US 2014/0005049 A1Published application

Active compound combinations

OwnerKerstin ILG, Ulrich Heinemann +2inventors

InventorsKerstin ILG, Ulrich Heinemann, Peter Dahmen, Ulrike Wachendorff-Neumann

Life of this patent

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Abstract

The invention relates to active compound combinations, in particular within a composition, which comprises (A) an amidine compound of formula (I) and a further fungicidally (B-1), insecticidally (B-2) active or plant growth regulating compound (B-3). Moreover, the invention relates to a method for curatively or preventively controlling the phytopathogenic fungi of plants or reducing the mycotoxin contamination of plant or plant parts, to the use of a combination according to the invention for the treatment of seed, to a method for protecting a seed and not at least to the treated seed.

Claims23

Dependent claims

A composition comprising

(A) at least one compound according to formula (I)
wherein
R1 is selected from the group consisting of hydrogen-a mercapto- (—SH) and a methyl group;
R2 is selected from the group consisting of a methyl- and an ethyl group;
R3 is selected from the group consisting of a methyl-, an ethyl- and an isopropyl group;
or alternatively R2 and R3 can form, together with the N-atom to which they are attached, a piperidyl-, a pyrrolidyl- or a 2,6-dimethylmorpholinyl-ring;
R4 is selected from the group consisting of a chlorine- or a fluorine atom, a trifluoromethyl-, a difluoromethyl- and a methyl group;
R5 and R6 independently from each other, are selected from the group consisting of a hydrogen atom, a methyl- and an ethyl group;
or can form, together with the C-atom to which they are attached, a cyclopropyl ring;
R7 is selected from the group consisting of a chlorine atom, a tert-butyl-, a methoxy-, an ethoxy-, a trimethylsilyl- and a triethylsilyl-group,
n is 1
or salts or stereoisomers thereof,
and
(B-I) at least one further active compound selected from the group consisting of
(B-I.2) inhibitors of the respiratory chain at complex I or II,
(B-I.3) inhibitors of the respiratory chain at complex III,
(B-I.4) Inhibitors of the mitosis and cell division,
(B-I.5) Compounds capable to have a multisite action,
(B-I.6) Compounds capable to induce a host defence,
(B-I.7) Inhibitors of the amino acid and/or protein biosynthesis,
(B-I.8) Inhibitors of the ATP production,
(B-I.9) Inhibitors of the cell wall synthesis,
(B-I.10) Inhibitors of the lipid and membrane synthesis,
(B-I.11) Inhibitors of the melanine biosynthesis,
(B-I.12) Inhibitors of the nucleic acid synthesis,
(B-I.13) Inhibitors of the signal transduction,
(B-I.14) Compounds capable to act as an uncoupler, and
(B-I.15) Further compounds
or
(B-II) at least one further insecticidally active compound, selected from the group consisting of
(B-II.1) Acetylcholinesterase (AChE) inhibitors,
(B-II.2) GABA-gated chloride channel antagonists,
(B-II.3) Sodium channel modulators/voltage-dependent sodium channel blockers,
(B-II.4) Nicotinergic acetylcholine receptor agonists,
(B-II.5) Allosteric acetylcholine receptor modulators (agonists),
(B-II.6) Chloride channel activators,
(B-II.7) Juvenile hormone mimics,
(B-II.8) Miscellaneous non-specific (multi-site) inhibitors,
(B-II.9) Selective homopteran feeding blockers,
(B-II.10) Mite growth inhibitors,
(B-II.11) Microbial disruptors of insect midgut membranes,
(B-II.12) Inhibitors of mitochondrial ATP synthase,
(B-II.13) Uncouplers of oxidative phoshorylation via disruption of the proton gradient,
(B-II.14) Nicotinic acetylcholine receptor channel blockers,
(B-II.15) Inhibitors of chitin biosynthesis, type 0,
(B-II.16) Inhibitors of chitin biosynthesis, type 1,
(B-II.17) Moulting disruptors,
(B-II.18) Ecdysone receptor agonists/disruptors,
(B-II.19) Octopamine receptor agonists,
(B-II.20) Mitochondrial complex III electron transport inhibitors,
(B-II.21) Mitochondrial complex I electron transport inhibitors,
(B-II.22) Voltage-dependent sodium channel blockers,
(B-II.23) Inhibitors of acetyl CoA carboxylase,
(B-II.24) Mitochondrial complex IV electron inhibitors,
(B-II.25) Mitochondrial complex II electron transport inhibitors,
(B-II.28) Ryanodine receptor modulators,
or
(B-III) at least one compound having plant growth regulating activity, selected from the group consisting of
(B-III.1) antiauxines,
(B-III.2) auxines,
(B-III.3) cytokinines,
(B-III.4) defoliating agents,
(B-III.5) ethylene inhibitors,
(B-III.6) ethylene generators,
(B-III.7) gibberellines,
(B-III.8) abscisinic acid, ancymidol, butralin, carbaryl, chlorphonium or its chloride, chlorpropham, dikegulac, dikegulac-sodium, flumetralin, fluoridamide, fosamine, glyphosine, isopyrimol, jasmonic acid, maleic acid hydrazide or its potassium salt, mepiquat or its chloride, piproctanyl or its bromide, prohydrojasmon, propham, 2,3,5-tri-iodobenzoic acid, 2,6-diisopropylnaphthaline, cloprop, 1-naphthylacetic acid ethylester, isoprothiolane, MCPB-ethyl [4-4-chloro-o-tolyloxy)butyric acid ethylester], N-acetylthiazolidine-4-carboxylic acid, n-decanol, pelargonic acid, N-phenylphthaliminic acid, tecnazene, triacontanol, 2,3-dihydro-5,6-diphenyl-1,4-oxathiin, 2-cyano-3-(2,4-dichlorophenyl)acrylic acid, 2-hydrazinoethanol, alorac, amidochlor, BTS 44584 [dimethyl(4-piperidinocarbonyloxy-2,5-xylyl)sulfonium-toluen-4-sulfonat], chloramben, chlorfluren, chlorfluren-methyl, dicamba-methyl, dichlorflurenol, dichlorflurenol-methyl, dimexano, etacelasil, hexafluoraceton-trihydrat, N-(2-ethyl-2H-pyrazol-3-yl)-N′-phenylurea, N-m-tolylphthalaminic acid, N-Pyrrolidinosuccinaminic acid, 3-tert-Butylphenoxyacetic acid propylester, pydanon, sodium (Z)-3-chloracrylate,
(B-III.9) morphactines,
(B-III.10) plant growth retarders/modifiers,
(B-III.11) plant growth stimulators,
(B-III.12) benzofluor, buminafos, carvone, ciobutide, clofencet, clofence-potassium, cloxyfonac, cloxyfonac-sodium, cyclanilide, cycloheximide, epocholeone, ethylchlozate, ethylene, fenridazon, heptopargil, holosulf, inabenfide, karetazan, lead arsenate, methasulfocarb, prohexadione, prohexadione-Calcium, pydanon, sintofen, triapenthenol, trinexapac and trinexapac-ethyl.

67 more elements

Dependencies are inferred from the claim text.

Facts

Application: 14/020,271Filed 6 Sep 2013
Priority: EP 09179444.616 Dec 2009
Published: 2 Jan 2014
Term ends: Not estimatedThe source records don’t support an estimate.

Classification3 codes

A01N 43/82
Having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms: five-membered rings with three ring hetero atoms
A01N 25/00
Biocides, pest repellants or attractants, or plant growth regulators, characterised by their
A01N
Preservation of bodies of humans or animals or plants or parts thereof

Family

Application61/287,475Us provisional application · filed 17 Dec 2009
Application12/969,694Division · filed 16 Dec 2010
Application14/020,271Division
US 2011/0152077 A1Published application
US 8,530,381 B2Related patent
US 2014/0005049 A1This patent

From the US filing history. Foreign family members aren’t listed.

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Abstract

A composition comprising

(A) at least one compound according to formula (I)
wherein
R1 is selected from the group consisting of hydrogen-a mercapto- (—SH) and a methyl group;
R2 is selected from the group consisting of a methyl- and an ethyl group;
R3 is selected from the group consisting of a methyl-, an ethyl- and an isopropyl group;
or alternatively R2 and R3 can form, together with the N-atom to which they are attached, a piperidyl-, a pyrrolidyl- or a 2,6-dimethylmorpholinyl-ring;
R4 is selected from the group consisting of a chlorine- or a fluorine atom, a trifluoromethyl-, a difluoromethyl- and a methyl group;
R5 and R6 independently from each other, are selected from the group consisting of a hydrogen atom, a methyl- and an ethyl group;
or can form, together with the C-atom to which they are attached, a cyclopropyl ring;
R7 is selected from the group consisting of a chlorine atom, a tert-butyl-, a methoxy-, an ethoxy-, a trimethylsilyl- and a triethylsilyl-group,
n is 1
or salts or stereoisomers thereof,
and
(B-I) at least one further active compound selected from the group consisting of
(B-I.2) inhibitors of the respiratory chain at complex I or II,
(B-I.3) inhibitors of the respiratory chain at complex III,
(B-I.4) Inhibitors of the mitosis and cell division,
(B-I.5) Compounds capable to have a multisite action,
(B-I.6) Compounds capable to induce a host defence,
(B-I.7) Inhibitors of the amino acid and/or protein biosynthesis,
(B-I.8) Inhibitors of the ATP production,
(B-I.9) Inhibitors of the cell wall synthesis,
(B-I.10) Inhibitors of the lipid and membrane synthesis,
(B-I.11) Inhibitors of the melanine biosynthesis,
(B-I.12) Inhibitors of the nucleic acid synthesis,
(B-I.13) Inhibitors of the signal transduction,
(B-I.14) Compounds capable to act as an uncoupler, and
(B-I.15) Further compounds
or
(B-II) at least one further insecticidally active compound, selected from the group consisting of
(B-II.1) Acetylcholinesterase (AChE) inhibitors,
(B-II.2) GABA-gated chloride channel antagonists,
(B-II.3) Sodium channel modulators/voltage-dependent sodium channel blockers,
(B-II.4) Nicotinergic acetylcholine receptor agonists,
(B-II.5) Allosteric acetylcholine receptor modulators (agonists),
(B-II.6) Chloride channel activators,
(B-II.7) Juvenile hormone mimics,
(B-II.8) Miscellaneous non-specific (multi-site) inhibitors,
(B-II.9) Selective homopteran feeding blockers,
(B-II.10) Mite growth inhibitors,
(B-II.11) Microbial disruptors of insect midgut membranes,
(B-II.12) Inhibitors of mitochondrial ATP synthase,
(B-II.13) Uncouplers of oxidative phoshorylation via disruption of the proton gradient,
(B-II.14) Nicotinic acetylcholine receptor channel blockers,
(B-II.15) Inhibitors of chitin biosynthesis, type 0,
(B-II.16) Inhibitors of chitin biosynthesis, type 1,
(B-II.17) Moulting disruptors,
(B-II.18) Ecdysone receptor agonists/disruptors,
(B-II.19) Octopamine receptor agonists,
(B-II.20) Mitochondrial complex III electron transport inhibitors,
(B-II.21) Mitochondrial complex I electron transport inhibitors,
(B-II.22) Voltage-dependent sodium channel blockers,
(B-II.23) Inhibitors of acetyl CoA carboxylase,
(B-II.24) Mitochondrial complex IV electron inhibitors,
(B-II.25) Mitochondrial complex II electron transport inhibitors,
(B-II.28) Ryanodine receptor modulators,
or
(B-III) at least one compound having plant growth regulating activity, selected from the group consisting of
(B-III.1) antiauxines,
(B-III.2) auxines,
(B-III.3) cytokinines,
(B-III.4) defoliating agents,
(B-III.5) ethylene inhibitors,
(B-III.6) ethylene generators,
(B-III.7) gibberellines,
(B-III.8) abscisinic acid, ancymidol, butralin, carbaryl, chlorphonium or its chloride, chlorpropham, dikegulac, dikegulac-sodium, flumetralin, fluoridamide, fosamine, glyphosine, isopyrimol, jasmonic acid, maleic acid hydrazide or its potassium salt, mepiquat or its chloride, piproctanyl or its bromide, prohydrojasmon, propham, 2,3,5-tri-iodobenzoic acid, 2,6-diisopropylnaphthaline, cloprop, 1-naphthylacetic acid ethylester, isoprothiolane, MCPB-ethyl [4-4-chloro-o-tolyloxy)butyric acid ethylester], N-acetylthiazolidine-4-carboxylic acid, n-decanol, pelargonic acid, N-phenylphthaliminic acid, tecnazene, triacontanol, 2,3-dihydro-5,6-diphenyl-1,4-oxathiin, 2-cyano-3-(2,4-dichlorophenyl)acrylic acid, 2-hydrazinoethanol, alorac, amidochlor, BTS 44584 [dimethyl(4-piperidinocarbonyloxy-2,5-xylyl)sulfonium-toluen-4-sulfonat], chloramben, chlorfluren, chlorfluren-methyl, dicamba-methyl, dichlorflurenol, dichlorflurenol-methyl, dimexano, etacelasil, hexafluoraceton-trihydrat, N-(2-ethyl-2H-pyrazol-3-yl)-N′-phenylurea, N-m-tolylphthalaminic acid, N-Pyrrolidinosuccinaminic acid, 3-tert-Butylphenoxyacetic acid propylester, pydanon, sodium (Z)-3-chloracrylate,
(B-III.9) morphactines,
(B-III.10) plant growth retarders/modifiers,
(B-III.11) plant growth stimulators,
(B-III.12) benzofluor, buminafos, carvone, ciobutide, clofencet, clofence-potassium, cloxyfonac, cloxyfonac-sodium, cyclanilide, cycloheximide, epocholeone, ethylchlozate, ethylene, fenridazon, heptopargil, holosulf, inabenfide, karetazan, lead arsenate, methasulfocarb, prohexadione, prohexadione-Calcium, pydanon, sintofen, triapenthenol, trinexapac and trinexapac-ethyl.

67 more elements

Facts

Application

14/020,271Filed 6 Sep 2013

Priority

EP 09179444.616 Dec 2009

Published

2 Jan 2014

Term ends

Not estimatedThe source records don’t support an estimate.

Classification3 codes

A01N 43/82
Having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms: five-membered rings with three ring hetero atoms
A01N 25/00
Biocides, pest repellants or attractants, or plant growth regulators, characterised by their
A01N
Preservation of bodies of humans or animals or plants or parts thereof

Family

Application61/287,475Us provisional application · filed 17 Dec 2009

Application12/969,694Division · filed 16 Dec 2010

Application14/020,271Division

US 2011/0152077 A1Published application

US 8,530,381 B2Related patent

US 2014/0005049 A1This patent

From the US filing history. Foreign family members aren’t listed.