Back to results
US 2011/0218219 A1Published application
Substituted sulphonamido phenoxybenzamides
AssigneeBayer Schering Pharma Aktiengesellschaft
InventorsIngo Hartung, Marion Hitchcock, Florian Puhler, Gerhard Siemeister, Roland Neuhaus
Life of this patent
Estimating the term…
Abstract
The present invention relates to substituted sulphonamido phenoxybenzamide compounds of general formula (I): in which A, R1, R2, R3, R4, R5, R6, R7, R8 and n are as defined in the claims, to pharmaceutical compositions and combinations containing said compounds, to methods of preparing said compounds, and to the use of said compounds or compositions for treating hyper-proliferative and/or angiogenesis disorders, as a sole agent or in combination with other active ingredients.
Claims21
A compound of general formula (I):
- in which:
- R1 is selected from the group comprising, preferably consisting of, halogen or —C≡C—H;
- R2 is hydrogen, halogen or alkyl;
- wherein at least one of R1 and R2 is halogen;
- R3 is hydrogen or alkyl;
- R4 is selected from the group comprising, preferably consisting of, halogen and cyano;
- R5 is C2-C6 alkyl;
- R6 is selected from the group comprising, preferably consisting of, hydrogen, halogen, cyano, alkoxy, amino, alkylamino, dialkylamino;
- R7 and R8 independently from each other are hydrogen, halogen or alkyl;
- A is selected from the group comprising, preferably consisting of, aryl and heteroaryl;
- n is an integer from 0 to 2.
8 more elements
Dependencies are inferred from the claim text.