Back to results
US 2004/0167101 A1Published application
Novel quinolinones and uses thereof
AssigneeARIAD Pharmaceuticals, Inc.
InventorsChester A. Metcalf III, William C. Shakespeare, Tomi K. Sawyer, Yihan Wang, Regine Bohacek, Rajeswari Sundaramoorthi
Life of this patent
Estimating the term…
Abstract
The invention relates to compounds of the general formula (and pharmaceutically acceptable derivatives thereof): 1 in which RA, RB, RC, RD, R5, R7, R9, R9a, AK, p, q, r and X are as defined herein, and to their preparation and use.
Claims6
A compound chosen from the following:
- 168 169 170
- wherein
- each occurence of Y is independently —O—, —S—, —NR1—, or a chemical bond linking R1 to P;
- each occurence of R1 is independently a substituted or unsubstituted aliphatic, heteroaliphatic, aryl or heteroaryl moiety, or, except in YR1 moieties in which Y is a covalent bond, R1 may also be H;
- and
- each alkyl and aryl group may be substituted or unsubstituted.
3 more elements
A compound chosen from the following:
- 171 172
A compound chosen from:
- 173 174
- wherein n is an integer from 0 to 6.
A compound chosen from the following:
- 175 176 177
- wherein each alkyl group may be substituted or unsubstituted.
A compound chosen from the following:
- 178 179
- wherein each alkyl group may be substituted or unsubstituted.
Dependencies are inferred from the claim text.