Triazolopyrimidines
AssigneeBayer CropScience AG
InventorsOlaf Gebauer, Jorg Nico Greul, Ulrich Heinemann, Hans-Ludwig Elbe, Bernd-Wieland Kruger, Ralf Dunkel, Arnd Voerste
Life of this patent
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Abstract
Novel triazolopyrimidines of the formula 1 in which R1, R2, R3 and X have the meanings given in the description, and acid addition salts thereof, a plurality of processes for preparing these novel substances and their use for controlling unwanted microorganisms. Novel amines and carbamates of the formulae indicated in the description, and processes for preparing these intermediates.
Claims17
Triazolopyriridines of the formula
- 52
- in which
- R1 represents hydroxyl, amino, alkylcarbonylamino, N-alkyl-N-alkoxycarbonylamino, alkoxycarbonylamino, represents optionally substituted alkoxy, optionally substituted alkenyloxy, optionally substituted alkinyloxy, optionally substituted cycloalkyloxy, optionally substituted alkylamino, optionally substituted dialkylamino, optionally substituted alkenylamino, optionally substituted alkinylamino, optionally substituted cycloalkylamino, optionally substituted N-cycloalkyl-N-alkylamino, optionally substituted alkylideneamino, optionally substituted heterocyclyloxy or a radical of the formula —S—R4, in which
- R4 represents optionally substituted alkyl, optionally substituted alkenyl, optionally substituted alkinyl or optionally substituted cycloalkyl,
- R2 represents hydrogen, optionally substituted alkyl, optionally substituted alkenyl, optionally substituted alkinyl, or optionally substituted cycloalkyl,
- R3 represents optionally substituted aryl, and
- X represents halogen,
- and also acid addition salts of those compounds of the formula (I),
- in which
- R1 represents amino.
Amines of the formula
- 56
- in which
- R6 represents isobutyl, 2-methoxyethyl or represents
- 57
Amines of the formula
- 60
- in which
- R6 represents isobutyl, 2-methoxyethyl or represents
- 61
Trifluoroisopropylamines of the formula
- 64
- in which
- R7 represents methyl, ethyl or propyl.
3-Trifluoromethyl-3-amino-propene of the formula
- 67
Carbamates of the formula
- 69
- in which
- R6 represents isobutyl, 2-methoxyethyl or represents
- 70
Carbamates of the formula
- 71
- in which
- R6 represents isobutyl, 2-methoxyethyl or represents
- 72
Carbamates of the formula
- 73
- in which
- R7 represents methyl, ethyl or propyl.
Dependencies are inferred from the claim text.