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AssigneeBayer Aktiengesellschaft
InventorsPeter Jeschke, Martin Fuesslein, Hans-Georg Schwarz, Joachim Telser, Yolanda Cancho Grande, Alexander Arlt, Steffen Mueller, Ulrich Ebbinghaus-Kintscher, Peter Loesel, Marc Linka, Arunas Jonas Damijonaitis, Iring Heisler, Andreas Turberg, Oleksandr Mandzhulo
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The present invention relates to novel heteroaryl-triazole compounds of the general formula (I), in which the structural elements X, R1, R2, R3 and R4 have the meaning given in the description, to formulations and compositions comprising such compounds and for their use in the control of animal pests including arthropods and insects in plant protection and to their use for control of ectoparasites on animals.
A compound of formula (I) or an enantiomer thereof or a salt thereof
A compound selected from tert-butyl {1-[1˜ (6-cyanopyrimidin-4-yl)-1H-1,2,4-triazol-5-yl] ethyl}carbamate, tert-butyl N-[(IS)-1-[2-(6-cyanopyrimidin-4-yl)-1,2,4-triazol-3-yl] ethyl]carbamate, tert-butyl N-[(IS)-1-[2-(6-cyanopyrimidin-4-yl)-5-methyl-1,2,4-triazol-3-yl] ethyl] carbamate, tert-butyl N-[(IS)-1-[2-(6-cyanopyrimidin-4-yl)-5-cyclopropyl-1,2,4-triazol-3-yl] ethyl]-carbamate, tert-butyl N-[(1S)-1-[2-(6-carbamoylpyrimidin-4-yl)-5-cyclopropyl-1,2,4-triazol-3-yl] ethyl] carbamate, tert-butyl N-[(IS)-1-[5-cyclopropyl-2-[6-(methylcarbamoyl) pyrimidin-4-yl]-1,2,4-triazol-3-yl] ethyl] carbamate, and tert-butyl N-[(IS)-1-[5-cyclopropyl-2-[6-(dimethylcarbamoyl) pyrimidin-4-yl]-1,2,4-triazol-3-yl]ethyl]carbamate, or salts thereof.
A compound selected from 6-[5-(1-aminoethyl)-1H-1,2,4-triazol˜]-yl] pyrimidine-4-carbonitrile hydrochloride, 6-[5-[(1S)-1-aminoethyl]-1,2,4-triazol-1-yl] pyrimidine-4-carbonitrile, 6-[5-[(IS)-1-aminoethyl]-3-methyl-1,2,4-triazol-1-yl] pyrimidine-4-carbonitrile hydrochloride, 6-[5-[(IS)-1-aminoethyl]-3-cyclopropyl-1,2,4-triazol-1-yl] pyrimidine-4-carbonitrile hydro-chloride, 6-[5-[(IS)-1-aminoethyl]-3-methyl-1,2,4-triazol-1-yl] pyrimidine-4-carboxamide hydrochloride, 6-[5-[(1S)-1-aminoethyl]-3-cyclopropyl-1,2,4-triazol-1-yl] pyrimidine-4-carboxamide hydro-chloride, 6-[5-[(IS)-1-aminoethyl]-1,2,4-triazol-1-yl] pyrimidine-4-carboxamide hydrochloride, methyl 6-[5-[(IS)-1-(tert-butoxycarbonylamino) ethyl]-3-cyclopropyl-1,2,4-triazol-1-yl] pyrimidine-4-carboxylate, 6-[5-[(IS)-1-aminoethyl]-3-cyclopropyl-1,2,4-triazol-1-yl]-N-methyl-pyrimidine-4-carboxamide hydrochloride, 6-[5-[(1S)-1-aminoethyl]-3-cyclopropyl-1,2,4-triazol-1-yl]-N,N-dimethyl-pyrimidine-4-carboxamide hydrochloride, or salts thereof, or free amines thereof.
A compound selected from 2-chloro-6-(1-cyanocyclopropyl) pyridine-4-carboxylic acid, 3-(trifluoromethoxy)-S-(trifluoromethylsulfonyl) benzoic acid, 3-bromo-5-(2,2-dichlorocyclopropyl) benzoic acid 3-bromo-5-(1,1,2,2-tetrafluoroethoxy) benzoic acid, 3-(1-fluoro-1-methyl-ethyl)-5-(trifluoromethoxy) benzoic acid, or 3,5-bis(difluoromethylsulfonyl) benzoic acid, or salts thereof.
Dependencies are inferred from the claim text.