US 2008/0167323 A1 · Substituted Triazole Derivatives as Oxytocin Antagonists

Abstract

The present invention relates to a class of substituted triazoles of formula (I) with activity as oxytocin antagonists, uses thereof, processes for the preparation thereof and compositions containing said inhibitors. These inhibitors have utility in a variety of therapeutic areas including sexual dysfunction, particularly premature ejaculation (P.E.).

Claims10

Dependent claims

A compound of formula (I)

or a tautomer thereof or a pharmaceutically acceptable salt or polymorph of said compound or tautomer or a prodrug thereof.

Dependencies are inferred from the claim text.

Facts

Application

11/909,290Filed 8 Mar 2006

Priority

21 Mar 2005

Published

10 Jul 2008

Term ends

Not estimatedThe source records don’t support an estimate.

Classification13 codes

C07D 401/14
Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a…:…
A61P 1/16
Drugs for disorders of the alimentary tract or the digestive system: for liver or gallbladder disorders, e.g. hepatoprotective agents,…
A61P 5/10
Drugs for disorders of the endocrine system: of the posterior pituitary hormones, e.g. oxytocin, ADH
A61P 9/04
Drugs for disorders of the cardiovascular system: inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure

Abstract

Claims10

Dependent claims

A compound of formula (I)

or a tautomer thereof or a pharmaceutically acceptable salt or polymorph of said compound or tautomer or a prodrug thereof.

Dependencies are inferred from the claim text.

Substituted Triazole Derivatives as Oxytocin Antagonists

Life of this patent

Abstract

Claims10

Substituted Triazole Derivatives as Oxytocin Antagonists

Life of this patent

Abstract

Claims10