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US 2010/0305111 A1Published application
Substituted piperidines
AssigneeBayer Schering Pharma Aktiengesellschaft
InventorsDirk Heimbach, Susanne Röhrig, Yolanda Cancho Grande, Eckhard Bender, Katja Zimmermann, Anja Buchmüller, Christoph Gerdes, Mark Jean Gnoth, Kersten Matthias Gericke, Mario Jeske
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Abstract
The invention relates to novel substituted piperidines, to processes for preparation thereof, to the use thereof for treatment and/or prophylaxis of diseases and to the use thereof for production of medicaments for treatment and/or prophylaxis of diseases, especially of cardiovascular diseases and tumour diseases.
Claims7
A compound of the formula
- in which
- R1 is trifluoromethyl, 1,1-difluoroethyl, 2,2-difluoroethyl, 2,2,2-trifluoroethyl, difluoromethoxy, trifluoromethoxy or ethyl,
- R2 is 2-hydroxyeth-1-yl, 2-methoxyeth-1-yl, 2-ethoxyeth-1-yl, cyclopropyl or 1-methoxycycloprop-1-yl,
- R3 is a group of the formula
- where
- * is the point of attachment to the carbonyl group,
- or a salt thereof.
4 more elements
Dependencies are inferred from the claim text.