2;
(SEQ ID:
183)
H-Apc-D-Bal -D-Trp-2-Fua-Lys-NH2;
(SEQ ID:
183)
H-Apc-D-Bal -D-Trp-2-Fua-NH2;
(SEQ ID:
184)
H-Apc-D-Bal -D-Trp-2-Pal-NH2;
(SEQ ID:
184)
H-Apc-D-Bal -D-Trp-3-Pal-NH2;
(SEQ ID:
184)
H-Apc-D-Bal -D-Trp-3-Thi-Apc-NH2;
(SEQ ID:
185)
H-Apc-D-Bal -D-Trp-3-Thi-Lys-NH2;
(SEQ ID:
185)
H-Apc-D-Bal -D-Trp-3-Thi-NH2;
(SEQ ID:
184)
H-Apc-D-Bal -D-Trp-4-Pal-NH2;
(SEQ ID:
184)
H-Apc-D-Bal -D-Trp-Pff-Apc-NH2;
(SEQ ID:
186)
H-Apc-D-Bal -D-Trp-Pff-Lys-NH2;
(SEQ ID:
186)
H-Apc-D-Bal -D-Trp-Pff-NH2;
(SEQ ID:
184)
H-Inp-D-1-Nal-D-Bal -2-Fua-Lys-NH2;
(SEQ ID:
187)
H-Inp-D-1-Nal-D-Bal -2-Fua-NH2;
(SEQ ID:
188)
H-Inp-D-1-Nal-D-Bal -2-Thi-Lys-NH2;
(SEQ ID:
187)
H-Inp-D-1-Nal-D-Bal -3-Thi-Lys-NH2;
(SEQ ID:
187)
H-Inp-D-1-Nal-D-Bal -Pff-Lys-NH2;
(SEQ ID:
187)
H-Inp-D-1-Nal-D-Bal -Pff-NH2;
(SEQ ID:
188)
H-Inp-D-1-Nal-D-Bal -Phe-Lys-NH2;
(SEQ ID:
187)
H-Inp-D-1-Nal-D-Bal -Taz-Lys-NH2;
(SEQ ID:
187)
H-Inp-D-1-Nal-D-Bal -Taz-NH2;
(SEQ ID:
188)
H-Inp-D-1-Nal-D-Trp-2-Fua-Apc-NH2;
(SEQ ID:
189)
H-Inp-D-1-Nal-D-Trp-2-Fua-Lys-NH2;
(SEQ ID:
189)
H-Inp-D-1-Nal-D-Trp-2-Fua-NH2;
(SEQ ID:
189)
H-Inp-D-1-Nal-D-Trp-3-Thi-Apc-NH2;
(SEQ ID:
190)
H-Inp-D-1-Nal-D-Trp-3-Thi-Lys-NH2;
(SEQ ID:
190)
H-Inp-D-1-Nal-D-Trp-Pff-Apc-NH2;
(SEQ ID:
191)
H-Inp-D-1-Nal-D-Trp-Pff-Lys-NH2;
(SEQ ID:
191)
H-Inp-D-1-Nal-D-Trp-Pff-NH2;
(SEQ ID:
192)
H-Inp-D-1-Nal-D-Trp-Taz-NH2;
(SEQ ID:
192)
H-Inp-D-2-Nal-D-Trp-2-Fua-Apc-NH2;
(SEQ ID:
193)
H-Inp-D-2-Nal-D-Trp-2-Fua-NH2;
(SEQ ID:
194)
H-Inp-D-2-Nal-D-Trp-2-Thi-Apc-NH2;
(SEQ ID:
193)
H-Inp-D-2-Nal-D-Trp-3-Thi-Apc-NH2;
(SEQ ID:
193)
H-Inp-D-2-Nal-D-Trp-3-Thi-Lys-NH2;
(SEQ ID:
195)
H-Inp-D-2-Nal-D-Trp-3-Thi-NH2;
(SEQ ID:
194)
H-Inp-D-2-Nal-D-Trp-Pff-Apc-NH2;
(SEQ ID:
193)
H-Inp-D-2-Nal-D-Trp-Pff-NH2;
(SEQ ID:
194)
H-Inp-D-2-Nal-D-Trp-Taz-Apc-NH2;
(SEQ ID:
193)
H-Inp-D-2-Nal-D-Trp-Taz-NH2;
(SEQ ID:
194)
H-Inp-D-Bal -D-Bal -2-Fua-Lys-NH2;
(SEQ ID:
196)
H-Inp-D-Bal -D-Bal -2-Fua-NH2;
(SEQ ID:
197)
H-Inp-D-Bal -D-Bal -2-Thi-Lys-NH2;
(SEQ ID:
196)
H-Inp-D-Bal -D-Bal -3-Thi-Lys-NH2;
(SEQ ID:
196)
H-Inp-D-Bal -D-Bal -Pff-Lys-NH2;
(SEQ ID:
196)
H-Inp-D-Bal -D-Bal -Pff-NH2;
(SEQ ID:
197)
H-Inp-D-Bal -D-Bal -Phe-Lys-NH2;
(SEQ ID:
196)
H-Inp-D-Bal -D-Bal -Taz-Lys-NH2;
(SEQ ID:
196)
H-Inp-D-Bal -D-Bal -Taz-NH2;
(SEQ ID:
197)
H-Inp-D-Bal -D-Trp-2-Fua-Apc-NH2;
(SEQ ID:
198)
H-Inp-D-Bal -D-Trp-2-Fua-Lys-NH2;
(SEQ ID:
198)
H-Inp-D-Bal -D-Trp-2-Fua-NH2;
(SEQ ID:
199)
H-Inp-D-Bal -D-Trp-3-Thi-Apc-NH2;
(SEQ ID:
200)
H-Inp-D-Bal -D-Trp-3-Thi-Lys-NH2;
(SEQ ID:
200)
H-Inp-D-Bal-D-Trp-Pff-Apc-NH2;
(SEQ ID:
201)
H-Inp-D-Bal -D-Trp-Pff-Lys-NH2;
(SEQ ID:
201)
H-Inp-D-Bal -D-Trp-Pff-NH2;
(SEQ ID:
199)
H-Inp-D-Bal -D-Trp-Taz-NH2;
(SEQ ID:
199)
H-Inp-D-Bip-D-Bal -2-Fua-Lys-NH2;
(SEQ ID:
202)
H-Inp-D-Bip-D-Bal -2-Fua-NH2;
(SEQ ID:
203)
H-Inp-D-Bip-D-Bal -2-Thi-Lys-NH2;
(SEQ ID:
202)
H-Inp-D-Bip-D-Bal -3-Thi-Lys-NH2;
(SEQ ID:
202)
H-Inp-D-Bip-D-Bal -Pff-Lys-NH2;
(SEQ ID:
202)
H-Inp-D-Bip-D-Bal -Pff-NH2;
(SEQ ID:
203)
H-Inp-D-Bip-D-Bal -Taz-Lys-NH2;
(SEQ ID:
204)
H-Inp-D-Bip-D-Bal -Taz-NH2;
(SEQ ID:
205)
H-Inp-D-Bip-D-Trp-2-Fua-Lys-NH2;
(SEQ ID:
206)
H-Inp-D-Bip-D-Trp-2-Fua-NH2;
(SEQ ID:
207)
H-Inp-D-Bip-D-Trp-2-Thi-Lys-NH2;
(SEQ ID:
206)
H-Inp-D-Bip-D-Trp-3-Thi-Lys-NH2;
(SEQ ID:
206)
H-Inp-D-Bip-D-Trp-Pff-Lys-NH2;
(SEQ ID:
206)
H-Inp-D-Bip-D-Trp-Pff-NH2;
(SEQ ID:
207)
H-Inp-D-Bip-D-Trp-Taz-Lys-NH2;
(SEQ ID:
206)
H-Inp-D-Bip-D-Trp-Taz-NH2;
(SEQ ID:
207)
H-Inp-D-1-Nal-D-Trp-3-Pal-Lys-NH2;
(SEQ ID:
128)
H-Inp-D-2-Nal-D-Trp-4-Pal-Lys-NH2;
(SEQ ID:
129)
H-Inp-D-2-Nal-D-Trp-Om-Lys-NH2;
(SEQ ID:
129)
H-Inp-D-Bip-D-Trp-Phe-Lys-NH2;
(SEQ ID:
130)
H-Inp-D-2-Nal-D-Trp-Thr(Bzl)-Lys-NH2;
(SEQ ID:
131)
H-Inp-D-2-Nal-D-Trp-Pff-Lys-NH2;
(SEQ ID:
131)
H-Inp-D-2-Nal-D-Trp-2-Thi-Lys-NH2;
(SEQ ID:
132)
H-Inp-D-2-Nal-D-Trp-Taz-Lys-NH2;
(SEQ ID:
132)
H-Inp-D-Dip-D-Trp-Phe-Lys-NH2;
(SEQ ID:
133)
H-Inp-D-Bpa-D-Trp-Phe-Lys-NH2;
(SEQ ID:
133)
H-Inp-D-2-Nal-D-Bpa-Phe-Lys-NH2;
(SEQ ID:
134)
H-Inp-D-2-Nal-D-Trp-Thr(Bzl)-NH2;
(SEQ ID:
138)
H-Inp-D-2-Nal-D-Trp-Pff-NH2;
(SEQ ID:
138)
H-Inp-D-2-Nal-D-Trp-Taz-NH2;
(SEQ ID:
138)
H-Inp-D-2-Nal-D-Dip-Phe-NH2;
(SEQ ID:
140)
H-Inp-D-2-Nal-D-Trp-3-Pal-Lys-NH2;
(SEQ ID:
143)
H-Inp-D-Trp-D-2-Nal(Ψ)-Pim;
(SEQ ID:
127)
H-Inp-D-Bal -D-Trp-2-Thi-Lys-NH2;
(SEQ ID:
144)
H-Inp-D-Bal -D-Trp-Phe-Lys-NH2;
(SEQ ID:
144)
H-Inp-D-1-Nal-D-Trp-2-Thi-Lys-NH2;
(SEQ ID:
128)
H-Inp-D-2-Nal-D-Trp-Phe-Apc-NH2;
(SEQ ID:
2)
H-Inp-D-1-Nal-D-Trp-Phe-Apc-NH2;
(SEQ ID:
2)
H-Inp-D-Bal-D-Trp-Phe-Apc-NH2;
(SEQ ID:
2)
H-Apc-D-2-Nal-D-Trp-Phe-Lys-NH2;
(SEQ ID:
145)
H-Apc-D-1-Nal-D-Trp-2-Thi-Lys-NH2;
(SEQ ID:
146)
H-Inp-D-2-Nal-D-Trp(Ψ)-Pim;
(SEQ ID:
149)
H-Inp-D-1-Nal-D-Trp(Ψ)-Pim;
(SEQ ID:
149)
H-Inp-D-Bal-D-Trp(Ψ)-Pim;
(SEQ ID:
149)
H-Aib-D-Ser(Bzl)-D-Trp(Ψ)-Pim;
(SEQ ID:
150)
H-Inp-D-1-Nal-D-Trp-Taz-Lys-NH2;
(SEQ ID:
151)
H-Inp-D-Bal -D-Trp-Taz-Lys-NH2;
(SEQ ID:
151)
H-Apc-D-1-Nal-D-Trp-Taz-Lys-NH2;
(SEQ ID:
152)
H-Apc-D-Bal -D-Trp-Taz-Lys-NH2;
(SEQ ID:
152)
H-Apc-D-Bal -D-Trp-2-Thi-Lys-NH2;
(SEQ ID:
153)
H-Apc-D-Bal -D-Trp-Phe-Lys-NH2;
(SEQ ID:
153)
H-Apc-D-1-Nal-D-Trp-Phe-Apc-NH2;
(SEQ ID:
154)
H-Apc-D-Bal -D-Trp-Phe-Apc-NH2;
(SEQ ID:
154)
H-Apc-D-1-Nal-D-1-Nal-Phe-Apc-NH2;
(SEQ ID:
155)
H-Apc-D-1-Nal-D-2-Nal-Phe-Apc-NH2;
(SEQ ID:
155)
H-Apc-D-1-Nal-D-1-Nal-Phe-Lys-NH2;
(SEQ ID:
156)
H-Apc-D-Bal-D-1-Nal-Phe-Apc-NH2;
(SEQ ID:
157)
H-Apc-D-Bal-D-2-Nal-Phe-Apc-NH2;
(SEQ ID:
157)
H-Apc-D-Bal-D-1-Nal-Phe-Lys-NH2;
(SEQ ID:
158)
H-Apc-D-Bal-D-2-Nal-Phe-Lys-NH2;
(SEQ ID:
158)
H-Apc-D-1-Nal-D-Trp-2-Thi-NH2;
(SEQ ID:
159)
H-Apc-D-Bal -D-Trp-Phe-NH2;
(SEQ ID:
160)
H-Apc-D-1-Nal-D-Trp-Taz-NH2;
(SEQ ID:
159)
H-Apc-D-Bal -D-Trp-2-Thi-NH2;
(SEQ ID:
161)
H-Apc-D-Bal -D-Trp-Taz-NH2;
(SEQ ID:
161)
H-Apc-D-2-Nal-D-Trp-2-Thi-NH2;
(SEQ ID:
162)
H-Apc-D-2-Nal-D-Trp-Taz-NH2;
(SEQ ID:
162)
H-Inp-D-1-Nal-D-Trp-Taz-Apc-NH2;
(SEQ ID:
163)
H-Inp-D-Bal-D-Trp-Taz-Apc-NH2;
(SEQ ID:
163)
H-Apc-D-1-Nal-D-Trp-Taz-Apc-NH2;
(SEQ ID:
164)
H-Apc-D-Bal -D-Trp-Taz-Apc-NH2;
(SEQ ID:
164)
H-Inp-D-2-Nal-D-Trp-3-Thi-Lys-NH2;
(SEQ ID:
195)
H-Inp-D-Bal -D-Trp-3-Thi-Lys-NH2;
(SEQ ID:
200)
H-Inp-D-Bal -D-Trp-2-Fua-Lys-NH2;
(SEQ ID:
198)
H-Inp-D-Bal -D-Trp-Pff-Lys-NH2;
(SEQ ID:
201)
H-Inp-D-Bal -D-Trp-3-Thi-Apc-NH2;
(SEQ ID:
200)
H-Inp-D-Bal -D-Trp-2-Fua-Apc-NH2;
(SEQ ID:
198)
H-Inp-D-Bal-D-Trp-Pff-Apc-NH2;
(SEQ ID:
201)
H-Apc-D-Bal -D-Trp-3-Thi-Lys-NH2;
(SEQ ID:
185)
H-Apc-D-Bal -D-Trp-2-Fua-Lys-NH2;
(SEQ ID:
183)
H-Apc-D-Bal -D-Trp-Pff-Lys-NH2;
(SEQ ID:
186)
H-Inp-D-Bal -D-Bal -Phe-Lys-NH2;
(SEQ ID:
196)
H-Inp-D-Bal -D-Bal -2-Thi-Lys-NH2;
(SEQ ID:
196)
H-Inp-D-Bal -D-Bal -3-Thi-Lys-NH2;
(SEQ ID:
196)
H-Inp-D-Bal -D-Bal -Taz-Lys-NH2;
(SEQ ID:
196)
H-Inp-D-Bal -D-Bal -2-Fua-Lys-NH2;
(SEQ ID:
196)
H-Inp-D-Bal -D-Bal -Pff-Lys-NH2;
(SEQ ID:
196)
H-Apc-D-Bal -D-Bal -Phe-Lys-NH2;
(SEQ ID:
181)
H-Apc-D-Bal -D-Bal -2-Thi-Lys-NH2;
(SEQ ID:
178)
H-Apc-D-Bal -D-Bal -3-Thi-Lys-NH2;
(SEQ ID:
179)
H-Apc-D-Bal -D-Bal -Taz-Lys-NH2;
(SEQ ID:
182)
H-Apc-D-Bal -D-Bal -2-Fua-Lys-NH2;
(SEQ ID:
176)
H-Apc-D-Bal -D-Bal -Pff-Lys-NH2;
(SEQ ID:
180)
H-Inp-D-1-Nal-D-Trp-3-Thi-Lys-NH2;
(SEQ ID:
190)
H-Inp-D-1-Nal-D-Trp-2-Fua-Lys-NH2;
(SEQ ID:
189)
H-Inp-D-1-Nal-D-Trp-Pff-Lys-NH2;
(SEQ ID:
191)
H-Inp-D-1-Nal-D-Bal -Phe-Lys-NH2;
(SEQ ID:
187)
H-Inp-D-1-Nal-D-Bal -2-Thi-Lys-NH2;
(SEQ ID:
187)
H-Inp-D-1-Nal-D-Bal -3-Thi-Lys-NH2;
(SEQ ID:
187)
H-Inp-D-1-Nal-D-Bal -Taz-Lys-NH2;
(SEQ ID:
187)
H-Inp-D-1-Nal-D-Bal -2-Fua-Lys-NH2;
(SEQ ID:
187)
H-Inp-D-1-Nal-D-Bal -Pff-Lys-NH2;
(SEQ ID:
187)
H-Inp-D-2-Nal-D-Trp-2-Thi-Apc-NH2;
(SEQ ID:
193)
H-Inp-D-2-Nal-D-Trp-3-Thi-Apc-NH2;
(SEQ ID:
193)
H-Inp-D-2-Nal-D-Trp-Taz-Apc-NH2;
(SEQ ID:
193)
H-Inp-D-2-Nal-D-Trp-2-Fua-Apc-NH2;
(SEQ ID:
193)
H-Inp-D-2-Nal-D-Trp-Pff-Apc-NH2;
(SEQ ID:
193)
H-Inp-D-1-Nal-D-Trp-3-Thi-Apc-NH2;
(SEQ ID:
190)
H-Inp-D-1-Nal-D-Trp-2-Fua-Apc-NH2;
(SEQ ID:
189)
H-Inp-D-1-Nal-D-Trp-Pff-Apc-NH2;
(SEQ ID:
191)
H-Apc-D-1-Nal-D-Trp-3-Thi-Lys-NH2;
(SEQ ID:
167)
H-Apc-D-1-Nal-D-Trp-2-Fua-Lys-NH2;
(SEQ ID:
165)
H-Apc-D-1-Nal-D-Trp-Pff-Lys-NH2;
(SEQ ID:
169)
H-Apc-D-2-Nal-D-Trp-2-Thi-Lys-NH2;
(SEQ ID:
172)
H-Apc-D-2-Nal-D-Trp-3-Thi-Lys-NH2;
(SEQ ID:
173)
H-Apc-D-2-Nal-D-Trp-Taz-Lys-NH2;
(SEQ ID:
175)
H-Apc-D-2-Nal-D-Trp-2-Fua-Lys-NH2;
(SEQ ID:
170)
H-Apc-D-2-Nal-D-Trp-Pff-Lys-NH2;
(SEQ ID:
174)
H-Inp-D-Bip-D-Trp-2-Thi-Lys-NH2;
(SEQ ID:
206)
H-Inp-D-Bip-D-Trp-3-Thi-Lys-NH2;
(SEQ ID:
206)
H-Inp-D-Bip-D-Trp-Taz-Lys-NH2;
(SEQ ID:
206)
H-Inp-D-Bip-D-Trp-2-Fua-Lys-NH2;
(SEQ ID:
206)
H-Inp-D-Bip-D-Trp-Pff-Lys-NH2;
(SEQ ID:
206)
H-Inp-D-Bip-D-Bal -2-Thi-Lys-NH2;
(SEQ ID:
202)
H-Inp-D-Bip-D-Bal -3-Thi-Lys-NH2;
(SEQ ID:
202)
H-Inp-D-Bip-D-Bal -Taz-Lys-NH2;
(SEQ ID:
204)
H-Inp-D-Bip-D-Bal -2-Fua-Lys-NH2;
(SEQ ID:
202)
H-Inp-D-Bip-D-Bal-Pff-Lys-NH2;
(SEQ ID:
202)
H-Apc-D-Bal -D-Trp-3-Thi-Apc-NH2;
(SEQ ID:
185)
H-Apc-D-Bal -D-Trp-2-Fua-Apc-NH2;
(SEQ ID:
183)
H-Apc-D-Bal -D-Trp-Pff-Apc-NH2;
(SEQ ID:
186)
H-Apc-D-Bal-D-Bal-Phe-Apc-NH2;
(SEQ ID:
181)
H-Apc-D-Bal -D-Bal -2-Thi-Apc-NH2;
(SEQ ID:
178)
H-Apc-D-Bal -D-Bal -3-Thi-Apc-NH2;
(SEQ ID:
179)
H-Apc-D-Bal -D-Bal -Taz-Apc-NH2;
(SEQ ID:
182)
H-Apc-D-Bal -D-Bal -2-Fua-Apc-NH2;
(SEQ ID:
176)
H-Apc-D-Bal -D-Bal -Pff-Apc-NH2;
(SEQ ID:
180)
H-Apc-D-1-Nal-D-Trp-3-Thi-Apc-NH2;
(SEQ ID:
167)
H-Apc-D-1-Nal-D-Trp-2-Fua-Apc-NH2;
(SEQ ID:
165)
H-Apc-D-1-Nal-D-Trp-Pff-Apc-NH2;
(SEQ ID:
169)
H-Apc-D-2-Nal-D-Trp-2-Thi-Apc-NH2;
(SEQ ID:
172)
H-Apc-D-2-Nal-D-Trp-3-Thi-Apc-NH2;
(SEQ ID:
173)
H-Apc-D-2-Nal-D-Trp-Taz-Apc-NH2;
(SEQ ID:
175)
H-Apc-D-2-Nal-D-Trp-2-Fua-Apc-NH2;
(SEQ ID:
170)
H-Apc-D-2-Nal-D-Trp-Pff-Apc-NH2;
(SEQ ID:
174)
H-Inp-D-Bal -D-Trp-Taz-NH2;
(SEQ ID:
199)
H-Inp-D-Bal -D-Trp-2-Fua-NH2;
(SEQ ID:
199)
H-Inp-D-Bal -D-Trp-Pff-NH2;
(SEQ ID:
199)
H-Apc-D-Bal -D-Trp-3-Thi-NH2;
(SEQ ID:
184)
H-Apc-D-Bal -D-Trp-2-Fua-NH2;
(SEQ ID:
184)
H-Apc-D-Bal -D-Trp-Pff-NH2;
(SEQ ID:
184)
H-Apc-D-Bal -D-Trp-4-Pal-NH2;
(SEQ ID:
184)
H-Apc-D-Bal -D-Trp-3-Pal-NH2;
(SEQ ID:
184)
H-Apc-D-Bal -D-Trp-2-Pal-NH2;
(SEQ ID:
184)
H-Inp-D-Bal -D-Bal -Taz-NH2;
(SEQ ID:
197)
H-Inp-D-Bal -D-Bal -2-Fua-NH2;
(SEQ ID:
197)
H-Inp-D-Bal -D-Bal -Pff-NH2;
(SEQ ID:
197)
H-Apc-D-Bal -D-Bal -Phe-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Bal -2-Thi-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Bal -3-Thi-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Bal -Taz-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Bal -2-Fua-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Bal -Pff-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Bal -4-Pal-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Bal -3-Pal-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Bal -2-Pal-NH2;
(SEQ ID:
177)
H-Inp-D-1-Nal-D-Trp-Taz-NH2;
(SEQ ID:
192)
H-Inp-D-1-Nal-D-Trp-2-Fua-NH2;
(SEQ ID:
189)
H-Inp-D-1-Nal-D-Trp-Pff-NH2;
(SEQ ID:
192)
H-Inp-D-1-Nal-D-Bal -Taz-NH2;
(SEQ ID:
188)
H-Inp-D-1-Nal-D-Bal -2-Fua-NH2;
(SEQ ID:
188)
H-Inp-D-1-Nal-D-Bal -Pff-NH2;
(SEQ ID:
188)
H-Inp-D-2-Nal-D-Trp-Taz-NH2;
(SEQ ID:
194)
H-Inp-D-2-Nal-D-Trp-2-Fua-NH2;
(SEQ ID:
194)
H-Inp-D-2-Nal-D-Trp-Pff-NH2;
(SEQ ID:
194)
H-Apc-D-1-Nal-D-Trp-3-Thi-NH2;
(SEQ ID:
168)
H-Apc-D-1-Nal-D-Trp-2-Fua-NH2;
(SEQ ID:
165)
H-Apc-D-1-Nal-D-Trp-Pff-NH2;
(SEQ ID:
168)
H-Apc-D-1-Nal-D-Trp-4-Pal-NH2;
(SEQ ID:
168)
H-Apc-D-1-Nal-D-Trp-3-Pal-NH2;
(SEQ ID:
166)
H-Apc-D-1-Nal-D-Trp-2-Pal-NH2;
(SEQ ID:
166)
H-Apc-D-2-Nal-D-Trp-3-Thi-NH2;
(SEQ ID:
171)
H-Apc-D-2-Nal-D-Trp-2-Fua-NH2;
(SEQ ID:
171)
H-Apc-D-2-Nal-D-Trp-Pff-NH2;
(SEQ ID:
171)
H-Apc-D-2-Nal-D-Trp-4-Pal-NH2;
(SEQ ID:
171)
H-Apc-D-2-Nal-D-Trp-3-Pal-NH2;
(SEQ ID:
171)
H-Apc-D-2-Nal-D-Trp-2-Pal-NH2;
(SEQ ID:
171)
H-Inp-D-Bip-D-Trp-Taz-NH2;
(SEQ ID:
207)
H-Inp-D-Bip-D-Trp-2-Fua-NH2;
(SEQ ID:
207)
H-Inp-D-Bip-D-Trp-Pff-NH2;
(SEQ ID:
207)
H-Inp-D-Bip-D-Bal -Taz-NH2;
(SEQ ID:
205)
H-Inp-D-Bip-D-Bal -2-Fua-NH2;
(SEQ ID:
203)
H-Inp-D-Bip-D-Bal -Pff-NH2;
(SEQ ID:
203)
H-Inp-D-1-Nal-D-Trp-2-Thi-Apc-NH2;
(SEQ ID:
208)
H-Inp-D-Bal -D-Trp-2-Thi-Apc-NH2;
(SEQ ID:
208)
H-Apc-D-1-Nal-D-Trp-2-Thi-Apc-NH2;
(SEQ ID:
209)
H-Apc-D-Bal -D-Trp-2-Thi-Apc-NH2;
(SEQ ID:
209)
H-Apc-D-1-Nal-D-Trp-Phe-Lys-NH2;
(SEQ ID:
145)
(Ser(n-octanoyl)15)hGhrelin(1-28)-NH2;
(SEQ ID:
210)
(Glu(NH-hexyl)15)hGhrelin(1-28)-NH2;
(SEQ ID:
211)
(Glu(NH-hexyl)3,15)hGhrelin(1-28)-NH2;
(SEQ ID:
212)
(Glu(NH-hexyl)3, Ser(n-octanoyl)15)hGhrelin(1-28)-NH2;
(SEQ ID:
213)
(Aib2, Glu(NH-hexyl)15)hGhrelin(1-28)-NH2;
(SEQ ID:
214)
(Aib2, Glu(NH-hexyl)3,15)hGhrelin(1-28)-NH2;
(SEQ ID:
215)
(Aib2,8, Glu(NH-hexyl)15)hGhrelin(1-28)-NH2;
(SEQ ID:
216)
(Aib2,8, Glu(NH-hexyl)3,15)hGhrelin(1-28)-NH2;
(SEQ ID:
217)
(Aib2,10, Glu(NH-hexyl)15)hGhrelin(1-28)-NH2;
(SEQ ID:
218)
(Aib2,10, Glu(NH-hexyl)3,15)hGhrelin(1-28)-NH2;
(SEQ ID:
219)
(Ser(n-octanoyl)16)hGhrelin(1-28)-NH2;
(SEQ ID:
220)
(Glu(NH-hexyl)16)hGhrelin(1-28)-NH2;
(SEQ ID:
221)
(Glu(NH-hexyl)3,16)hGhrelin(1-28)-NH2;
(SEQ ID:
222)
(Glu(NH-hexyl)3, Ser(n-octanoyl)16)hGhrelin(1-28)-NH2;
(SEQ ID:
223)
(Aib2, Glu(NH-hexyl)16)hGhrelin(1-28)-NH2;
(SEQ ID:
224)
(Aib2, Glu(NH-hexyl)3,16)hGhrelin(1-28)-NH2;
(SEQ ID:
225)
(Aib2,8, Glu(NH-hexyl)16)hGhrelin(1-28)-NH2;
(SEQ ID:
226)
(Aib2,8, Glu(NH-hexyl)3,16)hGhrelin(1-28)-NH2;
(SEQ ID:
227)
(Aib2,10, Glu(NH-hexyl)16)hGhrelin(1-28)-NH2;
(SEQ ID:
228)
(Aib2,10, Glu(NH-hexyl)3,16)hGhrelin(1-28)-NH2;
(SEQ ID:
229)
(Ser(n-octanoyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
230)
(Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
231)
(Glu(NH-hexyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
232)
(Glu(NH-hexyl)3, Ser(n-octanoyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
233)
(Dap(octanesulfonyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
234)
(Dap(octanesulfonyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
235)
(Dap(octanesulfonyl)3, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
236)
(Dap(octanesulfonyl)3, Ser(n-octanoyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
237)
(Glu(NH-hexyl)3, Dap(octanesulfonyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
238)
(Cys(S—(CH2)9CH3)17)hGhrelin(1-28)-NH2;
(SEQ ID:
239)
(Cys(S—(CH2)9CH3)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
240)
(Glu(NH-hexyl)3, Cys(S—(CH2)9CH3)17)hGhrelin(1-28)-NH2;
(SEQ ID:
241)
(Cys(S—(CH2)9CH3)3, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
242)
(Cys(S—(CH2)9CH3)3, Ser(n-octanoyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
243)
(Aib2, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
244)
(Aib2, Glu(NH-hexyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
245)
(Aib2, Thz7, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
246)
(Aib2, 4-Hyp7, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
246)
(Aib2, Dhp7, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
246)
(Aib2, Pip7, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
246)
(Aib2, Tic7, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
246)
(Aib2, Glu(NH-hexyl)3,17, Thz7)hGhrelin(1-28)-NH2;
(SEQ ID:
247)
(Aib2, Glu(NH-hexyl)3,17, 4-Hyp7)hGhrelin(1-28)-NH2;
(SEQ ID:
247)
(Aib2, Glu(NH-hexyl)3,17, Dhp7)hGhrelin(1-28)-NH2;
(SEQ ID:
247)
(Aib2, Glu(NH-hexyl)3,17, Pip7)hGhrelin(1-28)-NH2;
(SEQ ID:
247)
(Aib2, Glu(NH-hexyl)3,17, Tic7)hGhrelin(1-28)-NH2;
(SEQ ID:
247)
(Aib2,8, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
248)
(Aib2,8, Glu(NH-hexyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
249)
(Aib2, 3-Pal9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
250)
(Aib2, 4-Pal9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
250)
(Aib2, Taz9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
250)
(Aib2, 2-Thi9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
250)
(Aib2, Glu(NH-hexyl)3,17, 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
251)
(Aib2, Glu(NH-hexyl)3,17, 4-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
251)
(Aib2, Glu(NH-hexyl)3,17, Taz9)hGhrelin(1-28)-NH2;
(SEQ ID:
251)
(Aib2, Glu(NH-hexyl)3,17, 2-Thi9)hGhrelin(1-28)-NH2;
(SEQ ID:
251)
(Aib2,10, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
252)
(Aib2,10, Glu(NH-hexyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
253)
(Aib8, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
254)
(Taz9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
255)
(3-Pal9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
255)
(4-Pal9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
255)
(2-Thi9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
255)
(Glu(NH-hexyl)3,17, Aib8)hGhrelin(1-28)-NH2;
(SEQ ID:
256)
(Glu(NH-hexyl)3,17, Taz9)hGhrelin(1-28)-NH2;
(SEQ ID:
257)
(Glu(NH-hexyl)3,17, 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
257)
(Glu(NH-hexyl)3,17, 4-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
257)
(Glu(NH-hexyl)3,17, 2-Thi9)hGhrelin(1-28)-NH2;
(SEQ ID:
257)
(Aib1,2,10, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
258)
(Aib1,2,10, Glu(NH-hexyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
259)
(A5c2, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
260)
(A5c2, Glu(NH-hexyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
261)
(Glu(1-heptanol)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
262)
(Asp (1-heptanol)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
263)
(Glu(NH-hexyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
264)
(Asp(NH-hexyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
265)
(Aib2, Glu(NH-hexyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
266)
(Lys(biotinyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
267)
(Ser(n-octanoyl)18)hGhrelin(1-28)-NH2;
(SEQ ID:
268)
(Glu(NH-hexyl)18)hGhrelin(1-28)-NH2;
(SEQ ID:
269)
(Glu(NH-hexyl)3,18)hGhrelin(1-28)-NH2;
(SEQ ID:
270)
(Glu(NH-hexyl)3, Ser(n-octanoyl)18)hGhrelin(1-28)-NH2;
(SEQ ID:
271)
(Aib2, Glu(NH-hexyl)18)hGhrelin(1-28)-NH2;
(SEQ ID:
272)
(Aib2, Glu(NH-hexyl)3,18)hGhrelin(1-28)-NH2;
(SEQ ID:
273)
(Aib2,8, Glu(NH-hexyl)18)hGhrelin(1-28)-NH2;
(SEQ ID:
274)
(Aib2,8, Glu(NH-hexyl)3,18)hGhrelin(1-28)-NH2;
(SEQ ID:
275)
(Aib2,10, Glu(NH-hexyl)18)hGhrelin(1-28)-NH2;
(SEQ ID:
276)
(Aib2,10, Glu(NH-hexyl)3,18)hGhrelin(1-28)-NH2;
(SEQ ID:
277)
(Ser(n-octanoyl)19)hGhrelin(1-28)-NH2;
(SEQ ID:
278)
(Glu(NH-hexyl)19)hGhrelin(1-28)-NH2;
(SEQ ID:
279)
(Glu(NH-hexyl)3,19)hGhrelin(1-28)-NH2;
(SEQ ID:
280)
(Glu(NH-hexyl)3, Ser(n-octanoyl)19)hGhrelin(1-28)-NH2;
(SEQ ID:
281)
(Aib2, Glu(NH-hexyl)19)hGhrelin(1-28)-NH2;
(SEQ ID:
282)
(Aib2, Glu(NH-hexyl)3,19)hGhrelin(1-28)-NH2;
(SEQ ID:
283)
(Aib2,8, Glu(NH-hexyl)19)hGhrelin(1-28)-NH2;
(SEQ ID:
284)
(Aib2,8, Glu(NH-hexyl)3,19)hGhrelin(1-28)-NH2;
(SEQ ID:
285)
(Aib2,10, Glu(NH-hexyl)19)hGhrelin(1-28)-NH2;
(SEQ ID:
286)
(Aib2,10, Glu(NH-hexyl)3,19)hGhrelin(1-28)-NH2;
(SEQ ID:
287)
(Ser(n-octanoyl)20)hGhrelin(1-28)-NH2;
(SEQ ID:
288)
(Glu(NH-hexyl)20)hGhrelin(1-28)-NH2;
(SEQ ID:
289)
(Glu(NH-hexyl)3,20)hGhrelin(1-28)-NH2;
(SEQ ID:
290)
(Glu(NH-hexyl)3, Ser(n-octanoyl)20)hGhrelin(1-28)-NH2;
(SEQ ID:
291)
(Aib2, Glu(NH-hexyl)21hGhrelin(1-28)-NH2;
(SEQ ID:
292)
(Aib2, Glu(NH-hexyl)3,20)hGhrelin(1-28)-NH2;
(SEQ ID:
293)
(Aib2,8, Glu(NH-hexyl)9hGhrelin(1-28)-NH2;
(SEQ ID:
294)
(Aib2,8, Glu(NH-hexyl)3,20)hGhrelin(1-28)-NH2;
(SEQ ID:
295)
(Aib2,10, Glu(NH-hexyl)2,20)hGhrelin(1-28)-NH2;
(SEQ ID:
296)
(Aib2,10, Glu(NH-hexyl)3,20)hGhrelin(1-28)-NH2;
(SEQ ID:
297)
(Ac-Gly1, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
298)
(Ac-Gly1, Ser(n-octanoyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
299)
(Ac-Gly1, Glu(NH-hexyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
300)
Glu(NH-hexyl)3, Ser(n-octanoyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
301)
(Ac-Gly1, Dap(octanesulfonyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
302)
(Ac-Gly1, Dap(octanesulfonyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
303)
Dap(octanesulfonyl)3, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
304)
(Ac-Gly1, Dap(octanesulfonyl)3, Ser(n-octanoyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
305)
(Ac-Gly1, Glu(NH-hexyl)3, Dap(octanesulfonyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
306)
(Ac-Gly1, Cys(S—(CH2)9CH3)17)hGhrelin(1-28)-NH2;
(SEQ ID:
307)
(Ac-Gly1, Cys(S—(CH2)9CH3)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
308)
(Ac-Gly1, Glu(NH-hexyl)3, Cys(S—(CH2)9CH3)17)hGhrelin(1-28)-NH2;
(SEQ ID:
309)
(Ac-Gly1, Cys(S—(CH2)9CH3)3, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
310)
(Ac-Gly1, Cys(S—(CH2)9CH3)3, Ser(n-octanoyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
311)
(Ac-Gly1, Aib2, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
312)
(Ac-Gly1, Aib2, Thz7, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
313)
(Ac-Gly1, Aib2, 4-Hyp7, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
313)
(Ac-Gly1, Aib2, Dhp7, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
313)
(Ac-Gly1, Aib2, Pip7, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
313)
(Ac-Gly1, Aib2, Tic7, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
313)
(Ac-Gly1, Aib2, Glu(NH-hexyl)3,17, Thz7)hGhrelin(1-28)-NH2;
(SEQ ID:
314)
(Ac-Gly1, Aib2, Glu(NH-hexyl)3,17, 4-Hyp7)hGhrelin(1-28)-NH2;
(SEQ ID:
314)
(Ac-Gly1, Aib2, Glu(NH-hexyl)3,17, Dhp7)hGhrelin(1-28)-NH2;
(SEQ ID:
314)
(Ac-Gly1, Aib2, Glu(NH-hexyl)3,17, Pip7)hGhrelin(1-28)-NH2;
(SEQ ID:
314)
(Ac-Gly1, Aib2, Glu(NH-hexyl)3,17, Tic7)hGhrelin(1-28)-NH2;
(SEQ ID:
314)
(Ac-Gly1, Aib2,8, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
315)
(Ac-Gly1, Aib2, 3-Pal9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
316)
(Ac-Gly1, Aib2, 4-Pal9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
316)
(Ac-Gly1, Aib2, Taz9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
316)
(Ac-Gly1, Aib2, 2-Thi9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
316)
(Ac-Gly1, Aib2, Glu(NH-hexyl)3,17, 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
317)
(Ac-Gly1, Aib2, Glu(NH-hexyl)3,17, 4-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
317)
(Ac-Gly1, Aib2, Glu(NH-hexyl)3,17, Taz9)hGhrelin(1-28)-NH2;
(SEQ ID:
317)
(Ac-Gly1, Aib2, Glu(NH-hexyl)3,17, 2-Thi9)hGhrelin(1-28)-NH2;
(SEQ ID:
317)
(Ac-Gly1, Aib2,10, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
318)
(Ac-Gly1, Aib2,10, Glu(NH-hexyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
319)
(Ac-Gly1, Aib8, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
320)
(Ac-Gly1, Taz9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
321)
(Ac-Gly1, 3-Pal9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
321)
(Ac-Gly1, 4-Pal9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
321)
(Ac-Gly1, 2-Thi9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
321)
(Ac-Gly1, Glu(NH-hexyl)3,17, Aib8)hGhrelin(1-28)-NH2;
(SEQ ID:
322)
(Ac-Gly1, Glu(NH-hexyl)3,17, Taz9)hGhrelin(1-28)-NH2;
(SEQ ID:
323)
(Ac-Gly1, Glu(NH-hexyl)3,17, 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
323)
(Ac-Gly1, Glu(NH-hexyl)3,17, 4-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
323)
(Ac-Gly1, Glu(NH-hexyl)3,17, 2-Thi9)hGhrelin(1-28)-NH2;
(SEQ ID:
323)
(Ac-Gly1, Aib Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
324)
(Ac-Gly1, Aib Glu(NH-hexyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
325)
(Ac-Gly1, A5c2, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
326)
(Ac-Gly1, A5c2, Glu(NH-hexyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
327)
(Ac-Gly1, Glu(1-heptanol)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
328)
(Ac-Gly1, Asp(1-heptanol)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
329)
(Ac-Gly1, Glu(NH-hexyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
330)
(Ac-Gly1, Asp(NH-hexyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
331)
(Ac-Gly1, Aib2,10, Glu(NH-hexyl)3, Lys(biotinyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
332)
(Ac-Gly1, Glu(NH-hexyl)15)hGhrelin(1-28)-NH2;
(SEQ ID:
333)
(Ac-Gly1, Ser(n-octanoyl)15)hGhrelin(1-28)-NH2;
(SEQ ID:
334)
(Ac-Gly1, Glu(NH-hexyl)3,15)hGhrelin(1-28)-NH2;
(SEQ ID:
335)
(Ac-Gly1, Glu(NH-hexyl)3, Ser(n-octanoyl)15)hGhrelin(1-28)-NH2;
(SEQ ID:
336)
(Ac-Gly1, Aib2, Glu(NH-hexyl)15)hGhrelin(1-28)-NH2;
(SEQ ID:
337)
(Ac-Gly1, Aib2, Glu(NH-hexyl)3,15)hGhrelin(1-28)-NH2;
(SEQ ID:
338)
(Ac-Gly1, Glu(NH-hexyl)15)hGhrelin(1-28)-NH2;
(SEQ ID:
339)
(Ac-Gly1, Glu(NH-hexyl)3,15)hGhrelin(1-28)-NH2;
(SEQ ID:
340)
(Ac-Gly1, Aib2,10, Glu(NH-hexyl)15)hGhrelin(1-28)-NH2;
(SEQ ID:
341)
(Ac-Gly1, Aib2,10, Glu(NH-hexyl)3,15)hGhrelin(1-28)-NH2;
(SEQ ID:
342)
(Ac-Gly1, Glu(NH-hexyl)16)hGhrelin(1-28)-NH2;
(SEQ ID:
343)
(Ac-Gly1, Ser(n-octanoyl)16)hGhrelin(1-28)-NH2;
(SEQ ID:
344)
(Ac-Gly1, Glu(NH-hexyl)3,16)hGhrelin(1-28)-NH2;
(SEQ ID:
345)
(Ac-Gly1, Glu(NH-hexyl)3, Ser(n-octanoyl)16)hGhrelin(1-28)-NH2;
(SEQ ID:
346)
(Ac-Gly1, Aib2, Glu(NH-hexyl)16)hGhrelin(1-28)-NH2;
(SEQ ID:
347)
(Ac-Gly1, Aib2, Glu(NH-hexyl)3,16)hGhrelin(1-28)-NH2;
(SEQ ID:
348)
(Ac-Gly1, Glu(NH-hexyl)16)hGhrelin(1-28)-NH2;
(SEQ ID:
349)
(Ac-Gly1, Glu(NH-hexyl)3,16)hGhrelin(1-28)-NH2;
(SEQ ID:
350)
(Ac-Gly1, Aib2,10, Glu(NH-hexyl)16)hGhrelin(1-28)-NH2;
(SEQ ID:
351)
(Ac-Gly1, Aib2,10, Glu(NH-hexyl)3,16)hGhrelin(1-28)-NH2;
(SEQ ID:
352)
(Ac-Gly1, Glu(NH-hexyl)18)hGhrelin(1-28)-NH2;
(SEQ ID:
353)
(Ac-Gly1, Ser(n-octanoyl)18)hGhrelin(1-28)-NH2;
(SEQ ID:
354)
(Ac-Gly1, Glu(NH-hexyl)3,18)hGhrelin(1-28)-NH2;
(SEQ ID:
355)
(Ac-Gly1, Glu(NH-hexyl)3, Ser(n-octanoyl)18)hGhrelin(1-28)-NH2;
(SEQ ID:
356)
(Ac-Gly1, Aib2, Glu(NH-hexyl)18)hGhrelin(1-28)-NH2;
(SEQ ID:
357)
(Ac-Gly1, Aib2, Glu(NH-hexyl)3,18)hGhrelin(1-28)-NH2;
(SEQ ID:
358)
(Ac-Gly1, Glu(NH-hexyl)18)hGhrelin(1-28)-NH2;
(SEQ ID:
359)
(Ac-Gly1, Glu(NH-hexyl)3,18)hGhrelin(1-28)-NH2;
(SEQ ID:
360)
(Ac-Gly1, Aib2,10, Glu(NH-hexyl)18)hGhrelin(1-28)-NH2;
(SEQ ID:
361)
(Ac-Gly1, Aib2,10, Glu(NH-hexyl)3,18)hGhrelin(1-28)-NH2;
(SEQ ID:
362)
(Ac-Gly1, Glu(NH-hexyl)19)hGhrelin(1-28)-NH2;
(SEQ ID:
363)
(Ac-Gly1, Ser(n-octanoyl)19)hGhrelin(1-28)-NH2;
(SEQ ID:
364)
(Ac-Gly1, Glu(NH-hexyl)3,19)hGhrelin(1-28)-NH2;
(SEQ ID:
365)
(Ac-Gly1, Glu(NH-hexyl)3, Ser(n-octanoyl)19)hGhrelin(1-28)-NH2;
(SEQ ID:
366) (Ac-Gly1, Aib2, Glu(NH-hexyl)19)hGhrelin(1-28)-NH2;
(SEQ ID:
367)
(Ac-Gly1, Aib2, Glu(NH-hexyl)3,19)hGhrelin(1-28)-NH2;
(SEQ ID:
368)
(Ac-Gly1, Glu(NH-hexyl)19)hGhrelin(1-28)-NH2;
(SEQ ID:
369)
(Ac-Gly1, Glu(NH-hexyl)3,19)hGhrelin(1-28)-NH2;
(SEQ ID:
370)
(Ac-Gly1, Aib2,10, Glu(NH-hexyl)19)hGhrelin(1-28)-NH2;
(SEQ ID:
371)
(Ac-Gly1, Aib2,10, Glu(NH-hexyl)3,19)hGhrelin(1-28)-NH2;
(SEQ ID:
372)
(Ac-Gly1, Glu(NH-hexyl)9hGhrelin(1-28)-NH2;
(SEQ ID:
373)
(Ac-Gly1, Ser(n-octanoyl)20)hGhrelin(1-28)-NH2;
(SEQ ID:
374)
(Ac-Gly1, Glu(NH-hexyl)3,20)hGhrelin(1-28)-NH2;
(SEQ ID:
375)
(Ac-Gly1, Glu(NH-hexyl)3, Ser(n-octanoyl)20)hGhrelin(1-28)-NH2;
(SEQ ID:
376)
(Ac-Gly1, Aib2, Glu(NH-hexyl)9hGhrelin(1-28)-NH2;
(SEQ ID:
377)
(Ac-Gly1, Aib2, Glu(NH-hexyl)3,20)hGhrelin(1-28)-NH2;
(SEQ ID:
378)
(Ac-Gly1, Glu(NH-hexyl)20)hGhrelin(1-28)-NH2;
(SEQ ID:
379)
(Ac-Gly1, Glu(NH-hexyl)3,20)hGhrelin(1-28)-NH2;
(SEQ ID:
380)
(Ac-Gly1, Aib2,10, Glu(NH-hexyl)21hGhrelin(1-28)-NH2;
(SEQ ID:
381)
(Ac-Gly1, Aib2,10, Glu(NH-hexyl)3,20)hGhrelin(1-28)-NH2;
(SEQ ID:
382)
(Ac-Gly1, Aib Glu(NH-hexyl)3)hGhrelin(1-28)-NH2;
(SEQ ID:
385)
(1-Apc1, Aib2,10, Glu(NH-hexyl)3)-hGhrelin(1-28)NH2;
(SEQ ID:
385)
(Inp1)hGhrelin(1-28)-NH2;
(SEQ ID:
386)
(Inp1, Aib2)hGhrelin(1-28)-NH2;
(SEQ ID:
386)
(Inp1, Aib2, Glu(NH-hexyl)3)hGhrelin(1-28)-NH2;
(SEQ ID:
387)
(Inp1, Aib2,10)hGhrelin(1-28)-NH2;
(SEQ ID:
388)
(Inp1, Aib2,8)hGhrelin(1-28)-NH2;
(SEQ ID:
389)
(Inp1, Aib2, Ser(n-octanoyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
390)
(Inp1, Ser(n-octanoyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
390)
(Inp1, Aib2,8, Ser(n-octanoyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
389)
Ac-(Inp1, Aib Glu(NH-hexyl)3)hGhrelin(1-28)-NH2;
Ac-(1-Apc1, Aib2,10, Glu(NH-hexyl)3)hGhrelin(1-28)-NH2;
(Asp3(NH-heptyl))hGhrelin(1-28)-NH2;
(SEQ ID:
391)
(des-Ser2)hGhrelin(1-28)-NH2;
(SEQ ID:
392)
(des-Gly1, des-Ser2)hGhrelin(1-28)-NH2;
(SEQ ID:
392)
(Aib1)hGhrelin(1-28)-NH2;
(SEQ ID:
393)
(Asp3(O-hexyl))hGhrelin(1-28)-NH2;
(SEQ ID:
394)
Ser3)hGhrelin(1-28)-NH2;
(SEQ ID:
395)
(A5c5, Ser3)hGhrelin(1-28)-NH2;
(SEQ ID:
396)
(Aib2′4, Sera, 4-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
397)
(n-octanoyl-Gly1, Ser3)hGhrelin(1-28)-NH2;
(SEQ ID:
398)
(isobutyryl-Gly1, Ser3)hGhrelin(1-28)-NH2;
(SEQ ID:
398)
(n-butyryl-Gly1, Ser3)hGhrelin(1-28)-NH2;
(SEQ ID:
398)
(Aib1, Thr3)hGhrelin(1-28)-NH2;
(SEQ ID:
395)
(Aib2,4, Thr3, 4-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
397)
(n-octanoyl-Gly1, Thr3)hGhrelin(1-28)-NH2;
(SEQ ID:
399)
(isobutyryl-Gly1, Thr3)hGhrelin(1-28)-NH2;
(SEQ ID:
399)
(n-butyryl-Gly1, Thr3)hGhrelin(1-28)-NH2;
(SEQ ID:
399)
(Ac-Gly1)hGhrelin(1-28)-NH2;
(SEQ ID:
400)
(Ac-Gly1, Ser3)hGhrelin(1-28)-NH2, (SEQ ID:
400)
(Aib2, Lys(myristyl)17)hGhrelin-(1-28)-NH2;
and (SEQ ID:
383)
[Gly(myristyl)1, Aib2, Lys(myristyl)17]hGhrelin-(1-28)-NH2;
(SEQ ID:
384)
or a pharmaceutically acceptable salt thereof.

3,107 more elements

Dependencies are inferred from the claim text.

Facts

Application: 15/636,684Filed 29 Jun 2017
Priority: 8 Aug 2007
Published: 26 Oct 2017
Term ends: Not estimatedThe source records don’t support an estimate.

Classification53 codes

A61K 38/22
From animals; from humans: hormones
A61K 38/05
Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof: dipeptides
A61K 38/06
Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof: tripeptides
A61K 38/25
Hormones: growth hormone-releasing factor [GH-RF], i.e. somatoliberin

Family

Application60/963,951Us provisional application · filed 8 Aug 2007
Application12/672,681Continuation · filed 8 Feb 2010
Application14/524,088Continuation · filed 27 Oct 2014
Application14/997,678Division · filed 18 Jan 2016
Application15/636,684Division
Application14/997,678Continuation
US 2011/0160133 A1Published application
US 2015/0111823 A1Published application
US 2016/0206700 A1Published application
US 8,871,706 B2Related patent
US 2017/0304403 A1This patent

From the US filing history. Foreign family members aren’t listed.

Timeline

Citations

Open elsewhere

Abstract

(Dap3(octanesulfonyl))hGhrelin(1-28)-NH2;
(SEQ ID:
6)
(Aib2, A6c5)hGhrelin(1-28)-NH2;
(SEQ ID:
7)
(A6c5)hGhrelin(1-28)-NH2;
(SEQ ID:
8)
(Aib2,6)hGhrelin(1-28)-NH2;
(SEQ ID:
9)
(Aib2, A5c12)hGhrelin(1-28)-NH2;
(SEQ ID:
10)
(Aib2, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
11)
(Aib2, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
12)
(Aib2, Act6)hGhrelin(1-28)-NH2;
(SEQ ID:
9)
(Aib2, 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
13)
(Aib2, Dmt7)hGhrelin(1-28)-NH2;
(SEQ ID:
14)
(Aib2, Thz7)hGhrelin(1-28)-NH2;
(SEQ ID:
14)
(A5c2)hGhrelin(1-28)-NH2;
(SEQ ID:
15)
(Act2)hGhrelin(1-28)-NH2;
(SEQ ID:
15)
(Aib2, A5c5)hGhrelin(1-28)-NH2;
(SEQ ID:
7)
(Aib2, A6c5)hGhrelin(1-28)-NH2;
(SEQ ID:
7)
(Aib2,5)hGhrelin(1-28)-NH2;
(SEQ ID:
7)
(Aib2, hLeu5)hGhrelin(1-28)-NH2;
(SEQ ID:
7)
(Aib2, Cha5)hGhrelin(1-28)-NH2;
(SEQ ID:
7)
(Aib2,6)hGhrelin(1-28)-NH2;
(SEQ ID:
9)
(Aib2,Act6)hGhrelin(1-28)-NH2;
(SEQ ID:
9)
(Aib2, Thr6)hGhrelin(1-28)-NH2;
(SEQ ID:
9)
(Aib2, Abu6)hGhrelin(1-28)-NH2;
(SEQ ID:
9)
(Aib2, 4-Hyp7)hGhrelin(1-28)-NH2;
(SEQ ID:
14)
(Aib2,Thz7)hGhrelin(1-28)-NH2;
(SEQ ID:
14)
(Aib2, Pip7)hGhrelin(1-28)-NH2;
(SEQ ID:
14)
(Aib2, Dhp7)hGhrelin(1-28)-NH2;
(SEQ ID:
14)
(Aib2, Ktp7)hGhrelin(1-28)-NH2;
(SEQ ID:
14)
(Aib2,8)hGhrelin(1-28)-NH2;
(SEQ ID:
16)
(Aib2, 2-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
13)
(Aib2, 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
13)
(Aib2, 4-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
13)
(Aib2, Taz9)hGhrelin(1-28)-NH2;
(SEQ ID:
13)
(Aib2, 2-Thi9)hGhrelin(1-28)-NH2;
(SEQ ID:
13)
(Aib2, 2-Fua9)hGhrelin(1-28)-NH2;
(SEQ ID:
13)
(Aib2, Apc9)hGhrelin(1-28)-NH2;
(SEQ ID:
13)
(Aib2,9)hGhrelin(1-28)-NH2;
(SEQ ID:
13)
(Aib2,10)hGhrelin(1-28)-NH2;
(SEQ ID:
17)
(Aib2, Tic7)hGhrelin(1-28)-NH2;
(SEQ ID:
14)
(Aib6)hGhrelin(1-28)-NH2;
(SEQ ID:
18)
(A5c5)hGhrelin(1-28)-NH2;
(SEQ ID:
8)
(A6c5)hGhrelin(1-28)-NH2;
(SEQ ID:
8)
(Act6)hGhrelin(1-28)-NH2;
(SEQ ID:
18)
(3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
19)
(Dmt7)hGhrelin(1-28)-NH2;
(SEQ ID:
20)
(Thz7)hGhrelin(1-28)-NH2;
(SEQ ID:
20)
(Aib5)hGhrelin(1-28)-NH2;
(SEQ ID:
8)
(hLeu5)hGhrelin(1-28)-NH2;
(SEQ ID:
8)
(Cha5)hGhrelin(1-28)-NH2;
(SEQ ID:
8)
(Thr6)hGhrelin(1-28)-NH2;
(SEQ ID:
18)
(Abu6)hGhrelin(1-28)-NH2;
(SEQ ID:
18)
(4-Hyp7)hGhrelin(1-28)-NH2;
(SEQ ID:
20)
(Pip7)hGhrelin(1-28)-NH2;
(SEQ ID:
20)
(Dhp7)hGhrelin(1-28)-NH2;
(SEQ ID:
20)
(Ktp7)hGhrelin(1-28)-NH2;
(SEQ ID:
20)
(Aib8)hGhrelin(1-28)-NH2;
(SEQ ID:
21)
(2-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
19)
(4-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
19)
(Taz9)hGhrelin(1-28)-NH2;
(SEQ ID:
19)
(2-Thi9)hGhrelin(1-28)-NH2;
(SEQ ID:
19)
(2-Fua9)hGhrelin(1-28)-NH2;
(SEQ ID:
19)
(Apc9)hGhrelin(1-28)-NH2;
(SEQ ID:
19)
(Aib9)hGhrelin(1-28)-NH2;
(SEQ ID:
19)
(Aib10)hGhrelin(1-28)-NH2;
(SEQ ID:
22)
(Aib2, Dap3(octanesulfonyl), A6c5)hGhrelin(1-28)-NH2;
(SEQ ID:
23)
(Dap3(octanesulfonyl), A6c5)hGhrelin(1-28)-NH2;
(SEQ ID:
24)
(Aib2,6, Dap3(octanesulfonyl))hGhrelin(1-28)-NH2;
(SEQ ID:
25)
(Aib2, Dap3(octanesulfonyl), A5c12)hGhrelin(1-28)-NH2;
(SEQ ID:
26)
(Aib2, Dap3(octanesulfonyl), A5c12,Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
27)
(Aib2, Dap3(octanesulfonyl), A5c12,Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
28)
(Aib2, Dap3(octanesulfonyl), Act6)hGhrelin(1-28)-NH2;
(SEQ ID:
25)
(Aib2, Dap3(octanesulfonyl), 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
29)
(Aib2, Dap3(octanesulfonyl), Dmt7)hGhrelin(1-28)-NH2;
(SEQ ID:
30)
(Aib2, Dap3(octanesulfonyl), Thz7)hGhrelin(1-28)-NH2;
(SEQ ID:
30)
(A5c2, Dap3(octanesulfonyl))hGhrelin(1-28)-NH2;
(SEQ ID:
31)
(Acte, Dap3(octanesulfonyl))hGhrelin(1-28)-NH2;
(SEQ ID:
31)
(Aib2, Dap3(octanesulfonyl), A5c5)hGhrelin(1-28)-NH2;
(SEQ ID:
32)
(Aib2,5, Dap3(octanesulfonyl))hGhrelin(1-28)-NH2;
(SEQ ID:
32)
(Aib2, Dap3(octanesulfonyl), hLeu5)hGhrelin(1-28)-NH2;
(SEQ ID:
32)
(Aib2, Dap3(octanesulfonyl), Cha5)hGhrelin(1-28)-NH2;
(SEQ ID:
32)
(Aib2,6, Dap3(octanesulfonyl))hGhrelin(1-28)-NH2;
(SEQ ID:
25)
(Aib2, Dap3(octanesulfonyl), Thr6)hGhrelin(1-28)-NH2;
(SEQ ID:
25)
(Aib2, Dap3(octanesulfonyl), Abu6)hGhrelin(1-28)-NH2;
(SEQ ID:
25)
(Aib2, Dap3(octanesulfonyl), 4-Hyp7)hGhrelin(1-28)-NH2;
(SEQ ID:
30)
(Aib2, Dap3(octanesulfonyl), Pip7)hGhrelin(1-28)-NH2;
(SEQ ID:
30)
(Aib2, Dap3(octanesulfonyl), Dhp7)hGhrelin(1-28)-NH2;
(SEQ ID:
30)
(Aib2, Dap3(octanesulfonyl), Ktp7)hGhrelin(1-28)-NH2;
(SEQ ID:
30)
(Aib2,8, Dap3(octanesulfonyl))hGhrelin(1-28)-NH2;
(SEQ ID:
33)
(Aib2, Dap3(octanesulfonyl), 2-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
29)
(Aib2, Dap3(octanesulfonyl), 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
29)
(Aib2, Dap3(octanesulfonyl), 4-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
29)
(Aib2, Dap3(octanesulfonyl), Taz9)hGhrelin(1-28)-NH2;
(SEQ ID:
29)
(Aib2, Dap3(octanesulfonyl), 2-Thi9)hGhrelin(1-28)-NH2;
(SEQ ID:
29)
(Aib2, Dap3(octanesulfonyl), 2-Fua9)hGhrelin(1-28)-NH2;
(SEQ ID:
29)
(Aib2, Dap3(octanesulfonyl), Apc9)hGhrelin(1-28)-NH2;
(SEQ ID:
29)
(Aib2,9, Dap3(octanesulfonyl))hGhrelin(1-28)-NH2;
(SEQ ID:
29)
(Aib2,10, Dap3(octanesulfonyl))hGhrelin(1-28)-NH2;
(SEQ ID:
34)
(Dap3(octanesulfonyl), A6c5)hGhrelin(1-28)-NH2;
(SEQ ID:
24)
(Dap3(octanesulfonyl), Aib6)hGhrelin(1-28)-NH2;
(SEQ ID:
35)
(Dap3(octanesulfonyl), A5c12)hGhrelin(1-28)-NH2;
(SEQ ID:
36)
(Dap3(octanesulfonyl), A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
37)
(Dap3(octanesulfonyl), A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
38)
(Dap3(octanesulfonyl), Act6)hGhrelin(1-28)-NH2;
(SEQ ID:
35)
(Dap3(octanesulfonyl), 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
39)
(Dap3(octanesulfonyl), Dmt7)hGhrelin(1-28)-NH2;
(SEQ ID:
40)
(Dap3(octanesulfonyl), Thz7)hGhrelin(1-28)-NH2;
(SEQ ID:
40)
(Dap3(octanesulfonyl), A5c5)hGhrelin(1-28)-NH2;
(SEQ ID:
24)
(Dap3(octanesulfonyl), Aib5)hGhrelin(1-28)-NH2;
(SEQ ID:
24)
(Dap3(octanesulfonyl), hLeu5)hGhrelin(1-28)-NH2;
(SEQ ID:
24)
(Dap3(octanesulfonyl), Cha5)hGhrelin(1-28)-NH2;
(SEQ ID:
24)
(Dap3(octanesulfonyl), Thr6)hGhrelin(1-28)-NH2;
(SEQ ID:
35)
(Dap3(octanesulfonyl), Abu6)hGhrelin(1-28)-NH2;
(SEQ ID:
35)
(Dap3(octanesulfonyl), 4-Hyp7)hGhrelin(1-28)-NH2;
(SEQ ID:
40)
(Dap3(octanesulfonyl), Pip7)hGhrelin(1-28)-NH2;
(SEQ ID:
40)
(Dap3(octanesulfonyl), Dhp7)hGhrelin(1-28)-NH2;
(SEQ ID:
40)
(Dap3(octanesulfonyl), Ktp7)hGhrelin(1-28)-NH2;
(SEQ ID:
40)
(Dap3(octanesulfonyl), Aib8)hGhrelin(1-28)-NH2;
(SEQ ID:
41)
(Dap3(octanesulfonyl), 2-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
39)
(Dap3(octanesulfonyl), 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
39)
(Dap3(octanesulfonyl), 4-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
39)
(Dap3(octanesulfonyl), Taz9)hGhrelin(1-28)-NH2;
(SEQ ID:
39)
(Dap3(octanesulfonyl), 2-Thi9)hGhrelin(1-28)-NH2;
(SEQ ID:
39)
(Dap3(octanesulfonyl), 2-Fua9)hGhrelin(1-28)-NH2;
(SEQ ID:
39)
(Dap3(octanesulfonyl), Apc9)hGhrelin(1-28)-NH2;
(SEQ ID:
39)
(Dap3(octanesulfonyl), Aib9)hGhrelin(1-28)-NH2;
(SEQ ID:
39)
(Dap3(octanesulfonyl), Aib10hGhrelin(1-28)-NH2;
(SEQ ID:
42)
(Dap3(octanesulfonyl), A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
37)
(Dab3(octanesulfonyl), A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
37)
(Aib2, A6c5, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
43)
(A6c5, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
44)
(Aib2,6, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
45)
(Aib2, Actio, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
45)
(Aib2, 3-Pal9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
46)
(Aib2, Dmt7, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
47)
(Aib2, Thz7, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
47)
(Aib2, A5c5, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
43)
(Aib2,5, A5c12,Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
43)
(Aib2, hLeu5, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
43)
(Aib2, Cha5, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
43)
(Aib2,6, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
45)
(Aib2, Thr6, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
45)
(Aib2, Abu6, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
45)
(Aib2, 4-Hyp', A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
47)
(Aib2, Pip', A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
47)
(Aib2, Dhp7, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
47)
(Aib2, Ktp7, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
47)
(Aib2,8, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
48)
(Aib2, 2-Pal9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
46)
(Aib2, 3-Pal9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
46)
(Aib2, 4-Pal9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
46)
(Aib2, Taz9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
46)
(Aib2, 2-Thi9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
46)
(Aib2, 2-Fua9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
46)
(Aib2, Apc9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
46)
(Aib2,9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
46)
(Aib2,10, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
49)
(Dap3(octanesulfonyl), A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
38)
(Dab3(octanesulfonyl), A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
38)
(Aib2, A6c5, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
50)
(A6c5, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
51)
(Aib2,6, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
52)
(Aib2, Actio, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
52)
(Aib2, 3-Pal9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
53)
(Aib2, Dmt7, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
54)
(Aib2, Thz7, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
54)
(Aib2, A5c5,12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
50)
(Aib2,5, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
50)
(Aib2, hLeu5, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
50)
(Aib2, Cha5, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
50)
(Aib2,6, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
52)
(Aib2, Thr6, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
52)
(Aib2, Abu6, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
52)
(Aib2, 4-Hyp', A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
54)
(Aib2, Pip', A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
54)
(Aib2, Dhp7, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
54)
(Aib2, Ktp7, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
54)
(Aib2,8, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
55)
(Aib2, 2-Pal9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
53)
(Aib2, 3-Pal9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
53)
(Aib2, 4-Pal9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
53)
(Aib2, Taz9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
53)
(Aib2, 2-Thi9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
53)
(Aib2, 2-Fua9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
53)
(Aib2, Apc9,16, A5c12)hGhrelin(1-28)-NH2;
(SEQ ID:
53)
(Aib2,9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
53)
(Aib2,10, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
56)
(A6c5, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
44)
(Aib6, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
57)
(Act6, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
57)
(3-Pal9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
58)
(Dmt7, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
59)
(Thz7, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
59)
(A5c5,12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
44)
(Aib5, A5c12,Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
44)
(hLeu5, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
44)
(Cha5, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
44)
(Aib6, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
57)
(Thr6, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
57)
(Abu6, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
57)
(4-Hyp', A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
59)
(Pip7, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
59)
(Dhp7, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
59)
(Ktp7, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
59)
(Aib8, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
60)
(2-Pal9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
58)
(3-Pal9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
58)
(4-Pal9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
58)
(Taz9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
58)
(2-Thi9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
58)
(2-Fua9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
58)
(Apc9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
58)
(Aib9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
58)
(Aib10, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
61)
(Aib6, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
62)
(A5c5,12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
51)
(Actio, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
62)
(3-Pal9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
63)
(Dmt7, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
64)
(Thz7, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
64)
(Aib5, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
51)
(hLeu5, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
51)
(Cha5, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
51)
(Thr6, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
62)
(Abu6, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
62)
(4-Hyp A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
64)
(Pip7, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
64)
(Dhp7, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
64)
(Ktp7, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
64)
(Aib8, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
65)
(2-Pal9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
63)
(3-Pal9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
63)
(4-Pal9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
63)
(Taz9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
63)
(2-Thi9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
63)
(2-Fua9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
63)
(Apc9,16, A5c12)hGhrelin(1-28)-NH2;
(SEQ ID:
63)
(Aib9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
63)
(Aib10, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
66)
(Aib2, Glu3(NH-hexyl), A6c5)hGhrelin(1-28)-NH2;
(SEQ ID:
67)
(Glu3(NH-hexyl), A6c5)hGhrelin(1-28)-NH2;
(SEQ ID:
68)
(Aib2,6, Glu3(NH-hexyl))hGhrelin(1-28)-NH2;
(SEQ ID:
69)
(Aib2, Glu3(NH-hexyl), Act6)hGhrelin(1-28)-NH2;
(SEQ ID:
69)
(Aib2, Glu3(NH-hexyl), 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
70)
(Aib2, Glu3(NH-hexyl), Dmt7)hGhrelin(1-28)-NH2;
(SEQ ID:
71)
(Aib2, Glu3(NH-hexyl), Thz7)hGhrelin(1-28)-NH2;
(SEQ ID:
71)
(Aib2, Glu3(NH-hexyl), A5c5)hGhrelin(1-28)-NH2;
(SEQ ID:
67)
(Aib2,5, Glu3(NH-hexyl))hGhrelin(1-28)-NH2;
(SEQ ID:
67)
(Aib2, Glu3(NH-hexyl), hLeu5)hGhrelin(1-28)-NH2;
(SEQ ID:
67)
(Aib2, Cha5)hGhrelin(1-28)-NH2;
(SEQ ID:
7)
(Aib2′6, Glu3(NH-hexyl))hGhrelin(1-28)-NH2;
(SEQ ID:
69)
(Aib2, Glu3(NH-hexyl), Thr6)hGhrelin(1-28)-NH2;
(SEQ ID:
69)
(Aib2, Glu3(NH-hexyl), Abu6)hGhrelin(1-28)-NH2;
(SEQ ID:
69)
(Aib2, Glu3(NH-hexyl), 4-Hyp7)hGhrelin(1-28)-NH2;
(SEQ ID:
71)
(Aib2, Glu3(NH-hexyl), Pip7)hGhrelin(1-28)-NH2;
(SEQ ID:
71)
(Aib2, Glu3(NH-hexyl), Dhp7)hGhrelin(1-28)-NH2;
(SEQ ID:
71)
(Aib2, Glu3(NH-hexyl), Ktp7)hGhrelin(1-28)-NH2;
(SEQ ID:
71)
(Aib2,8, Glu3(NH-hexyl))hGhrelin(1-28)-NH2;
(SEQ ID:
72)
(Aib2, Glu3(NH-hexyl), 2-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
70)
(Aib2, Glu3(NH-hexyl), 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
70)
(Aib2, Glu3(NH-hexyl), 4-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
70)
(Aib2, Glu3(NH-hexyl), Taz9)hGhrelin(1-28)-NH2;
(SEQ ID:
70)
(Aib2, Glu3(NH-hexyl), 2-Thi9)hGhrelin(1-28)-NH2;
(SEQ ID:
70)
(Aib2, Glu3(NH-hexyl), 2-Fua9)hGhrelin(1-28)-NH2;
(SEQ ID:
70)
(Aib2, Glu3(NH-hexyl), Apc9)hGhrelin(1-28)-NH2;
(SEQ ID:
70)
(Aib2,9, Glu3(NH-hexyl))hGhrelin(1-28)-NH2;
(SEQ ID:
70)
(Aib2,10, Glu3(NH-hexyl))hGhrelin(1-28)-NH2;
(SEQ ID:
73)
(Glu3(NH-hexyl), Aib6)hGhrelin(1-28)-NH2;
(SEQ ID:
74)
(Glu3(NH-hexyl), A5c5)hGhrelin(1-28)-NH2;
(SEQ ID:
68)
(Glu3(NH-hexyl), Act6)hGhrelin(1-28)-NH2;
(SEQ ID:
74)
(Glu3(NH-hexyl), 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
75)
(Glu3(NH-hexyl), Dmt7)hGhrelin(1-28)-NH2;
(SEQ ID:
76)
(Glu3(NH-hexyl), Thz7)hGhrelin(1-28)-NH2;
(SEQ ID:
76)
(Glu3(NH-hexyl), Aib5)hGhrelin(1-28)-NH2;
(SEQ ID:
68)
(Glu3(NH-hexyl), hLeu5)hGhrelin(1-28)-NH2;
(SEQ ID:
68)
(Glu3(NH-hexyl), Cha5)hGhrelin(1-28)-NH2;
(SEQ ID:
68)
(Glu3(NH-hexyl), Thr6)hGhrelin(1-28)-NH2;
(SEQ ID:
74)
(Glu3(NH-hexyl), Abu6)hGhrelin(1-28)-NH2;
(SEQ ID:
74)
(Glu3(NH-hexyl), 4-Hyp7)hGhrelin(1-28)-NH2;
(SEQ ID:
76)
(Glu3(NH-hexyl), Pip7)hGhrelin(1-28)-NH2;
(SEQ ID:
76)
(Glu3(NH-hexyl), Dhp7)hGhrelin(1-28)-NH2;
(SEQ ID:
76)
(Glu3(NH-hexyl), Ktp7)hGhrelin(1-28)-NH2;
(SEQ ID:
76)
(Glu3(NH-hexyl), Aib8)hGhrelin(1-28)-NH2;
(SEQ ID:
41)
(Glu3(NH-hexyl), 2-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
75)
(Glu3(NH-hexyl), 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
75)
(Glu3(NH-hexyl), 4-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
75)
(Glu3(NH-hexyl), Taz9)hGhrelin(1-28)-NH2;
(SEQ ID:
75)
(Glu3(NH-hexyl), 2-Thi9)hGhrelin(1-28)-NH2;
(SEQ ID:
75)
(Glu3(NH-hexyl), 2-Fua9)hGhrelin(1-28)-NH2;
(SEQ ID:
75)
(Glu3(NH-hexyl), Apc9)hGhrelin(1-28)-NH2;
(SEQ ID:
75)
(Glu3(NH-hexyl), Aib9)hGhrelin(1-28)-NH2;
(SEQ ID:
75)
(Glu3(NH-hexyl), Aib9hGhrelin(1-28)-NH2;
(SEQ ID:
42)
(Aib2, Glu3(NH-hexyl), A6c5, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
77)
(A6c5, Glu3(NH-hexyl), A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
78)
(Aib2,6, Glu3(NH-hexyl), A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
79)
(Aib2, Glu3(NH-hexyl), Actio, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
79)
(Aib2, Glu3(NH-hexyl), 3-Pal9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
80)
(Aib2, Glu3(NH-hexyl), Dmt7, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
81)
(Aib2, Glu3(NH-hexyl), Thz7, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
81)
(Aib2, Glu3(NH-hexyl), A5c5,12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
77)
(Aib2,5, Glu3(NH-hexyl), A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
77)
(Aib2, hLeu5, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
43)
(Aib2, Glu3(NH-hexyl), Cha5, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
77)
(Aib2,6, Glu3(NH-hexyl), A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
79)
(Aib2, Glu3(NH-hexyl), Thr6, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
79)
(Aib2, Glu3(NH-hexyl), Abu6, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
79)
(Aib2, Glu3(NH-hexyl), 4-Hyp', A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
81)
(Aib2, Glu3(NH-hexyl), Pip', A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
81)
(Aib2, Glu3(NH-hexyl), Dhp7, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
81)
(Aib2, Glu3(NH-hexyl), Ktp7, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
81)
(Aib2,8, Glu3(NH-hexyl), A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
82)
(Aib2, Glu3(NH-hexyl), 2-Pal9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
80)
(Aib2, Glu3(NH-hexyl), 3-Pal9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
80)
(Aib2, Glu3(NH-hexyl), 4-Pal9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
80)
(Aib2, Glu3(NH-hexyl), Taz9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
80)
(Aib2, Glu3(NH-hexyl), 2-Thi9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
80)
(Aib2, Glu3(NH-hexyl), 2-Fua9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
80)
(Aib2, Glu3(NH-hexyl), Apc9, A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
80)
(Aib2,9, Glu3(NH-hexyl), A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
80)
(Aib2,12, Glu3(NH-hexyl), 4-Pal9, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
125)
(Aib2,10, Glu3(NH-hexyl), A5c12, Orn15)hGhrelin(1-28)-NH2;
(SEQ ID:
83)
(Aib2, Glu3(NH-hexyl), A6c5, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
84)
(Glu3(NH-hexyl), A6c5, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
85)
(Aib2,6, Glu3(NH-hexyl), A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
86)
(Aib2, Glu3(NH-hexyl), Act6, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
86)
(Aib2, Glu3(NH-hexyl), 3-Pal9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
87)
(Aib2, Glu3(NH-hexyl), Dmt7, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
88)
(Aib2, Glu3(NH-hexyl), Thz7, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
88)
(Aib2, Glu3(NH-hexyl), A5c5,12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
84)
(Aib2,5, Glu3(NH-hexyl), A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
84)
(Aib2, Glu3(NH-hexyl), hLeu5, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
84)
(Aib2, Glu3(NH-hexyl), Cha5, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
84)
(Aib2,6, Glu3(NH-hexyl), A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
86)
(Aib2, Glu3(NH-hexyl), Thr6, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
86)
(Aib2, Glu3(NH-hexyl), Abu6, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
86)
(Aib2, Glu3(NH-hexyl), 4-Hyp', A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
88)
(Aib2, Glu3(NH-hexyl), Pip', A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
88)
(Aib2, Glu3(NH-hexyl), Dhp7, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
88)
(Aib2, Glu3(NH-hexyl), Ktp7, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
88)
(Aib2,8, Glu3(NH-hexyl), A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
89)
(Aib2, Glu3(NH-hexyl), 2-Pal9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
87)
(Aib2, Glu3(NH-hexyl), 3-Pal9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
87)
(Aib2, Glu3(NH-hexyl), 4-Pal9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
87)
(Aib2, Glu3(NH-hexyl), Taz9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
87)
(Aib2, Glu3(NH-hexyl), 2-Thi9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
87)
(Aib2, Glu3(NH-hexyl), 2-Fua9, A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
87)
(Aib2, Glu3(NH-hexyl), Apc9,16, A5c12)hGhrelin(1-28)-NH2;
(SEQ ID:
87)
(Aib2,9, Glu3(NH-hexyl), A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
87)
(Aib2,10, Glu3(NH-hexyl), A5c12, Apc16)hGhrelin(1-28)-NH2;
(SEQ ID:
90)
(Glu3(O-hexyl))hGhrelin(1-28)-NH2;
(SEQ ID:
91)
(Aib2)hGhrelin(1-28)-NH2;
(SEQ ID:
15)
(Glu3(NH-hexyl))hGhrelin(1-28)-NH2;
(SEQ ID:
91)
(Aib2, Glu3(O-hexyl))hGhrelin(1-28)-NH2;
(SEQ ID:
92)
Glu3(O-hexyl))hGhrelin(1-28)-NH2;
(SEQ ID:
93)
(Aib2, Glu3(NH-hexyl))hGhrelin(1-28)-NH2;
(SEQ ID:
92)
(Dap3(octanesulfonyl))hGhrelin(1-28)-NH2;
(SEQ ID:
6)
(Aib2, Dap3(octanesulfonyl))hGhrelin(1-28)-NH2;
(SEQ ID:
94)
Dap3(octanesulfonyl))hGhrelin(1-28)-NH2;
(SEQ ID:
93)
(Ava2, Dap3(octanesulfonyl))hGhrelin(2-28)-NH2;
(SEQ ID:
126)
(Ac-Gly1)hGhrelin(1-5)-NH2;
(SEQ ID:
95)
(Ac-Gly1)hGhrelin(1-6)-NH2;
(SEQ ID:
96)
(Ac-Gly1)hGhrelin(1-7)-NH2;
(SEQ ID:
97)
(Ac-Gly1, Aib2)hGhrelin(1-28)-NH2;
(SEQ ID:
98)
(Ac-Gly1, Aib2, Glu3(NH-hexyl))hGhrelin(1-5)-NH2;
(SEQ ID:
99)
(Ac-Gly1, Aib2, Glu3(NH-hexyl))hGhrelin(1-6)-NH2;
(SEQ ID:
100)
(Ac-Gly1, Aib2, Glu3(NH-hexyl))hGhrelin(1-7)-NH2;
(SEQ ID:
101)
(Ac-Gly1, Aib2, Glu3(NH-hexyl))hGhrelin(1-28)-NH2;
(SEQ ID:
102)
(Ac-Gly1, Aib2, Glu3(NH-hexyl), Arg8)hGhrelin(1-8)-NH2;
(SEQ ID:
103)
(Ac-Gly1, Aib2, Glu3(NH-hexyl), Lys8)hGhrelin(1-8)-NH2;
(SEQ ID:
103)
(n-butyryl-Gly1)hGhrelin(1-28)-NH2;
(SEQ ID:
104)
(n-butyryl-Gly1, Aib2, Glu3(NH-hexyl))hGhrelin(1-28)-NH2;
(SEQ ID:
105)
(isobutyryl-Gly1)hGhrelin(1-28)-NH2;
(SEQ ID:
104)
(n-octanoyl-Gly1)hGhrelin(1-28)-NH2, (SEQ ID:
104)
Cys3(S(CH2)9CH3)hGhrelin(1-28)-NH2;
(SEQ ID:
106)
(Aib2, Ser3)hGhrelin(1-28)-NH2;
(SEQ ID:
15)
(Aib2,6, Ser3)hGhrelin(1-28)-NH2 (SEQ ID:
9)
(Aib2, Ser3, 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
13)
(Aib2, Ser3, Thz7)hGhrelin(1-28)-NH2;
(SEQ ID:
14)
(Aib2, Ser3, Cha5)hGhrelin(1-28)-NH2;
(SEQ ID:
7)
(Aib2, Ser3, Abu6)hGhrelin(1-28)-NH2;
(SEQ ID:
9)
(Aib2, Ser3, 4-Hyp7)hGhrelin(1-28)-NH2;
(SEQ ID:
14)
(Aib2, Ser3, Taz9)hGhrelin(1-28)-NH2;
(SEQ ID:
13)
(Aib2, Ser3, Dhp7)hGhrelin(1-28)-NH2;
(SEQ ID:
14)
(Aib2,8, Ser3)hGhrelin(1-28)-NH2;
(SEQ ID:
16)
(Aib2, Ser3, Pip7)hGhrelin(1-28)-NH2;
(SEQ ID:
14)
(Ac-Gly1, Aib2,10, Ser3)hGhrelin(1-28)-NH2;
(SEQ ID:
107)
(Aib2,10, Ser3)hGhrelin(1-28)-NH2;
(SEQ ID:
17)
(n-butyryl-Gly1, Aib2, Ser3)hGhrelin(1-28)-NH2;
(SEQ ID:
108)
(Ac-Gly1, Aib2, Ser3)hGhrelin(1-28)-NH2;
(SEQ ID:
98)
(Aib2, Ser3, Tic7)hGhrelin(1-28)-NH2;
(SEQ ID:
14)
(Ac-Gly1, Aib2, Ser3, Arg8)hGhrelin(1-28)-NH2;
(SEQ ID:
109)
(Ser3, Aib8)hGhrelin(1-28)-NH2;
(SEQ ID:
110)
(Ser3, Taz9)hGhrelin(1-28)-NH2;
(SEQ ID:
19)
(Ser3, 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
19)
(Ser3, 4-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
19)
(Aib2, Ser3, 2-Thi9)hGhrelin(1-28)-NH2;
(SEQ ID:
13)
(Ser3, 2-Thi9)hGhrelin(1-28)-NH2;
(SEQ ID:
19)
(Ser3, 4-Hyp7)hGhrelin(1-28)-NH2;
(SEQ ID:
20)
(Aib2, Ser3, Tic7)hGhrelin(1-28)-NH2;
(SEQ ID:
14)
(Aib2, Thr3)hGhrelin(1-28)-NH2;
(SEQ ID:
111)
(Aib2,6, Thr3)hGhrelin(1-28)-NH2;
(SEQ ID:
112)
(A5c5, Thr3)hGhrelin(1-28)-NH2;
(SEQ ID:
113)
(Aib2, Thr3, 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
114)
(Aib2, Thr3, Thz7)hGhrelin(1-28)-NH2;
(SEQ ID:
115)
(Aib2, Thr3, Cha5)hGhrelin(1-28)-NH2;
(SEQ ID:
116)
(Aib2, Thr3, Abu6)hGhrelin(1-28)-NH2;
(SEQ ID:
112)
(Aib2, Thr3, 4-Hyp7)hGhrelin(1-28)-NH2;
(SEQ ID:
115)
(Aib2, Thr3, Taz9)hGhrelin(1-28)-NH2;
(SEQ ID:
114)
(Aib2, Thr3, Dhp7)hGhrelin(1-28)-NH2;
(SEQ ID:
115)
(Aib2,8, Thr3)hGhrelin(1-28)-NH2;
(SEQ ID:
117)
(Aib2, Thr3, Pip7)hGhrelin(1-28)-NH2;
(SEQ ID:
115)
(Ac-Gly1, Aib2,10, Thr3)hGhrelin(1-28)-NH2;
(SEQ ID:
118)
(Aib2,10, Thr3)hGhrelin(1-28)-NH2;
(SEQ ID:
118)
(n-butyryl-Gly1, Aib2, Thr3)hGhrelin(1-28)-NH2;
(SEQ ID:
119)
(Ac-Gly1, Aib2, Thr3)hGhrelin(1-28)-NH2;
(SEQ ID:
119)
(Aib2, Thr3, Tic7)hGhrelin(1-28)-NH2;
(SEQ ID:
115)
(Ac-Gly1, Aib2, Thr3, Arg8)hGhrelin(1-28)-NH2;
(SEQ ID:
120)
(Thr3, Aib8)hGhrelin(1-28)-NH2;
(SEQ ID:
121)
(Thr3, Taz9)hGhrelin(1-28)-NH2;
(SEQ ID:
122)
(Thr3, 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
122)
(Thr3, 4-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
122)
(Aib2, Thr3, 2-Thi9)hGhrelin(1-28)-NH2;
(SEQ ID:
114)
(Thr3, 2-Thi9)hGhrelin(1-28)-NH2;
(SEQ ID:
122)
(Thr3, 4-Hyp7)hGhrelin(1-28)-NH2;
(SEQ ID:
123)
(Aib2, Thr3, Tic7)hGhrelin(1-28)-NH2;
(SEQ ID:
115)
(Ac-Gly1, Glu3(NH-hexyl))hGhrelin(1-28)-NH2;
(SEQ ID:
124)
H-Inp-D-1-Nal-D-Trp-3-Pal-Lys-NH2;
(SEQ ID:
128)
H-Inp-D-2-Nal-D-Trp-4-Pal-Lys-NH2;
(SEQ ID:
129)
H-Inp-D-2-Nal-D-Trp-Om-Lys-NH2;
(SEQ ID:
129)
H-Inp-D-Bip-D-Trp-Phe-Lys-NH2;
(SEQ ID:
130)
H-Inp-D-2-Nal-D-Trp-Thr(Bzl)-Lys-NH2;
(SEQ ID:
131)
H-Inp-D-2-Nal-D-Trp-Pff-Lys-NH2;
(SEQ ID:
131)
H-Inp-D-2-Nal-D-Trp-2-Thi-Lys-NH2;
(SEQ ID:
132)
H-Inp-D-2-Nal-D-Trp-Taz-Lys-NH2;
(SEQ ID:
132)
H-Inp-D-Dip-D-Trp-Phe-Lys-NH2;
(SEQ ID:
133)
H-Inp-D-Bpa-D-Trp-Phe-Lys-NH2;
(SEQ ID:
133)
H-Inp-D-2-Nal-D-Bpa-Phe-Lys-NH2;
(SEQ ID:
134)
H-Inp-D-2-Nal-D-Trp-3-Pal-NH2;
(SEQ ID:
135)
H-Inp-D-2-Nal-D-Trp-4-Pal-NH2;
(SEQ ID:
135)
H-Inp-D-1-Nal-D-Trp-3-Pal-NH2;
(SEQ ID:
136)
H-Inp-D-Bip-D-Trp-Phe-NH2;
(SEQ ID:
137)
H-Inp-D-2-Nal-D-Trp-Thr(Bzl)-NH2;
(SEQ ID:
138)
H-Inp-D-2-Nal-D-Trp-Pff-NH2;
(SEQ ID:
138)
H-Inp-D-2-Nal-D-Trp-2-Thi-NH2;
(SEQ ID:
138)
H-Inp-D-2-Nal-D-Trp-Taz-NH2;
(SEQ ID:
138)
H-Inp-D-Dip-D-Trp-Phe-NH2;
(SEQ ID:
139)
H-Inp-D-2-Nal-D-Dip-Phe-NH2;
(SEQ ID:
140)
H-Inp-D-Bal -D-Trp-Phe-NH2;
(SEQ ID:
141)
H-Inp-D-2-Nal-D-Bal -Phe-NH2;
(SEQ ID:
142)
H-Inp-D-2-Nal-D-Trp-3-Pal-Lys-NH2;
(SEQ ID:
143)
H-Inp-D-Trp-D-2-Nal(Ψ)-Pim;
(SEQ ID:
127)
H-Inp-D-Bal -D-Trp-2-Thi-Lys-NH2;
(SEQ ID:
144)
H-Inp-D-Bal -D-Trp-Phe-Lys-NH2;
(SEQ ID:
144)
H-Inp-D-1-Nal-D-Trp-2-Thi-Lys-NH2;
(SEQ ID:
128)
H-Inp-D-2-Nal-D-Trp-Phe-Apc-NH2;
(SEQ ID:
2)
H-Inp-D-1-Nal-D-Trp-Phe-Apc-NH2;
(SEQ ID:
2)
H-Inp-D-Bal-D-Trp-Phe-Apc-NH2;
(SEQ ID:
2)
H-Apc-D-2-Nal-D-Trp-Phe-Lys-NH2;
(SEQ ID:
145)
H-Apc-D-1-Nal-D-Trp-2-Thi-Lys-NH2;
(SEQ ID:
146)
H-Inp-D-1-Nal-D-Trp-2-Thi-NH2;
(SEQ ID:
147)
H-Apc-D-1-Nal-D-Trp-Phe-NH2;
(SEQ ID:
148)
H-Inp-D-2-Nal-D-Trp(Ψ)-Pim;
(SEQ ID:
149)
H-Inp-D-1-Nal-D-Trp(Ψ)-Pim;
(SEQ ID:
149)
H-Inp-D-Bal-D-Trp(Ψ)-Pim;
(SEQ ID:
149)
H-Aib-D-Ser(Bzl)-D-Trp(Ψ)-Pim;
(SEQ ID:
150)
H-Inp-D-1-Nal-D-Trp-Taz-Lys-NH2;
(SEQ ID:
151)
H-Inp-D-Bal -D-Trp-Taz-Lys-NH2;
(SEQ ID:
151)
H-Apc-D-1-Nal-D-Trp-Taz-Lys-NH2;
(SEQ ID:
152)
H-Apc-D-Bal -D-Trp-Taz-Lys-NH2;
(SEQ ID:
152)
H-Apc-D-Bal -D-Trp-2-Thi-Lys-NH2;
(SEQ ID:
153)
H-Apc-D-Bal -D-Trp-Phe-Lys-NH2;
(SEQ ID:
153)
H-Apc-D-1-Nal-D-Trp-Phe-Apc-NH2;
(SEQ ID:
154)
H-Apc-D-Bal -D-Trp-Phe-Apc-NH2;
(SEQ ID:
154)
H-Apc-D-1-Nal-D-1-Nal-Phe-Apc-NH2;
(SEQ ID:
155)
H-Apc-D-1-Nal-D-2-Nal-Phe-Apc-NH2;
(SEQ ID:
155)
H-Apc-D-1-Nal-D-1-Nal-Phe-Lys-NH2;
(SEQ ID:
156)
H-Apc-D-Bal-D-1-Nal-Phe-Apc-NH2;
(SEQ ID:
157)
H-Apc-D-Bal-D-2-Nal-Phe-Apc-NH2;
(SEQ ID:
157)
H-Apc-D-Bal-D-1-Nal-Phe-Lys-NH2;
(SEQ ID:
158)
H-Apc-D-Bal-D-2-Nal-Phe-Lys-NH2;
(SEQ ID:
158)
H-Apc-D-1-Nal-D-Trp-2-Thi-NH2;
(SEQ ID:
159)
H-Apc-D-Bal -D-Trp-Phe-NH2;
(SEQ ID:
160)
H-Apc-D-1-Nal-D-Trp-Taz-NH2;
(SEQ ID:
159)
H-Apc-D-Bal -D-Trp-2-Thi-NH2;
(SEQ ID:
161)
H-Apc-D-Bal -D-Trp-Taz-NH2;
(SEQ ID:
161)
H-Apc-D-2-Nal-D-Trp-2-Thi-NH2;
(SEQ ID:
162)
H-Apc-D-2-Nal-D-Trp-Taz-NH2;
(SEQ ID:
162)
H-Inp-D-1-Nal-D-Trp-Taz-Apc-NH2;
(SEQ ID:
163)
H-Inp-D-Bal-D-Trp-Taz-Apc-NH2;
(SEQ ID:
163)
H-Apc-D-1-Nal-D-Trp-Taz-Apc-NH2;
(SEQ ID:
164)
H-Apc-D-Bal -D-Trp-Taz-Apc-NH2;
(SEQ ID:
164)
H-Apc-D-1-Nal-D-Trp-2-Fua-Apc-NH2;
(SEQ ID:
165)
H-Apc-D-1-Nal-D-Trp-2-Fua-Lys-NH2;
(SEQ ID:
165)
H-Apc-D-1-Nal-D-Trp-2-Fua-NH2;
(SEQ ID:
165)
H-Apc-D-1-Nal-D-Trp-2-Pal-NH2;
(SEQ ID:
166)
H-Apc-D-1-Nal-D-Trp-3-Pal-NH2;
(SEQ ID:
166)
H-Apc-D-1-Nal-D-Trp-3-Thi-Apc-NH2;
(SEQ ID:
167)
H-Apc-D-1-Nal-D-Trp-3-Thi-Lys-NH2;
(SEQ ID:
167)
H-Apc-D-1-Nal-D-Trp-3-Thi-NH2;
(SEQ ID:
168)
H-Apc-D-1-Nal-D-Trp-4-Pal-NH2;
(SEQ ID:
168)
H-Apc-D-1-Nal-D-Trp-Pff-Apc-NH2;
(SEQ ID:
169)
H-Apc-D-1-Nal-D-Trp-Pff-Lys-NH2;
(SEQ ID:
169)
H-Apc-D-1-Nal-D-Trp-Pff-NH2;
(SEQ ID:
168)
H-Apc-D-2-Nal-D-Trp-2-Fua-Apc-NH2;
(SEQ ID:
170)
H-Apc-D-2-Nal-D-Trp-2-Fua-Lys-NH2;
(SEQ ID:
170)
H-Apc-D-2-Nal-D-Trp-2-Fua-NH2;
(SEQ ID:
171)
H-Apc-D-2-Nal-D-Trp-2-Pal-NH2;
(SEQ ID:
171)
H-Apc-D-2-Nal-D-Trp-2-Thi-Apc-NH2;
(SEQ ID:
172)
H-Apc-D-2-Nal-D-Trp-2-Thi-Lys-NH2;
(SEQ ID:
172)
H-Apc-D-2-Nal-D-Trp-3-Pal-NH2;
(SEQ ID:
171)
H-Apc-D-2-Nal-D-Trp-3-Thi-Apc-NH2;
(SEQ ID:
173)
H-Apc-D-2-Nal-D-Trp-3-Thi-Lys-NH2;
(SEQ ID:
173)
H-Apc-D-2-Nal-D-Trp-3-Thi-NH2;
(SEQ ID:
171)
H-Apc-D-2-Nal-D-Trp-4-Pal-NH2;
(SEQ ID:
171)
H-Apc-D-2-Nal-D-Trp-Pff-Apc-NH2;
(SEQ ID:
174)
H-Apc-D-2-Nal-D-Trp-Pff-Lys-NH2;
(SEQ ID:
174)
H-Apc-D-2-Nal-D-Trp-Pff-NH2;
(SEQ ID:
171)
H-Apc-D-2-Nal-D-Trp-Taz-Apc-NH2;
(SEQ ID:
175)
H-Apc-D-2-Nal-D-Trp-Taz-Lys-NH2;
(SEQ ID:
175)
H-Apc-D-Bal -D-Bal -2-Fua-Apc-NH2;
(SEQ ID:
176)
H-Apc-D-Bal -D-Bal -2-Fua-Lys-NH2;
(SEQ ID:
176)
H-Apc-D-Bal -D-Bal -2-Fua-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Bal -2-Pal-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Bal -2-Thi-Apc-NH2;
(SEQ ID:
178)
H-Apc-D-Bal -D-Bal -2-Thi-Lys-NH2;
(SEQ ID:
178)
H-Apc-D-Bal -D-Bal -2-Thi-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Bal -3-Pal-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Bal -3-Thi-Apc-NH2;
(SEQ ID:
179)
H-Apc-D-Bal -D-Bal -3-Thi-Lys-NH2;
(SEQ ID:
179)
H-Apc-D-Bal -D-Bal -3-Thi-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Bal -4-Pal-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Bal -Pff-Apc-NH2;
(SEQ ID:
180)
H-Apc-D-Bal -D-Bal -Pff-Lys-NH2;
(SEQ ID:
180)
H-Apc-D-Bal -D-Bal -Pff-NH2;
(SEQ ID:
177)
H-Apc-D-Bal-D-Bal-Phe-Apc-NH2;
(SEQ ID:
181)
H-Apc-D-Bal -D-Bal -Phe-Lys-NH2;
(SEQ ID:
181)
H-Apc-D-Bal -D-Bal -Phe-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Bal -Taz-Apc-NH2;
(SEQ ID:
182)
H-Apc-D-Bal -D-Bal -Taz-Lys-NH2;
(SEQ ID:
182)
H-Apc-D-Bal -D-Bal -Taz-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Trp-2-Fua-Apc-NH2;
(SEQ ID:
183)
H-Apc-D-Bal -D-Trp-2-Fua-Lys-NH2;
(SEQ ID:
183)
H-Apc-D-Bal -D-Trp-2-Fua-NH2;
(SEQ ID:
184)
H-Apc-D-Bal -D-Trp-2-Pal-NH2;
(SEQ ID:
184)
H-Apc-D-Bal -D-Trp-3-Pal-NH2;
(SEQ ID:
184)
H-Apc-D-Bal -D-Trp-3-Thi-Apc-NH2;
(SEQ ID:
185)
H-Apc-D-Bal -D-Trp-3-Thi-Lys-NH2;
(SEQ ID:
185)
H-Apc-D-Bal -D-Trp-3-Thi-NH2;
(SEQ ID:
184)
H-Apc-D-Bal -D-Trp-4-Pal-NH2;
(SEQ ID:
184)
H-Apc-D-Bal -D-Trp-Pff-Apc-NH2;
(SEQ ID:
186)
H-Apc-D-Bal -D-Trp-Pff-Lys-NH2;
(SEQ ID:
186)
H-Apc-D-Bal -D-Trp-Pff-NH2;
(SEQ ID:
184)
H-Inp-D-1-Nal-D-Bal -2-Fua-Lys-NH2;
(SEQ ID:
187)
H-Inp-D-1-Nal-D-Bal -2-Fua-NH2;
(SEQ ID:
188)
H-Inp-D-1-Nal-D-Bal -2-Thi-Lys-NH2;
(SEQ ID:
187)
H-Inp-D-1-Nal-D-Bal -3-Thi-Lys-NH2;
(SEQ ID:
187)
H-Inp-D-1-Nal-D-Bal -Pff-Lys-NH2;
(SEQ ID:
187)
H-Inp-D-1-Nal-D-Bal -Pff-NH2;
(SEQ ID:
188)
H-Inp-D-1-Nal-D-Bal -Phe-Lys-NH2;
(SEQ ID:
187)
H-Inp-D-1-Nal-D-Bal -Taz-Lys-NH2;
(SEQ ID:
187)
H-Inp-D-1-Nal-D-Bal -Taz-NH2;
(SEQ ID:
188)
H-Inp-D-1-Nal-D-Trp-2-Fua-Apc-NH2;
(SEQ ID:
189)
H-Inp-D-1-Nal-D-Trp-2-Fua-Lys-NH2;
(SEQ ID:
189)
H-Inp-D-1-Nal-D-Trp-2-Fua-NH2;
(SEQ ID:
189)
H-Inp-D-1-Nal-D-Trp-3-Thi-Apc-NH2;
(SEQ ID:
190)
H-Inp-D-1-Nal-D-Trp-3-Thi-Lys-NH2;
(SEQ ID:
190)
H-Inp-D-1-Nal-D-Trp-Pff-Apc-NH2;
(SEQ ID:
191)
H-Inp-D-1-Nal-D-Trp-Pff-Lys-NH2;
(SEQ ID:
191)
H-Inp-D-1-Nal-D-Trp-Pff-NH2;
(SEQ ID:
192)
H-Inp-D-1-Nal-D-Trp-Taz-NH2;
(SEQ ID:
192)
H-Inp-D-2-Nal-D-Trp-2-Fua-Apc-NH2;
(SEQ ID:
193)
H-Inp-D-2-Nal-D-Trp-2-Fua-NH2;
(SEQ ID:
194)
H-Inp-D-2-Nal-D-Trp-2-Thi-Apc-NH2;
(SEQ ID:
193)
H-Inp-D-2-Nal-D-Trp-3-Thi-Apc-NH2;
(SEQ ID:
193)
H-Inp-D-2-Nal-D-Trp-3-Thi-Lys-NH2;
(SEQ ID:
195)
H-Inp-D-2-Nal-D-Trp-3-Thi-NH2;
(SEQ ID:
194)
H-Inp-D-2-Nal-D-Trp-Pff-Apc-NH2;
(SEQ ID:
193)
H-Inp-D-2-Nal-D-Trp-Pff-NH2;
(SEQ ID:
194)
H-Inp-D-2-Nal-D-Trp-Taz-Apc-NH2;
(SEQ ID:
193)
H-Inp-D-2-Nal-D-Trp-Taz-NH2;
(SEQ ID:
194)
H-Inp-D-Bal -D-Bal -2-Fua-Lys-NH2;
(SEQ ID:
196)
H-Inp-D-Bal -D-Bal -2-Fua-NH2;
(SEQ ID:
197)
H-Inp-D-Bal -D-Bal -2-Thi-Lys-NH2;
(SEQ ID:
196)
H-Inp-D-Bal -D-Bal -3-Thi-Lys-NH2;
(SEQ ID:
196)
H-Inp-D-Bal -D-Bal -Pff-Lys-NH2;
(SEQ ID:
196)
H-Inp-D-Bal -D-Bal -Pff-NH2;
(SEQ ID:
197)
H-Inp-D-Bal -D-Bal -Phe-Lys-NH2;
(SEQ ID:
196)
H-Inp-D-Bal -D-Bal -Taz-Lys-NH2;
(SEQ ID:
196)
H-Inp-D-Bal -D-Bal -Taz-NH2;
(SEQ ID:
197)
H-Inp-D-Bal -D-Trp-2-Fua-Apc-NH2;
(SEQ ID:
198)
H-Inp-D-Bal -D-Trp-2-Fua-Lys-NH2;
(SEQ ID:
198)
H-Inp-D-Bal -D-Trp-2-Fua-NH2;
(SEQ ID:
199)
H-Inp-D-Bal -D-Trp-3-Thi-Apc-NH2;
(SEQ ID:
200)
H-Inp-D-Bal -D-Trp-3-Thi-Lys-NH2;
(SEQ ID:
200)
H-Inp-D-Bal-D-Trp-Pff-Apc-NH2;
(SEQ ID:
201)
H-Inp-D-Bal -D-Trp-Pff-Lys-NH2;
(SEQ ID:
201)
H-Inp-D-Bal -D-Trp-Pff-NH2;
(SEQ ID:
199)
H-Inp-D-Bal -D-Trp-Taz-NH2;
(SEQ ID:
199)
H-Inp-D-Bip-D-Bal -2-Fua-Lys-NH2;
(SEQ ID:
202)
H-Inp-D-Bip-D-Bal -2-Fua-NH2;
(SEQ ID:
203)
H-Inp-D-Bip-D-Bal -2-Thi-Lys-NH2;
(SEQ ID:
202)
H-Inp-D-Bip-D-Bal -3-Thi-Lys-NH2;
(SEQ ID:
202)
H-Inp-D-Bip-D-Bal -Pff-Lys-NH2;
(SEQ ID:
202)
H-Inp-D-Bip-D-Bal -Pff-NH2;
(SEQ ID:
203)
H-Inp-D-Bip-D-Bal -Taz-Lys-NH2;
(SEQ ID:
204)
H-Inp-D-Bip-D-Bal -Taz-NH2;
(SEQ ID:
205)
H-Inp-D-Bip-D-Trp-2-Fua-Lys-NH2;
(SEQ ID:
206)
H-Inp-D-Bip-D-Trp-2-Fua-NH2;
(SEQ ID:
207)
H-Inp-D-Bip-D-Trp-2-Thi-Lys-NH2;
(SEQ ID:
206)
H-Inp-D-Bip-D-Trp-3-Thi-Lys-NH2;
(SEQ ID:
206)
H-Inp-D-Bip-D-Trp-Pff-Lys-NH2;
(SEQ ID:
206)
H-Inp-D-Bip-D-Trp-Pff-NH2;
(SEQ ID:
207)
H-Inp-D-Bip-D-Trp-Taz-Lys-NH2;
(SEQ ID:
206)
H-Inp-D-Bip-D-Trp-Taz-NH2;
(SEQ ID:
207)
H-Inp-D-1-Nal-D-Trp-3-Pal-Lys-NH2;
(SEQ ID:
128)
H-Inp-D-2-Nal-D-Trp-4-Pal-Lys-NH2;
(SEQ ID:
129)
H-Inp-D-2-Nal-D-Trp-Om-Lys-NH2;
(SEQ ID:
129)
H-Inp-D-Bip-D-Trp-Phe-Lys-NH2;
(SEQ ID:
130)
H-Inp-D-2-Nal-D-Trp-Thr(Bzl)-Lys-NH2;
(SEQ ID:
131)
H-Inp-D-2-Nal-D-Trp-Pff-Lys-NH2;
(SEQ ID:
131)
H-Inp-D-2-Nal-D-Trp-2-Thi-Lys-NH2;
(SEQ ID:
132)
H-Inp-D-2-Nal-D-Trp-Taz-Lys-NH2;
(SEQ ID:
132)
H-Inp-D-Dip-D-Trp-Phe-Lys-NH2;
(SEQ ID:
133)
H-Inp-D-Bpa-D-Trp-Phe-Lys-NH2;
(SEQ ID:
133)
H-Inp-D-2-Nal-D-Bpa-Phe-Lys-NH2;
(SEQ ID:
134)
H-Inp-D-2-Nal-D-Trp-Thr(Bzl)-NH2;
(SEQ ID:
138)
H-Inp-D-2-Nal-D-Trp-Pff-NH2;
(SEQ ID:
138)
H-Inp-D-2-Nal-D-Trp-Taz-NH2;
(SEQ ID:
138)
H-Inp-D-2-Nal-D-Dip-Phe-NH2;
(SEQ ID:
140)
H-Inp-D-2-Nal-D-Trp-3-Pal-Lys-NH2;
(SEQ ID:
143)
H-Inp-D-Trp-D-2-Nal(Ψ)-Pim;
(SEQ ID:
127)
H-Inp-D-Bal -D-Trp-2-Thi-Lys-NH2;
(SEQ ID:
144)
H-Inp-D-Bal -D-Trp-Phe-Lys-NH2;
(SEQ ID:
144)
H-Inp-D-1-Nal-D-Trp-2-Thi-Lys-NH2;
(SEQ ID:
128)
H-Inp-D-2-Nal-D-Trp-Phe-Apc-NH2;
(SEQ ID:
2)
H-Inp-D-1-Nal-D-Trp-Phe-Apc-NH2;
(SEQ ID:
2)
H-Inp-D-Bal-D-Trp-Phe-Apc-NH2;
(SEQ ID:
2)
H-Apc-D-2-Nal-D-Trp-Phe-Lys-NH2;
(SEQ ID:
145)
H-Apc-D-1-Nal-D-Trp-2-Thi-Lys-NH2;
(SEQ ID:
146)
H-Inp-D-2-Nal-D-Trp(Ψ)-Pim;
(SEQ ID:
149)
H-Inp-D-1-Nal-D-Trp(Ψ)-Pim;
(SEQ ID:
149)
H-Inp-D-Bal-D-Trp(Ψ)-Pim;
(SEQ ID:
149)
H-Aib-D-Ser(Bzl)-D-Trp(Ψ)-Pim;
(SEQ ID:
150)
H-Inp-D-1-Nal-D-Trp-Taz-Lys-NH2;
(SEQ ID:
151)
H-Inp-D-Bal -D-Trp-Taz-Lys-NH2;
(SEQ ID:
151)
H-Apc-D-1-Nal-D-Trp-Taz-Lys-NH2;
(SEQ ID:
152)
H-Apc-D-Bal -D-Trp-Taz-Lys-NH2;
(SEQ ID:
152)
H-Apc-D-Bal -D-Trp-2-Thi-Lys-NH2;
(SEQ ID:
153)
H-Apc-D-Bal -D-Trp-Phe-Lys-NH2;
(SEQ ID:
153)
H-Apc-D-1-Nal-D-Trp-Phe-Apc-NH2;
(SEQ ID:
154)
H-Apc-D-Bal -D-Trp-Phe-Apc-NH2;
(SEQ ID:
154)
H-Apc-D-1-Nal-D-1-Nal-Phe-Apc-NH2;
(SEQ ID:
155)
H-Apc-D-1-Nal-D-2-Nal-Phe-Apc-NH2;
(SEQ ID:
155)
H-Apc-D-1-Nal-D-1-Nal-Phe-Lys-NH2;
(SEQ ID:
156)
H-Apc-D-Bal-D-1-Nal-Phe-Apc-NH2;
(SEQ ID:
157)
H-Apc-D-Bal-D-2-Nal-Phe-Apc-NH2;
(SEQ ID:
157)
H-Apc-D-Bal-D-1-Nal-Phe-Lys-NH2;
(SEQ ID:
158)
H-Apc-D-Bal-D-2-Nal-Phe-Lys-NH2;
(SEQ ID:
158)
H-Apc-D-1-Nal-D-Trp-2-Thi-NH2;
(SEQ ID:
159)
H-Apc-D-Bal -D-Trp-Phe-NH2;
(SEQ ID:
160)
H-Apc-D-1-Nal-D-Trp-Taz-NH2;
(SEQ ID:
159)
H-Apc-D-Bal -D-Trp-2-Thi-NH2;
(SEQ ID:
161)
H-Apc-D-Bal -D-Trp-Taz-NH2;
(SEQ ID:
161)
H-Apc-D-2-Nal-D-Trp-2-Thi-NH2;
(SEQ ID:
162)
H-Apc-D-2-Nal-D-Trp-Taz-NH2;
(SEQ ID:
162)
H-Inp-D-1-Nal-D-Trp-Taz-Apc-NH2;
(SEQ ID:
163)
H-Inp-D-Bal-D-Trp-Taz-Apc-NH2;
(SEQ ID:
163)
H-Apc-D-1-Nal-D-Trp-Taz-Apc-NH2;
(SEQ ID:
164)
H-Apc-D-Bal -D-Trp-Taz-Apc-NH2;
(SEQ ID:
164)
H-Inp-D-2-Nal-D-Trp-3-Thi-Lys-NH2;
(SEQ ID:
195)
H-Inp-D-Bal -D-Trp-3-Thi-Lys-NH2;
(SEQ ID:
200)
H-Inp-D-Bal -D-Trp-2-Fua-Lys-NH2;
(SEQ ID:
198)
H-Inp-D-Bal -D-Trp-Pff-Lys-NH2;
(SEQ ID:
201)
H-Inp-D-Bal -D-Trp-3-Thi-Apc-NH2;
(SEQ ID:
200)
H-Inp-D-Bal -D-Trp-2-Fua-Apc-NH2;
(SEQ ID:
198)
H-Inp-D-Bal-D-Trp-Pff-Apc-NH2;
(SEQ ID:
201)
H-Apc-D-Bal -D-Trp-3-Thi-Lys-NH2;
(SEQ ID:
185)
H-Apc-D-Bal -D-Trp-2-Fua-Lys-NH2;
(SEQ ID:
183)
H-Apc-D-Bal -D-Trp-Pff-Lys-NH2;
(SEQ ID:
186)
H-Inp-D-Bal -D-Bal -Phe-Lys-NH2;
(SEQ ID:
196)
H-Inp-D-Bal -D-Bal -2-Thi-Lys-NH2;
(SEQ ID:
196)
H-Inp-D-Bal -D-Bal -3-Thi-Lys-NH2;
(SEQ ID:
196)
H-Inp-D-Bal -D-Bal -Taz-Lys-NH2;
(SEQ ID:
196)
H-Inp-D-Bal -D-Bal -2-Fua-Lys-NH2;
(SEQ ID:
196)
H-Inp-D-Bal -D-Bal -Pff-Lys-NH2;
(SEQ ID:
196)
H-Apc-D-Bal -D-Bal -Phe-Lys-NH2;
(SEQ ID:
181)
H-Apc-D-Bal -D-Bal -2-Thi-Lys-NH2;
(SEQ ID:
178)
H-Apc-D-Bal -D-Bal -3-Thi-Lys-NH2;
(SEQ ID:
179)
H-Apc-D-Bal -D-Bal -Taz-Lys-NH2;
(SEQ ID:
182)
H-Apc-D-Bal -D-Bal -2-Fua-Lys-NH2;
(SEQ ID:
176)
H-Apc-D-Bal -D-Bal -Pff-Lys-NH2;
(SEQ ID:
180)
H-Inp-D-1-Nal-D-Trp-3-Thi-Lys-NH2;
(SEQ ID:
190)
H-Inp-D-1-Nal-D-Trp-2-Fua-Lys-NH2;
(SEQ ID:
189)
H-Inp-D-1-Nal-D-Trp-Pff-Lys-NH2;
(SEQ ID:
191)
H-Inp-D-1-Nal-D-Bal -Phe-Lys-NH2;
(SEQ ID:
187)
H-Inp-D-1-Nal-D-Bal -2-Thi-Lys-NH2;
(SEQ ID:
187)
H-Inp-D-1-Nal-D-Bal -3-Thi-Lys-NH2;
(SEQ ID:
187)
H-Inp-D-1-Nal-D-Bal -Taz-Lys-NH2;
(SEQ ID:
187)
H-Inp-D-1-Nal-D-Bal -2-Fua-Lys-NH2;
(SEQ ID:
187)
H-Inp-D-1-Nal-D-Bal -Pff-Lys-NH2;
(SEQ ID:
187)
H-Inp-D-2-Nal-D-Trp-2-Thi-Apc-NH2;
(SEQ ID:
193)
H-Inp-D-2-Nal-D-Trp-3-Thi-Apc-NH2;
(SEQ ID:
193)
H-Inp-D-2-Nal-D-Trp-Taz-Apc-NH2;
(SEQ ID:
193)
H-Inp-D-2-Nal-D-Trp-2-Fua-Apc-NH2;
(SEQ ID:
193)
H-Inp-D-2-Nal-D-Trp-Pff-Apc-NH2;
(SEQ ID:
193)
H-Inp-D-1-Nal-D-Trp-3-Thi-Apc-NH2;
(SEQ ID:
190)
H-Inp-D-1-Nal-D-Trp-2-Fua-Apc-NH2;
(SEQ ID:
189)
H-Inp-D-1-Nal-D-Trp-Pff-Apc-NH2;
(SEQ ID:
191)
H-Apc-D-1-Nal-D-Trp-3-Thi-Lys-NH2;
(SEQ ID:
167)
H-Apc-D-1-Nal-D-Trp-2-Fua-Lys-NH2;
(SEQ ID:
165)
H-Apc-D-1-Nal-D-Trp-Pff-Lys-NH2;
(SEQ ID:
169)
H-Apc-D-2-Nal-D-Trp-2-Thi-Lys-NH2;
(SEQ ID:
172)
H-Apc-D-2-Nal-D-Trp-3-Thi-Lys-NH2;
(SEQ ID:
173)
H-Apc-D-2-Nal-D-Trp-Taz-Lys-NH2;
(SEQ ID:
175)
H-Apc-D-2-Nal-D-Trp-2-Fua-Lys-NH2;
(SEQ ID:
170)
H-Apc-D-2-Nal-D-Trp-Pff-Lys-NH2;
(SEQ ID:
174)
H-Inp-D-Bip-D-Trp-2-Thi-Lys-NH2;
(SEQ ID:
206)
H-Inp-D-Bip-D-Trp-3-Thi-Lys-NH2;
(SEQ ID:
206)
H-Inp-D-Bip-D-Trp-Taz-Lys-NH2;
(SEQ ID:
206)
H-Inp-D-Bip-D-Trp-2-Fua-Lys-NH2;
(SEQ ID:
206)
H-Inp-D-Bip-D-Trp-Pff-Lys-NH2;
(SEQ ID:
206)
H-Inp-D-Bip-D-Bal -2-Thi-Lys-NH2;
(SEQ ID:
202)
H-Inp-D-Bip-D-Bal -3-Thi-Lys-NH2;
(SEQ ID:
202)
H-Inp-D-Bip-D-Bal -Taz-Lys-NH2;
(SEQ ID:
204)
H-Inp-D-Bip-D-Bal -2-Fua-Lys-NH2;
(SEQ ID:
202)
H-Inp-D-Bip-D-Bal-Pff-Lys-NH2;
(SEQ ID:
202)
H-Apc-D-Bal -D-Trp-3-Thi-Apc-NH2;
(SEQ ID:
185)
H-Apc-D-Bal -D-Trp-2-Fua-Apc-NH2;
(SEQ ID:
183)
H-Apc-D-Bal -D-Trp-Pff-Apc-NH2;
(SEQ ID:
186)
H-Apc-D-Bal-D-Bal-Phe-Apc-NH2;
(SEQ ID:
181)
H-Apc-D-Bal -D-Bal -2-Thi-Apc-NH2;
(SEQ ID:
178)
H-Apc-D-Bal -D-Bal -3-Thi-Apc-NH2;
(SEQ ID:
179)
H-Apc-D-Bal -D-Bal -Taz-Apc-NH2;
(SEQ ID:
182)
H-Apc-D-Bal -D-Bal -2-Fua-Apc-NH2;
(SEQ ID:
176)
H-Apc-D-Bal -D-Bal -Pff-Apc-NH2;
(SEQ ID:
180)
H-Apc-D-1-Nal-D-Trp-3-Thi-Apc-NH2;
(SEQ ID:
167)
H-Apc-D-1-Nal-D-Trp-2-Fua-Apc-NH2;
(SEQ ID:
165)
H-Apc-D-1-Nal-D-Trp-Pff-Apc-NH2;
(SEQ ID:
169)
H-Apc-D-2-Nal-D-Trp-2-Thi-Apc-NH2;
(SEQ ID:
172)
H-Apc-D-2-Nal-D-Trp-3-Thi-Apc-NH2;
(SEQ ID:
173)
H-Apc-D-2-Nal-D-Trp-Taz-Apc-NH2;
(SEQ ID:
175)
H-Apc-D-2-Nal-D-Trp-2-Fua-Apc-NH2;
(SEQ ID:
170)
H-Apc-D-2-Nal-D-Trp-Pff-Apc-NH2;
(SEQ ID:
174)
H-Inp-D-Bal -D-Trp-Taz-NH2;
(SEQ ID:
199)
H-Inp-D-Bal -D-Trp-2-Fua-NH2;
(SEQ ID:
199)
H-Inp-D-Bal -D-Trp-Pff-NH2;
(SEQ ID:
199)
H-Apc-D-Bal -D-Trp-3-Thi-NH2;
(SEQ ID:
184)
H-Apc-D-Bal -D-Trp-2-Fua-NH2;
(SEQ ID:
184)
H-Apc-D-Bal -D-Trp-Pff-NH2;
(SEQ ID:
184)
H-Apc-D-Bal -D-Trp-4-Pal-NH2;
(SEQ ID:
184)
H-Apc-D-Bal -D-Trp-3-Pal-NH2;
(SEQ ID:
184)
H-Apc-D-Bal -D-Trp-2-Pal-NH2;
(SEQ ID:
184)
H-Inp-D-Bal -D-Bal -Taz-NH2;
(SEQ ID:
197)
H-Inp-D-Bal -D-Bal -2-Fua-NH2;
(SEQ ID:
197)
H-Inp-D-Bal -D-Bal -Pff-NH2;
(SEQ ID:
197)
H-Apc-D-Bal -D-Bal -Phe-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Bal -2-Thi-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Bal -3-Thi-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Bal -Taz-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Bal -2-Fua-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Bal -Pff-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Bal -4-Pal-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Bal -3-Pal-NH2;
(SEQ ID:
177)
H-Apc-D-Bal -D-Bal -2-Pal-NH2;
(SEQ ID:
177)
H-Inp-D-1-Nal-D-Trp-Taz-NH2;
(SEQ ID:
192)
H-Inp-D-1-Nal-D-Trp-2-Fua-NH2;
(SEQ ID:
189)
H-Inp-D-1-Nal-D-Trp-Pff-NH2;
(SEQ ID:
192)
H-Inp-D-1-Nal-D-Bal -Taz-NH2;
(SEQ ID:
188)
H-Inp-D-1-Nal-D-Bal -2-Fua-NH2;
(SEQ ID:
188)
H-Inp-D-1-Nal-D-Bal -Pff-NH2;
(SEQ ID:
188)
H-Inp-D-2-Nal-D-Trp-Taz-NH2;
(SEQ ID:
194)
H-Inp-D-2-Nal-D-Trp-2-Fua-NH2;
(SEQ ID:
194)
H-Inp-D-2-Nal-D-Trp-Pff-NH2;
(SEQ ID:
194)
H-Apc-D-1-Nal-D-Trp-3-Thi-NH2;
(SEQ ID:
168)
H-Apc-D-1-Nal-D-Trp-2-Fua-NH2;
(SEQ ID:
165)
H-Apc-D-1-Nal-D-Trp-Pff-NH2;
(SEQ ID:
168)
H-Apc-D-1-Nal-D-Trp-4-Pal-NH2;
(SEQ ID:
168)
H-Apc-D-1-Nal-D-Trp-3-Pal-NH2;
(SEQ ID:
166)
H-Apc-D-1-Nal-D-Trp-2-Pal-NH2;
(SEQ ID:
166)
H-Apc-D-2-Nal-D-Trp-3-Thi-NH2;
(SEQ ID:
171)
H-Apc-D-2-Nal-D-Trp-2-Fua-NH2;
(SEQ ID:
171)
H-Apc-D-2-Nal-D-Trp-Pff-NH2;
(SEQ ID:
171)
H-Apc-D-2-Nal-D-Trp-4-Pal-NH2;
(SEQ ID:
171)
H-Apc-D-2-Nal-D-Trp-3-Pal-NH2;
(SEQ ID:
171)
H-Apc-D-2-Nal-D-Trp-2-Pal-NH2;
(SEQ ID:
171)
H-Inp-D-Bip-D-Trp-Taz-NH2;
(SEQ ID:
207)
H-Inp-D-Bip-D-Trp-2-Fua-NH2;
(SEQ ID:
207)
H-Inp-D-Bip-D-Trp-Pff-NH2;
(SEQ ID:
207)
H-Inp-D-Bip-D-Bal -Taz-NH2;
(SEQ ID:
205)
H-Inp-D-Bip-D-Bal -2-Fua-NH2;
(SEQ ID:
203)
H-Inp-D-Bip-D-Bal -Pff-NH2;
(SEQ ID:
203)
H-Inp-D-1-Nal-D-Trp-2-Thi-Apc-NH2;
(SEQ ID:
208)
H-Inp-D-Bal -D-Trp-2-Thi-Apc-NH2;
(SEQ ID:
208)
H-Apc-D-1-Nal-D-Trp-2-Thi-Apc-NH2;
(SEQ ID:
209)
H-Apc-D-Bal -D-Trp-2-Thi-Apc-NH2;
(SEQ ID:
209)
H-Apc-D-1-Nal-D-Trp-Phe-Lys-NH2;
(SEQ ID:
145)
(Ser(n-octanoyl)15)hGhrelin(1-28)-NH2;
(SEQ ID:
210)
(Glu(NH-hexyl)15)hGhrelin(1-28)-NH2;
(SEQ ID:
211)
(Glu(NH-hexyl)3,15)hGhrelin(1-28)-NH2;
(SEQ ID:
212)
(Glu(NH-hexyl)3, Ser(n-octanoyl)15)hGhrelin(1-28)-NH2;
(SEQ ID:
213)
(Aib2, Glu(NH-hexyl)15)hGhrelin(1-28)-NH2;
(SEQ ID:
214)
(Aib2, Glu(NH-hexyl)3,15)hGhrelin(1-28)-NH2;
(SEQ ID:
215)
(Aib2,8, Glu(NH-hexyl)15)hGhrelin(1-28)-NH2;
(SEQ ID:
216)
(Aib2,8, Glu(NH-hexyl)3,15)hGhrelin(1-28)-NH2;
(SEQ ID:
217)
(Aib2,10, Glu(NH-hexyl)15)hGhrelin(1-28)-NH2;
(SEQ ID:
218)
(Aib2,10, Glu(NH-hexyl)3,15)hGhrelin(1-28)-NH2;
(SEQ ID:
219)
(Ser(n-octanoyl)16)hGhrelin(1-28)-NH2;
(SEQ ID:
220)
(Glu(NH-hexyl)16)hGhrelin(1-28)-NH2;
(SEQ ID:
221)
(Glu(NH-hexyl)3,16)hGhrelin(1-28)-NH2;
(SEQ ID:
222)
(Glu(NH-hexyl)3, Ser(n-octanoyl)16)hGhrelin(1-28)-NH2;
(SEQ ID:
223)
(Aib2, Glu(NH-hexyl)16)hGhrelin(1-28)-NH2;
(SEQ ID:
224)
(Aib2, Glu(NH-hexyl)3,16)hGhrelin(1-28)-NH2;
(SEQ ID:
225)
(Aib2,8, Glu(NH-hexyl)16)hGhrelin(1-28)-NH2;
(SEQ ID:
226)
(Aib2,8, Glu(NH-hexyl)3,16)hGhrelin(1-28)-NH2;
(SEQ ID:
227)
(Aib2,10, Glu(NH-hexyl)16)hGhrelin(1-28)-NH2;
(SEQ ID:
228)
(Aib2,10, Glu(NH-hexyl)3,16)hGhrelin(1-28)-NH2;
(SEQ ID:
229)
(Ser(n-octanoyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
230)
(Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
231)
(Glu(NH-hexyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
232)
(Glu(NH-hexyl)3, Ser(n-octanoyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
233)
(Dap(octanesulfonyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
234)
(Dap(octanesulfonyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
235)
(Dap(octanesulfonyl)3, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
236)
(Dap(octanesulfonyl)3, Ser(n-octanoyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
237)
(Glu(NH-hexyl)3, Dap(octanesulfonyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
238)
(Cys(S—(CH2)9CH3)17)hGhrelin(1-28)-NH2;
(SEQ ID:
239)
(Cys(S—(CH2)9CH3)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
240)
(Glu(NH-hexyl)3, Cys(S—(CH2)9CH3)17)hGhrelin(1-28)-NH2;
(SEQ ID:
241)
(Cys(S—(CH2)9CH3)3, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
242)
(Cys(S—(CH2)9CH3)3, Ser(n-octanoyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
243)
(Aib2, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
244)
(Aib2, Glu(NH-hexyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
245)
(Aib2, Thz7, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
246)
(Aib2, 4-Hyp7, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
246)
(Aib2, Dhp7, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
246)
(Aib2, Pip7, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
246)
(Aib2, Tic7, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
246)
(Aib2, Glu(NH-hexyl)3,17, Thz7)hGhrelin(1-28)-NH2;
(SEQ ID:
247)
(Aib2, Glu(NH-hexyl)3,17, 4-Hyp7)hGhrelin(1-28)-NH2;
(SEQ ID:
247)
(Aib2, Glu(NH-hexyl)3,17, Dhp7)hGhrelin(1-28)-NH2;
(SEQ ID:
247)
(Aib2, Glu(NH-hexyl)3,17, Pip7)hGhrelin(1-28)-NH2;
(SEQ ID:
247)
(Aib2, Glu(NH-hexyl)3,17, Tic7)hGhrelin(1-28)-NH2;
(SEQ ID:
247)
(Aib2,8, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
248)
(Aib2,8, Glu(NH-hexyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
249)
(Aib2, 3-Pal9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
250)
(Aib2, 4-Pal9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
250)
(Aib2, Taz9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
250)
(Aib2, 2-Thi9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
250)
(Aib2, Glu(NH-hexyl)3,17, 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
251)
(Aib2, Glu(NH-hexyl)3,17, 4-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
251)
(Aib2, Glu(NH-hexyl)3,17, Taz9)hGhrelin(1-28)-NH2;
(SEQ ID:
251)
(Aib2, Glu(NH-hexyl)3,17, 2-Thi9)hGhrelin(1-28)-NH2;
(SEQ ID:
251)
(Aib2,10, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
252)
(Aib2,10, Glu(NH-hexyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
253)
(Aib8, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
254)
(Taz9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
255)
(3-Pal9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
255)
(4-Pal9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
255)
(2-Thi9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
255)
(Glu(NH-hexyl)3,17, Aib8)hGhrelin(1-28)-NH2;
(SEQ ID:
256)
(Glu(NH-hexyl)3,17, Taz9)hGhrelin(1-28)-NH2;
(SEQ ID:
257)
(Glu(NH-hexyl)3,17, 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
257)
(Glu(NH-hexyl)3,17, 4-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
257)
(Glu(NH-hexyl)3,17, 2-Thi9)hGhrelin(1-28)-NH2;
(SEQ ID:
257)
(Aib1,2,10, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
258)
(Aib1,2,10, Glu(NH-hexyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
259)
(A5c2, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
260)
(A5c2, Glu(NH-hexyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
261)
(Glu(1-heptanol)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
262)
(Asp (1-heptanol)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
263)
(Glu(NH-hexyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
264)
(Asp(NH-hexyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
265)
(Aib2, Glu(NH-hexyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
266)
(Lys(biotinyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
267)
(Ser(n-octanoyl)18)hGhrelin(1-28)-NH2;
(SEQ ID:
268)
(Glu(NH-hexyl)18)hGhrelin(1-28)-NH2;
(SEQ ID:
269)
(Glu(NH-hexyl)3,18)hGhrelin(1-28)-NH2;
(SEQ ID:
270)
(Glu(NH-hexyl)3, Ser(n-octanoyl)18)hGhrelin(1-28)-NH2;
(SEQ ID:
271)
(Aib2, Glu(NH-hexyl)18)hGhrelin(1-28)-NH2;
(SEQ ID:
272)
(Aib2, Glu(NH-hexyl)3,18)hGhrelin(1-28)-NH2;
(SEQ ID:
273)
(Aib2,8, Glu(NH-hexyl)18)hGhrelin(1-28)-NH2;
(SEQ ID:
274)
(Aib2,8, Glu(NH-hexyl)3,18)hGhrelin(1-28)-NH2;
(SEQ ID:
275)
(Aib2,10, Glu(NH-hexyl)18)hGhrelin(1-28)-NH2;
(SEQ ID:
276)
(Aib2,10, Glu(NH-hexyl)3,18)hGhrelin(1-28)-NH2;
(SEQ ID:
277)
(Ser(n-octanoyl)19)hGhrelin(1-28)-NH2;
(SEQ ID:
278)
(Glu(NH-hexyl)19)hGhrelin(1-28)-NH2;
(SEQ ID:
279)
(Glu(NH-hexyl)3,19)hGhrelin(1-28)-NH2;
(SEQ ID:
280)
(Glu(NH-hexyl)3, Ser(n-octanoyl)19)hGhrelin(1-28)-NH2;
(SEQ ID:
281)
(Aib2, Glu(NH-hexyl)19)hGhrelin(1-28)-NH2;
(SEQ ID:
282)
(Aib2, Glu(NH-hexyl)3,19)hGhrelin(1-28)-NH2;
(SEQ ID:
283)
(Aib2,8, Glu(NH-hexyl)19)hGhrelin(1-28)-NH2;
(SEQ ID:
284)
(Aib2,8, Glu(NH-hexyl)3,19)hGhrelin(1-28)-NH2;
(SEQ ID:
285)
(Aib2,10, Glu(NH-hexyl)19)hGhrelin(1-28)-NH2;
(SEQ ID:
286)
(Aib2,10, Glu(NH-hexyl)3,19)hGhrelin(1-28)-NH2;
(SEQ ID:
287)
(Ser(n-octanoyl)20)hGhrelin(1-28)-NH2;
(SEQ ID:
288)
(Glu(NH-hexyl)20)hGhrelin(1-28)-NH2;
(SEQ ID:
289)
(Glu(NH-hexyl)3,20)hGhrelin(1-28)-NH2;
(SEQ ID:
290)
(Glu(NH-hexyl)3, Ser(n-octanoyl)20)hGhrelin(1-28)-NH2;
(SEQ ID:
291)
(Aib2, Glu(NH-hexyl)21hGhrelin(1-28)-NH2;
(SEQ ID:
292)
(Aib2, Glu(NH-hexyl)3,20)hGhrelin(1-28)-NH2;
(SEQ ID:
293)
(Aib2,8, Glu(NH-hexyl)9hGhrelin(1-28)-NH2;
(SEQ ID:
294)
(Aib2,8, Glu(NH-hexyl)3,20)hGhrelin(1-28)-NH2;
(SEQ ID:
295)
(Aib2,10, Glu(NH-hexyl)2,20)hGhrelin(1-28)-NH2;
(SEQ ID:
296)
(Aib2,10, Glu(NH-hexyl)3,20)hGhrelin(1-28)-NH2;
(SEQ ID:
297)
(Ac-Gly1, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
298)
(Ac-Gly1, Ser(n-octanoyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
299)
(Ac-Gly1, Glu(NH-hexyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
300)
Glu(NH-hexyl)3, Ser(n-octanoyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
301)
(Ac-Gly1, Dap(octanesulfonyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
302)
(Ac-Gly1, Dap(octanesulfonyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
303)
Dap(octanesulfonyl)3, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
304)
(Ac-Gly1, Dap(octanesulfonyl)3, Ser(n-octanoyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
305)
(Ac-Gly1, Glu(NH-hexyl)3, Dap(octanesulfonyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
306)
(Ac-Gly1, Cys(S—(CH2)9CH3)17)hGhrelin(1-28)-NH2;
(SEQ ID:
307)
(Ac-Gly1, Cys(S—(CH2)9CH3)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
308)
(Ac-Gly1, Glu(NH-hexyl)3, Cys(S—(CH2)9CH3)17)hGhrelin(1-28)-NH2;
(SEQ ID:
309)
(Ac-Gly1, Cys(S—(CH2)9CH3)3, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
310)
(Ac-Gly1, Cys(S—(CH2)9CH3)3, Ser(n-octanoyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
311)
(Ac-Gly1, Aib2, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
312)
(Ac-Gly1, Aib2, Thz7, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
313)
(Ac-Gly1, Aib2, 4-Hyp7, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
313)
(Ac-Gly1, Aib2, Dhp7, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
313)
(Ac-Gly1, Aib2, Pip7, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
313)
(Ac-Gly1, Aib2, Tic7, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
313)
(Ac-Gly1, Aib2, Glu(NH-hexyl)3,17, Thz7)hGhrelin(1-28)-NH2;
(SEQ ID:
314)
(Ac-Gly1, Aib2, Glu(NH-hexyl)3,17, 4-Hyp7)hGhrelin(1-28)-NH2;
(SEQ ID:
314)
(Ac-Gly1, Aib2, Glu(NH-hexyl)3,17, Dhp7)hGhrelin(1-28)-NH2;
(SEQ ID:
314)
(Ac-Gly1, Aib2, Glu(NH-hexyl)3,17, Pip7)hGhrelin(1-28)-NH2;
(SEQ ID:
314)
(Ac-Gly1, Aib2, Glu(NH-hexyl)3,17, Tic7)hGhrelin(1-28)-NH2;
(SEQ ID:
314)
(Ac-Gly1, Aib2,8, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
315)
(Ac-Gly1, Aib2, 3-Pal9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
316)
(Ac-Gly1, Aib2, 4-Pal9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
316)
(Ac-Gly1, Aib2, Taz9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
316)
(Ac-Gly1, Aib2, 2-Thi9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
316)
(Ac-Gly1, Aib2, Glu(NH-hexyl)3,17, 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
317)
(Ac-Gly1, Aib2, Glu(NH-hexyl)3,17, 4-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
317)
(Ac-Gly1, Aib2, Glu(NH-hexyl)3,17, Taz9)hGhrelin(1-28)-NH2;
(SEQ ID:
317)
(Ac-Gly1, Aib2, Glu(NH-hexyl)3,17, 2-Thi9)hGhrelin(1-28)-NH2;
(SEQ ID:
317)
(Ac-Gly1, Aib2,10, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
318)
(Ac-Gly1, Aib2,10, Glu(NH-hexyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
319)
(Ac-Gly1, Aib8, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
320)
(Ac-Gly1, Taz9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
321)
(Ac-Gly1, 3-Pal9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
321)
(Ac-Gly1, 4-Pal9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
321)
(Ac-Gly1, 2-Thi9, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
321)
(Ac-Gly1, Glu(NH-hexyl)3,17, Aib8)hGhrelin(1-28)-NH2;
(SEQ ID:
322)
(Ac-Gly1, Glu(NH-hexyl)3,17, Taz9)hGhrelin(1-28)-NH2;
(SEQ ID:
323)
(Ac-Gly1, Glu(NH-hexyl)3,17, 3-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
323)
(Ac-Gly1, Glu(NH-hexyl)3,17, 4-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
323)
(Ac-Gly1, Glu(NH-hexyl)3,17, 2-Thi9)hGhrelin(1-28)-NH2;
(SEQ ID:
323)
(Ac-Gly1, Aib Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
324)
(Ac-Gly1, Aib Glu(NH-hexyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
325)
(Ac-Gly1, A5c2, Glu(NH-hexyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
326)
(Ac-Gly1, A5c2, Glu(NH-hexyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
327)
(Ac-Gly1, Glu(1-heptanol)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
328)
(Ac-Gly1, Asp(1-heptanol)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
329)
(Ac-Gly1, Glu(NH-hexyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
330)
(Ac-Gly1, Asp(NH-hexyl)3,17)hGhrelin(1-28)-NH2;
(SEQ ID:
331)
(Ac-Gly1, Aib2,10, Glu(NH-hexyl)3, Lys(biotinyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
332)
(Ac-Gly1, Glu(NH-hexyl)15)hGhrelin(1-28)-NH2;
(SEQ ID:
333)
(Ac-Gly1, Ser(n-octanoyl)15)hGhrelin(1-28)-NH2;
(SEQ ID:
334)
(Ac-Gly1, Glu(NH-hexyl)3,15)hGhrelin(1-28)-NH2;
(SEQ ID:
335)
(Ac-Gly1, Glu(NH-hexyl)3, Ser(n-octanoyl)15)hGhrelin(1-28)-NH2;
(SEQ ID:
336)
(Ac-Gly1, Aib2, Glu(NH-hexyl)15)hGhrelin(1-28)-NH2;
(SEQ ID:
337)
(Ac-Gly1, Aib2, Glu(NH-hexyl)3,15)hGhrelin(1-28)-NH2;
(SEQ ID:
338)
(Ac-Gly1, Glu(NH-hexyl)15)hGhrelin(1-28)-NH2;
(SEQ ID:
339)
(Ac-Gly1, Glu(NH-hexyl)3,15)hGhrelin(1-28)-NH2;
(SEQ ID:
340)
(Ac-Gly1, Aib2,10, Glu(NH-hexyl)15)hGhrelin(1-28)-NH2;
(SEQ ID:
341)
(Ac-Gly1, Aib2,10, Glu(NH-hexyl)3,15)hGhrelin(1-28)-NH2;
(SEQ ID:
342)
(Ac-Gly1, Glu(NH-hexyl)16)hGhrelin(1-28)-NH2;
(SEQ ID:
343)
(Ac-Gly1, Ser(n-octanoyl)16)hGhrelin(1-28)-NH2;
(SEQ ID:
344)
(Ac-Gly1, Glu(NH-hexyl)3,16)hGhrelin(1-28)-NH2;
(SEQ ID:
345)
(Ac-Gly1, Glu(NH-hexyl)3, Ser(n-octanoyl)16)hGhrelin(1-28)-NH2;
(SEQ ID:
346)
(Ac-Gly1, Aib2, Glu(NH-hexyl)16)hGhrelin(1-28)-NH2;
(SEQ ID:
347)
(Ac-Gly1, Aib2, Glu(NH-hexyl)3,16)hGhrelin(1-28)-NH2;
(SEQ ID:
348)
(Ac-Gly1, Glu(NH-hexyl)16)hGhrelin(1-28)-NH2;
(SEQ ID:
349)
(Ac-Gly1, Glu(NH-hexyl)3,16)hGhrelin(1-28)-NH2;
(SEQ ID:
350)
(Ac-Gly1, Aib2,10, Glu(NH-hexyl)16)hGhrelin(1-28)-NH2;
(SEQ ID:
351)
(Ac-Gly1, Aib2,10, Glu(NH-hexyl)3,16)hGhrelin(1-28)-NH2;
(SEQ ID:
352)
(Ac-Gly1, Glu(NH-hexyl)18)hGhrelin(1-28)-NH2;
(SEQ ID:
353)
(Ac-Gly1, Ser(n-octanoyl)18)hGhrelin(1-28)-NH2;
(SEQ ID:
354)
(Ac-Gly1, Glu(NH-hexyl)3,18)hGhrelin(1-28)-NH2;
(SEQ ID:
355)
(Ac-Gly1, Glu(NH-hexyl)3, Ser(n-octanoyl)18)hGhrelin(1-28)-NH2;
(SEQ ID:
356)
(Ac-Gly1, Aib2, Glu(NH-hexyl)18)hGhrelin(1-28)-NH2;
(SEQ ID:
357)
(Ac-Gly1, Aib2, Glu(NH-hexyl)3,18)hGhrelin(1-28)-NH2;
(SEQ ID:
358)
(Ac-Gly1, Glu(NH-hexyl)18)hGhrelin(1-28)-NH2;
(SEQ ID:
359)
(Ac-Gly1, Glu(NH-hexyl)3,18)hGhrelin(1-28)-NH2;
(SEQ ID:
360)
(Ac-Gly1, Aib2,10, Glu(NH-hexyl)18)hGhrelin(1-28)-NH2;
(SEQ ID:
361)
(Ac-Gly1, Aib2,10, Glu(NH-hexyl)3,18)hGhrelin(1-28)-NH2;
(SEQ ID:
362)
(Ac-Gly1, Glu(NH-hexyl)19)hGhrelin(1-28)-NH2;
(SEQ ID:
363)
(Ac-Gly1, Ser(n-octanoyl)19)hGhrelin(1-28)-NH2;
(SEQ ID:
364)
(Ac-Gly1, Glu(NH-hexyl)3,19)hGhrelin(1-28)-NH2;
(SEQ ID:
365)
(Ac-Gly1, Glu(NH-hexyl)3, Ser(n-octanoyl)19)hGhrelin(1-28)-NH2;
(SEQ ID:
366) (Ac-Gly1, Aib2, Glu(NH-hexyl)19)hGhrelin(1-28)-NH2;
(SEQ ID:
367)
(Ac-Gly1, Aib2, Glu(NH-hexyl)3,19)hGhrelin(1-28)-NH2;
(SEQ ID:
368)
(Ac-Gly1, Glu(NH-hexyl)19)hGhrelin(1-28)-NH2;
(SEQ ID:
369)
(Ac-Gly1, Glu(NH-hexyl)3,19)hGhrelin(1-28)-NH2;
(SEQ ID:
370)
(Ac-Gly1, Aib2,10, Glu(NH-hexyl)19)hGhrelin(1-28)-NH2;
(SEQ ID:
371)
(Ac-Gly1, Aib2,10, Glu(NH-hexyl)3,19)hGhrelin(1-28)-NH2;
(SEQ ID:
372)
(Ac-Gly1, Glu(NH-hexyl)9hGhrelin(1-28)-NH2;
(SEQ ID:
373)
(Ac-Gly1, Ser(n-octanoyl)20)hGhrelin(1-28)-NH2;
(SEQ ID:
374)
(Ac-Gly1, Glu(NH-hexyl)3,20)hGhrelin(1-28)-NH2;
(SEQ ID:
375)
(Ac-Gly1, Glu(NH-hexyl)3, Ser(n-octanoyl)20)hGhrelin(1-28)-NH2;
(SEQ ID:
376)
(Ac-Gly1, Aib2, Glu(NH-hexyl)9hGhrelin(1-28)-NH2;
(SEQ ID:
377)
(Ac-Gly1, Aib2, Glu(NH-hexyl)3,20)hGhrelin(1-28)-NH2;
(SEQ ID:
378)
(Ac-Gly1, Glu(NH-hexyl)20)hGhrelin(1-28)-NH2;
(SEQ ID:
379)
(Ac-Gly1, Glu(NH-hexyl)3,20)hGhrelin(1-28)-NH2;
(SEQ ID:
380)
(Ac-Gly1, Aib2,10, Glu(NH-hexyl)21hGhrelin(1-28)-NH2;
(SEQ ID:
381)
(Ac-Gly1, Aib2,10, Glu(NH-hexyl)3,20)hGhrelin(1-28)-NH2;
(SEQ ID:
382)
(Ac-Gly1, Aib Glu(NH-hexyl)3)hGhrelin(1-28)-NH2;
(SEQ ID:
385)
(1-Apc1, Aib2,10, Glu(NH-hexyl)3)-hGhrelin(1-28)NH2;
(SEQ ID:
385)
(Inp1)hGhrelin(1-28)-NH2;
(SEQ ID:
386)
(Inp1, Aib2)hGhrelin(1-28)-NH2;
(SEQ ID:
386)
(Inp1, Aib2, Glu(NH-hexyl)3)hGhrelin(1-28)-NH2;
(SEQ ID:
387)
(Inp1, Aib2,10)hGhrelin(1-28)-NH2;
(SEQ ID:
388)
(Inp1, Aib2,8)hGhrelin(1-28)-NH2;
(SEQ ID:
389)
(Inp1, Aib2, Ser(n-octanoyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
390)
(Inp1, Ser(n-octanoyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
390)
(Inp1, Aib2,8, Ser(n-octanoyl)17)hGhrelin(1-28)-NH2;
(SEQ ID:
389)
Ac-(Inp1, Aib Glu(NH-hexyl)3)hGhrelin(1-28)-NH2;
Ac-(1-Apc1, Aib2,10, Glu(NH-hexyl)3)hGhrelin(1-28)-NH2;
(Asp3(NH-heptyl))hGhrelin(1-28)-NH2;
(SEQ ID:
391)
(des-Ser2)hGhrelin(1-28)-NH2;
(SEQ ID:
392)
(des-Gly1, des-Ser2)hGhrelin(1-28)-NH2;
(SEQ ID:
392)
(Aib1)hGhrelin(1-28)-NH2;
(SEQ ID:
393)
(Asp3(O-hexyl))hGhrelin(1-28)-NH2;
(SEQ ID:
394)
Ser3)hGhrelin(1-28)-NH2;
(SEQ ID:
395)
(A5c5, Ser3)hGhrelin(1-28)-NH2;
(SEQ ID:
396)
(Aib2′4, Sera, 4-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
397)
(n-octanoyl-Gly1, Ser3)hGhrelin(1-28)-NH2;
(SEQ ID:
398)
(isobutyryl-Gly1, Ser3)hGhrelin(1-28)-NH2;
(SEQ ID:
398)
(n-butyryl-Gly1, Ser3)hGhrelin(1-28)-NH2;
(SEQ ID:
398)
(Aib1, Thr3)hGhrelin(1-28)-NH2;
(SEQ ID:
395)
(Aib2,4, Thr3, 4-Pal9)hGhrelin(1-28)-NH2;
(SEQ ID:
397)
(n-octanoyl-Gly1, Thr3)hGhrelin(1-28)-NH2;
(SEQ ID:
399)
(isobutyryl-Gly1, Thr3)hGhrelin(1-28)-NH2;
(SEQ ID:
399)
(n-butyryl-Gly1, Thr3)hGhrelin(1-28)-NH2;
(SEQ ID:
399)
(Ac-Gly1)hGhrelin(1-28)-NH2;
(SEQ ID:
400)
(Ac-Gly1, Ser3)hGhrelin(1-28)-NH2, (SEQ ID:
400)
(Aib2, Lys(myristyl)17)hGhrelin-(1-28)-NH2;
and (SEQ ID:
383)
[Gly(myristyl)1, Aib2, Lys(myristyl)17]hGhrelin-(1-28)-NH2;
(SEQ ID:
384)
or a pharmaceutically acceptable salt thereof.

3,107 more elements

Facts

Application

15/636,684Filed 29 Jun 2017

Priority

8 Aug 2007

Published

26 Oct 2017

Term ends

Not estimatedThe source records don’t support an estimate.

Classification53 codes

A61K 38/22
From animals; from humans: hormones
A61K 38/05
Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof: dipeptides
A61K 38/06
Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof: tripeptides
A61K 38/25
Hormones: growth hormone-releasing factor [GH-RF], i.e. somatoliberin

Family

Application60/963,951Us provisional application · filed 8 Aug 2007

Application12/672,681Continuation · filed 8 Feb 2010

Application14/524,088Continuation · filed 27 Oct 2014

Application14/997,678Division · filed 18 Jan 2016

Application15/636,684Division

Application14/997,678Continuation

US 2011/0160133 A1Published application

US 2015/0111823 A1Published application

US 2016/0206700 A1Published application

US 8,871,706 B2Related patent

US 2017/0304403 A1This patent

From the US filing history. Foreign family members aren’t listed.