Solid pharmaceutical preparation
AssigneeTakeda Pharaceutical Company Limited
InventorMasahiko Koike
Life of this patent
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Abstract
The present invention provides a solid preparation containing an insulin sensitizer and an active ingredient (except insulin sensitizers), which shows in vivo dissolution behavior of an insulin sensitizer, which is similar to the dissolution behavior of an insulin sensitizer from “a solid preparation containing an insulin sensitizer alone as an active ingredient”. The present invention provides a solid preparation containing (1) a layer containing an insulin sensitizer, and (2) a layer containing (a) an active ingredient (except insulin sensitizers), (b) microcrystalline cellulose having a mean particle size of 5-25 μm, (c) microcrystalline cellulose having a mean particle size of 30-100 μm and (d) polyvinylpyrrolidone K-90.
Claims12
A solid preparation comprising (1) a layer containing an insulin sensitizer and (2) a layer containing (a) an active ingredient (except insulin sensitizers), (b) microcrystalline cellulose having a mean particle size of 5-25 μm, (c) microcrystalline cellulose having a mean particle size of 30-100 μm and (d) polyvinylpyrrolidone K-90.
A solid preparation comprising (1) metformin or a salt thereof, (2) microcrystalline cellulose having a mean particle size of 5-25 μm and (3) microcrystalline cellulose having a mean particle size of 30-100 μm, wherein release of the metformin or a salt thereof is controlled.
Dependencies are inferred from the claim text.