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US 2003/0171431 A1Published application
Intermediate and process for producing fluorinated carboxylic acid derivative from the same
AssigneeTaisho Pharmaceutical Co., Ltd.
InventorsAtsuro Nakazato, Toshihito Kumagai, Kazunari Sakagami, Takeo Taguchi
Life of this patent
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Abstract
The present invention relates to a 2-fluoro-2-(3-oxobicyclopentyl)acetate derivative represented by the formula (1): 1 The compound according to the present invention is useful for efficient syntheses of 2-amino-6-fluorobicyclo[3.1.0]hexane-2,6-dicarboxylic acids.
Claims4
A 2-fluoro-2-(3-oxocyclopentyl)acetate derivative represented by the formula (1):
- 11
- (wherein R1 is a C1-10 alkyl group, a C3-8 cycloalkyl group, a C3-8 cycloalkyl C1-6 alkyl group, an aryl group, an aryl C1-6 alkyl group, a C1-6 alkoxy C1-6 alkyl group, a C1-6 hydroxyalkyl group, a C1-6 alkylthio C1-6 alkyl group, a C1-6 mercaptoalkyl group, a tetrahydrofuranyl group, or a tetrahydropyranyl group;
- and X1 is a chlorine atom, a bromine atom, or an iodine atom).
Dependencies are inferred from the claim text.