Deuterium-enriched risperidone
AssigneeProtia, LLC
InventorAnthony W. Czarnik
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Abstract
The present application describes deuterium-enriched risperidone, pharmaceutically acceptable salt forms thereof, and methods of treating using the same.
Claims43
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A deuterium-enriched compound, wherein the compound is selected from:
- or a pharmaceutically acceptable salt, wherein when one of R1-R27 is present, it is selected from H or D.
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A deuterium-enriched compound, wherein the compound is:
- or a pharmaceutically acceptable salt thereof.
A deuterium-enriched compound, wherein the compound is:
- or a pharmaceutically acceptable salt thereof, wherein R1-8 and R12-27 are selected from H and D.
A deuterium-enriched compound, wherein the compound is:
- or a pharmaceutically acceptable salt thereof, wherein R1-15 and R25-27 are selected from H and D.
A deuterium-enriched compound, wherein the compound is:
- or a pharmaceutically acceptable salt thereof, wherein R1-24 are selected from H and D.
A deuterium-enriched compound, wherein the compound is:
- or a pharmaceutically acceptable salt thereof, wherein R1-24 are selected from H and D.
A deuterium-enriched compound, wherein the compound is:
- or a pharmaceutically acceptable salt thereof.
A deuterium-enriched compound, wherein the compound is:
- or a pharmaceutically acceptable salt thereof.
A pharmaceutical composition, comprising:
- a pharmaceutically acceptable carrier and a therapeutically effective amount of at least one compound selected from:
- or a pharmaceutically acceptable salt form thereof.
A method for treating schizophrenia comprising:
- administering, to a patient in need thereof, a therapeutically effective amount of a compound selected from:
- or a pharmaceutically acceptable salt form thereof.
Dependencies are inferred from the claim text.