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US 10,299,478 B2Granted
Pyrazolyltriazolylpyridines as pesticides
AssigneeBayer Animal Health GmbH
InventorsHans-Georg Schwarz, Werner Hallenbach, Ulrich Görgens, Kerstin Ilg, Andreas Turberg
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Abstract
The invention encompasses novel pyrazolyltriazolylpyridines of the general formula (I) in which the radicals A1-A4, W, Q, R1, R5 and Z1-Z3 have the meanings given in the description. Also described are processes for preparing the compounds of the formula (I). The compounds according to the invention are especially suitable for controlling insects and arachnids in agriculture, and ectoparasites in veterinary medicine.
Claims18
A compound of formula (I)
- in which
- R1 represents hydrogen, in each case optionally substituted C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C7-cycloalkyl, C3-C7-cycloalkyl-C1-C6-alkyl, C1-C6-alkylcarbonyl, C1-C6-alkoxycarbonyl, C1-C6-alkoxy-C1-C6-alkyl, aryl-C1-C6-alkyl, heteroaryl-C1-C6-alkyl;
- chemical moieties
- A1 represents CR2 or nitrogen,
- A2 represents nitrogen,
- A3 represents CR3 or nitrogen and
- A4 represents CR4 or nitrogen,
- but where not more than three of the chemical moieties A1 to A4 simultaneously represent nitrogen;
- R2, R3 and R4 independently of one another represent hydrogen, halogen, cyano, nitro, in each case optionally substituted C1-C6-alkyl, C3-C7-cycloalkyl, C1-C6-alkoxy, N—(C1-C6-alkoxy)imino-C1-C3-alkyl, C1-C6-alkylsulphanyl, C1-C6-alkylsulphinyl, C1-C6-alkylsulphonyl, N—(C1-C6-alkyl)amino, N,N-di(C1-C6-alkyl)amino, C1-C6-alkylsulphonylamino, or N—(C1-C6-alkyl)-C1-C6-alkylsulphonylamino;
- W represents oxygen or sulphur;
- Q represents hydrogen, formyl, hydroxy, amino or one of the in each case optionally substituted moieties C1-C6-alkyl, C1-C6-alkyloxy, C2-C6-alkenyl, C2-C6-alkynyl, C3-C7-cycloalkyl, hetero-C1-C6-cycloalkyl, C3-C6-cycloalkyl-C1-C6-alkyl, aryl-C1-C6-alkyl, heteroaryl-C1-C6-alkyl or represents a moiety N—(C1-C6-alkyl)amino, N—(C1-C6-alkylcarbonyl)amino, N,N-di(C1-C6-alkyl)amino;
- or
- Q represents an unsaturated 6-membered carbocycle which is optionally polysubstituted by V or represents an unsaturated 5- or 6-membered heterocyclic ring which is optionally polysubstituted by V, where
- V represents halogen, cyano, nitro, or one of the moieties C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C7-cycloalkyl, C1-C6-alkoxy, N—(C1-C6-alkoxy)imino-C1-C6-alkyl, C1-C6-alkylsulphanyl, C1-C6-alkylsulphinyl, C1-C6-alkylsulphonyl, N—(C1-C6-alkyl)amino or N,N-di(C1-C6-alkyl)amino, each of which is optionally substituted;
- R5 independently of one another represent hydrogen, halogen, cyano, nitro, amino, in each case optionally substituted C1-C6-alkyl, C1-C6-alkyloxy, C1-C6-alkylcarbonyl, C1-C6-alkylsulphanyl, C1-C6-alkylsulphinyl, C1-C6-alkylsulphonyl, N—(C1-C6)-alkylamino or N,N-di(C1-C6-alkyl)amino;
- Z1 represents optionally substituted C1-C6-alkyl;
- Z2 represents hydrogen, halogen, cyano, nitro or in each case optionally substituted C1-C6-alkyl, C1-C6-alkylcarbonyl, C1-C6-alkylsulphanyl, C1-C6-alkylsulphinyl, C1-C6-alkylsulphonyl;
- and
- Z3 represents hydrogen or in each case optionally substituted C1-C6-alkyl, C3-C7-cycloalkyl, C3-C6-alkenyl, C3-C6-alkynyl, aryl or hetaryl.
16 more elements
Dependencies are inferred from the claim text.