Therapeutic compounds and uses thereof
AssigneesGenetech, Inc., Constellation Pharmaceuticals, Inc.
InventorsBrian K. Albrecht, Daniel J. Burdick, Alexandre Cote, Martin Duplessis, Christopher G. Nasveschuk, Alexander M. Taylor
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Abstract
The invention relates to compounds of formula (I) and salts thereof: wherein R1-R3 have any of the values defined in the specification. The compounds and salts are useful for treating PCAF mediated disorders and/or GCN5 mediated disorders. The invention also provides pharmaceutical compositions comprising a compound of formula (I), or a pharmaceutically acceptable salt thereof, as well as and methods of using said compounds, salts, or compositions in the treatment of various disorders.
Claims7
A compound of formula (I), or a salt thereof:
- wherein:
- R1 is selected from the group consisting of methyl, chloro, and bromo;
- R2 is C1-4 alkyl, C2-4 alkenyl, cyclopropyl, or cyclopropylmethyl;
- and
- R3 is selected from the group consisting of:
Dependencies are inferred from the claim text.