Back to results
US 11,958,810 B2Granted
Preparation of optionally substituted dihydroisoquinolines
AssigneeBASF SE
InventorsBernd Mueller, Michael Rack, Michael Seet, Ana Escribano Cuesta, Jan Klaas Lohmann, Georg Christoph Rudolf, Markus Nett, Rainer Hoffmann
Life of this patent
Estimating the term…
Abstract
Preparation of optionally substituted dihydroisoquinolines. The present invention relates to a process for the preparation of optionally substituted dihydroi-soquinolines of the formula I.
Claims10
A process for preparing a compound of formula I,
- wherein
- R3, R4 are independently selected from C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C1-C6-halogenalkyl, C2-C6-halogenalkenyl and C2-C6-halogenalkynl;
- R78 is independently selected from halogen, C1-C6-alkyl, C1-C6-alkoxy, C1-C6-halogenalkyl and C1-C6-halogenalkoxy;
- o is 0, 1, 2 or 3;
- Y is selected from C1-C6-alkyl, C1-C6-halogenalkyl, phenyl and benzyl, wherein phenyl and benzyl are unsubstituted or substituted by CN, NO2, halogen, C1-C6-halogenalkyl or C1-C6-alkoxy.
- comprising one step reaction of a compound of the formula II
- wherein R3, R4, o and R78 are as defined above with a compound of formula III
- wherein Y is as defined above.
5 more elements
Dependencies are inferred from the claim text.